Profile: Activate Scientific GmbH specializes in multifunctional heterocylic synthons, scaffolds and boronic acids. We produce and distribute novel reactive intermediates, exclusive building blocks (Exclusive Blocks™) and series of synthons for drug discovery. We provide boronic acids such as alkylboronic acids, arylboronic acids, borontrifluorides, heterocyclic boronic and vinyl boronic acids. Our products include alicyclic, azepines, azetidines, aromatics, bridged compounds, chromans, dioxoles and furans.
| • Allylboronic acid piracol ester
IUPAC Name: 4,4,5,5-tetramethyl-2-prop-2-enyl-1,3,2-dioxaborolane | CAS Registry Number: 72824-04-5 Synonyms: Pinacol allylboronate, Allylboronic acid pinacol ester, 324647_ALDRICH, Allylboronic acid pinacol cyclic ester, A1135G1, ST5408244, 2-Allyl-4,4,5,5-tetramethyl-1,3,2-dioxaborolane
InChIKey: YMHIEPNFCBNQQU-UHFFFAOYSA-N | ||||||||
| • Amifampridine
IUPAC Name: pyridine-3,4-diamine | CAS Registry Number: 54-96-6 Synonyms: 3,4-Pyridinediamine, 3,4-DIAMINOPYRIDINE, Diamino-3,4 pyridine, 4,5-Diaminopyridine, Pyridine, 3,4-diamino-, pyridine-3,4-diamine, 3,4 Diaminopyridine, 3-amino-4-pyridinylamine, WLN: T6NJ CZ DZ, SC10, MLS001304911, MLS001333181, MLS001333182, 3,4-Pyridinediamine (9CI), D7148_SIGMA, EINECS 200-220-9, 3,4-DAP, NSC 521760, ALBB-005969, BRN 0110232
InChIKey: OYTKINVCDFNREN-UHFFFAOYSA-N | ||||||||
| • Azetidine-3-ylmethyl-carbamic Acid Tert-butyl Ester
IUPAC Name: tert-butyl N-(azetidin-3-ylmethyl)carbamate | CAS Registry Number: 91188-15-7 Synonyms: 3-Boc-aminomethylazetidine, 3-(n-boc-aminomethyl)azetidine, 3-(boc-aminomethyl)azetidine, tert-butyl N-(azetidin-3-ylmethyl)carbamate, 3-boc-aminomethyl-azetidine, tert-butyl azetidin-3-ylmethylcarbamate, 3-(n-boc)aminomethylazetidine, tert-butylazetidin-3-ylmethylcarbamate, AG-H-74115, tert-butyl [(azetidin-3-yl)methyl]carbamate, azetidine-3-ylmethyl-carbamic acid tert-butyl ester, CARBAMIC ACID, N-(3-AZETIDINYLMETHYL)-, 1,1-DIMETHYLETHYL ESTER, 3-{[(tert-Butoxycarbonyl)amino]methyl}azetidine, 3-[[(TERT-BUTOXYCARBONYL)AMINO]METHYL]AZETIDINE, PubChem10158, AC1Q1NEP, AGN-PC-00OYUH, SureCN1034818, CTK3I6612, azetidin-3-yl(neopentyl)carbamate
InChIKey: MOLUHRBHXXGWDP-UHFFFAOYSA-N | ||||||||
| • Beaucage reagent
IUPAC Name: 1,1-dioxobenzo[c]dithiol-3-one | CAS Registry Number: 66304-01-6 Synonyms: B1027_SIGMA, AIDS211144, AIDS-211144, ZINC00389835, CID3009847, 3H-1,2-Benzodithiol-3-one 1,1-dioxide, 3H-1,2-Benzodithiol-3-one, 1,1-dioxide
InChIKey: JUDOLRSMWHVKGX-UHFFFAOYSA-N | ||||||||
| • Benzenamine, 3-fluoro-4-(4-methyl-1H-imidazol-1-yl)-
IUPAC Name: 3-fluoro-4-(4-methylimidazol-1-yl)aniline | CAS Registry Number: 252340-70-8 Synonyms: 3-FLUORO-4-(4-METHYL-1H-IMIDAZOL-1-YL)BENZENAMINE, PubChem8281, SureCN1616928, CTK3J8351, MolPort-000-140-293, ANW-57886, AKOS005258734, AG-E-76714, AK-29937, EN000364, KB-70773, 3-Fluoro-4-(4-methylimidazole)benzenamine, AB1006559, 3-fluoro-4-(4-methyl-1-imidazolyl)aniline, 3-fluoranyl-4-(4-methylimidazol-1-yl)aniline, B-1777, 3-fluoro-4-(4-methyl-1H-imidazol-1-yl)aniline, A817724, I14-11320, [3-Fluoro-4-(4-methylimidazol-1-yl)phenyl]amine;3-Fluoro-4-(4-methyl-1H-imidazol-1-yl)aniline;3-Fluoro-4-(4-methyl-imidazol-1-yl)-phenylamine;
InChIKey: XUDKNXYCYIYBIG-UHFFFAOYSA-N | ||||||||
| • Benzeneboronic acid, m-carboxy-
IUPAC Name: 3-boronobenzoic acid | CAS Registry Number: 25487-66-5 Synonyms: 3-Boronobenzoic acid, 3-Carboxyphenylboronic acid, 456764_ALDRICH, ALBB-006101, FS000841, ST5405809, TL8002069
InChIKey: DBVFWZMQJQMJCB-UHFFFAOYSA-N | ||||||||
| • Carbamic acid, [2-(3-azetidinyl)ethyl]-, 1,1-dimethylethyl ester
IUPAC Name: tert-butyl N-[2-(azetidin-3-yl)ethyl]carbamate | CAS Registry Number: 162696-31-3 Synonyms: 3-Boc-aminoethylazetidine, tert-butyl 2-(azetidin-3-yl)ethylcarbamate, 3-(N-Boc-Aminoethyl)azetidine, tert-butyl N-[2-(azetidin-3-yl)ethyl]carbamate, CARBAMIC ACID, N-[2-(3-AZETIDINYL)ETHYL]-, 1,1-DIMETHYLETHYL ESTER, SureCN5969026, CTK7G9279, MolPort-000-140-286, AKOS005258722, 3-(2-BOC-AMINOETHYL)AZETIDINE, AG-C-78717, AM81152, PB32810, RP04257, 3-(2-N-BOC-AMINOETHYL)AZETIDINE, AK-29911, 3-(N-BOC)-(2-AMINOETHYL)AZETIDINE, AB1006554, 2-(AZETIN-3-YL)-1-(N-BOC)ETHYLAMINE, A26668
InChIKey: CSPJUZSNJFANNU-UHFFFAOYSA-N | ||||||||
| • Carbamic acid, methyl(3R)-3-piperidinyl-, 1,1-dimethylethyl ester (9CI)
IUPAC Name: tert-butyl N-methyl-N-[(3R)-piperidin-3-yl]carbamate | CAS Registry Number: 309962-67-2 Synonyms: (R)-TERT-BUTYL METHYL(PIPERIDIN-3-YL)CARBAMATE, Methyl-(R)-piperidin-3-yl-carbamic acid tert-butyl ester, (R)-3-N-Boc-3-(Methylamino)piperidine, SureCN1267151, CTK3J6570, R-3-Boc-3-methylaminopiperidine, MolPort-000-140-272, (R)-3-Boc-3-methylaminopiperidine, ANW-49069, AKOS007930615, R-3-N-Boc-3-(Methylamino)piperidine, AG-F-02863, AM90337, PB23729, AK-29124, BR-29124, KB-54910, AB1006535, FT-0648176, W5318
InChIKey: RTXNDTNDOHQMTI-SECBINFHSA-N | ||||||||
| • Carbamic acid, methyl(3S)-3-piperidinyl-, 1,1-dimethylethyl ester
IUPAC Name: tert-butyl N-methyl-N-[(3S)-piperidin-3-yl]carbamate | CAS Registry Number: 309962-63-8 Synonyms: (S)-tert-Butyl methyl(piperidin-3-yl)carbamate, (S)-3-N-Boc-3-(methylamino)piperidine, (S)-3-Boc-3-methylaminopiperidine, Methyl-(S)-piperidin-3-yl-carbamic acid tert-butyl ester, SureCN2521256, CTK4G6259, S-3-Boc-3-methylaminopiperidine, MolPort-000-140-273, ANW-52346, AKOS007930616, AKOS015899804, AG-F-02862, AM90336, PB32805, AK-29123, BR-29123, KB-54917, AB1006536, FT-0648175, W5317
InChIKey: RTXNDTNDOHQMTI-VIFPVBQESA-N | ||||||||
| • Diisopropyl Squarate
IUPAC Name: 3,4-di(propan-2-yloxy)cyclobut-3-ene-1,2-dione | CAS Registry Number: 61699-62-5 Synonyms: Diisopropyl squarate, 338230_ALDRICH, 3,4-Diisopropoxy-3-cyclobutene-1,2-dione, MolPort-000-139-713, CID182314, ZINC02545328, D2840G1, D2207
InChIKey: KCZPGGVPQXQGEJ-UHFFFAOYSA-N | ||||||||
| • Dipicolinic Acid
IUPAC Name: pyridine-2,6-dicarboxylic acid | CAS Registry Number: 499-83-2 Synonyms: Dipicolinic acid, Dipicolinate, 2,6-Pyridinedicarboxylic acid, 2,6-Dipicolinic acid, zinc dipicolinate, 2,6-Dicarboxypyridine, DPAC, PYRIDINE-2,6-DICARBOXYLIC ACID, pyridine carboxylate, 6d, 2,6-pyridinedicarboxylate, Oprea1_533632, C7H5NO4, P63808_ALDRICH, MLS000080748, NSC 176, ARONIS021542, IFLab1_001781, NSC176, 02321_FLUKA, CHEBI:46837
InChIKey: WJJMNDUMQPNECX-UHFFFAOYSA-N | ||||||||
| • α-Pyridone
IUPAC Name: 1H-pyridin-2-one | CAS Registry Number: 142-08-5 Synonyms: 2-Pyridinol, 2-Pyridone, 2-HYDROXYPYRIDINE, 2(1H)-Pyridinone, 2-Oxopyridine, 2-Pyridinone, alpha-Pyridone, Pyridin-2-ol, 2(1H)-Pyridone, .alpha.-Pyridone, Pyridinol, 2(lH)-Pyridinone, Pyridone-2 [French], pyridin-2(1H)-one, H56800_ALDRICH, 56380_FLUKA, CHEBI:16540, EINECS 205-520-3, NSC172522, AIDS081857
InChIKey: UBQKCCHYAOITMY-UHFFFAOYSA-N | ||||||||
| • Imidazo[1,2-A]pyrazine, 5,6,7,8-Tetrahydro-2-(trifluoromethyl)-
IUPAC Name: 2-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazine | CAS Registry Number: 126069-70-3 Synonyms: 2-(Trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazine, 2-(trifluoromethyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine, IMIDAZO[1,2-A]PYRAZINE, 5,6,7,8-TETRAHYDRO-2-(TRIFLUOROMETHYL)-, PubChem17803, AC1Q4JFG, SureCN108034, AGN-PC-0028GK, MolPort-002-680-136, ANW-52018, AKOS005255469, AB53003, QC-8387, AK-24652, BR-24652, KB-16051, AM20080198, S14-1822, I14-15761, I14-32749, 2-(Trifluoromethyl)-5,6,7,8-tetrahydroimidazo-[1,2-a]pyrazine
InChIKey: RHYZIHOBSWRZDL-UHFFFAOYSA-N | ||||||||
| • Isoquinoline-1-Carboxylic Acid
IUPAC Name: isoquinoline-1-carboxylic acid | CAS Registry Number: 486-73-7 Synonyms: 1-Isoquinolinecarboxylic acid, Isoquinoline-1-carboxylic acid, 150134_ALDRICH, 58752_FLUKA, ALBB-005987, EINECS 207-639-6, NSC218351, AI3-61946, ST5308467
InChIKey: XAAKCCMYRKZRAK-UHFFFAOYSA-N | ||||||||
| • Lomefloxacin (3-Aminopyrazole)
IUPAC Name: 1H-pyrazol-5-amine | CAS Registry Number: 1820-80-0 Synonyms: 3-Aminopyrazole, 3-Pyrazolamine, 1H-Pyrazol-3-amine, Pyrazol-3-ylamine, 3-Amino-1H-pyrazole, 160644_ALDRICH, ALBB-004467, NSC76122, EINECS 217-338-1, NSC 76122, SBB004401, STK292780, ZINC04674340, FS000814, TL8001457, InChI=1/C3H5N3/c4-3-1-2-5-6-3/h1-2H,(H3,4,5,6
InChIKey: JVVRJMXHNUAPHW-UHFFFAOYSA-N | ||||||||
| • Methyl 3-Oxocyclopentanecarboxylate
IUPAC Name: methyl 3-oxocyclopentane-1-carboxylate | CAS Registry Number: 32811-75-9 Synonyms: Methyl 3-oxocyclopentanecarboxylate, NSC41335, CID237640, O3033M500, Cyclopentanecarboxylic acid, 3-oxo-, methyl ester
InChIKey: KTGCFXSELRVRFH-UHFFFAOYSA-N | ||||||||
| • N-(5-Methyl-2-Pyridyl)acetamide
IUPAC Name: N-(5-methylpyridin-2-yl)acetamide | CAS Registry Number: 4931-47-9 Synonyms: ZINC00334302, N-(5-methylpyridin-2-yl)acetamide, CID818995, AI-942/25034577
InChIKey: ARHIRVVLQAQUCO-UHFFFAOYSA-N | ||||||||
| • N-Boc-3-hydroxyazetidine
IUPAC Name: tert-butyl 3-hydroxyazetidine-1-carboxylate | CAS Registry Number: 141699-55-0 Synonyms: ZINC02527471, ALBB-009728, 1-BOC-3-(HYDROXY)AZETIDINE, CID2756801, FS011275, tert-butyl 3-hydroxyazetidine-1-carboxylate, TL8000922
InChIKey: XRRXRQJQQKMFBC-UHFFFAOYSA-N | ||||||||
| • N-BOC-pyrrole-2-boronic Acid
IUPAC Name: [1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrol-2-yl]boronic acid | CAS Registry Number: 135884-31-0 Synonyms: N-Boc-2-pyrroleboronic acid, N-Boc-2-pyrryl boronic acid, N-Boc-pyrrole-2-boronic acid, 15047_FLUKA, B2016G1, TL8007173, 1-(T-Butoxycarbonyl)Pyrrole-2-Boronic Acid
InChIKey: ZWGMJLNXIVRFRJ-UHFFFAOYSA-N | ||||||||
| • Ortho phenylPhenol
IUPAC Name: 2-phenylphenol | CAS Registry Number: 90-43-7 Synonyms: 2-Phenylphenol, 2-Hydroxybiphenyl, o-Hydroxybiphenyl, Biphenyl-2-ol, 2-Biphenylol, o-Hydroxydiphenyl, Orthoxenol, 2-Hydroxydiphenyl, Torsite, o-Diphenylol, O-PHENYLPHENOL, Phenylphenol, Biphenylol, o-Biphenylol, Dowicide 1, Hydroxdiphenyl, Nectryl, Topane, o-Xenol, o-Xonal
InChIKey: LLEMOWNGBBNAJR-UHFFFAOYSA-N | ||||||||
| • Phenethylboronic acid
IUPAC Name: 2-phenylethylboronic acid | CAS Registry Number: 34420-17-2 Synonyms: Phenylethane boronic acid, PEBA, 2-phenylethylboronic acid, Alkylboronic Acid, 21, 588423_ALDRICH, Boronic acid, (2-phenylethyl)-, BM536, DB01963, TL8007138, PBA
InChIKey: VPRUMANMDWQMNF-UHFFFAOYSA-N | ||||||||
| • Piperazine, 1-(4-piperidinyl)-
IUPAC Name: 1-piperidin-4-ylpiperazine | CAS Registry Number: 142013-66-9 Synonyms: 1-(piperidin-4-yl)piperazine, 4-Piperazine-piperidine, 4-Piperazine-piperidine 3HCl, SureCN336575, AGN-PC-00P2WS, SureCN1400974, KSC491G1F, CHEMBL76508, 1-(4-Piperidinyl)-piperazine, MolPort-000-140-280, 1-PIPERIDIN-4-YLPIPERAZINE, ACT02126, ANW-75381, AKOS010951412, AK-81377, KB-40305, AB1006546, AM20080318, FT-0645810, W3094
InChIKey: ZHYYBDZASCMDMP-UHFFFAOYSA-N | ||||||||
| • Piperazinone, 1,5-diethyl-, (S)-
IUPAC Name: (5S)-1,5-diethylpiperazin-2-one | CAS Registry Number: 106576-36-7 Synonyms: Piperazinone, 1,5-diethyl-, (S), (S)-1,5-DIETHYLPIPERAZINONE, (S)-1,5-Diethyl-piperazin-2-one, CTK0H3746, Piperazinone,1,5-diethyl-,(S), AKOS006312671, AKOS015838644, AG-D-21091, AK-32774, KB-80034, AB1006565, B-1472, I14-0684, (5S)-1,5-Diethylpiperazin-2-one;2-Piperazinone, 1,5-diethyl-, (5S)-;(S)-1,5-Diethylpiperazin-2-one;Piperazinone,1,5-diethyl-, (S)- (9CI);(S)-Piperazinone,1,5-diethyl;MFCD09878610;, (S)-1,5-Diethyl-Piperazinone; (S)-1,5-Diethylpiperizin-2-one; (5S)-1,5-Diethylpiperizin-2-one; (S)-Piperazinone,1,5-diethyl
InChIKey: IYZRHXDFJURKOL-ZETCQYMHSA-N | ||||||||
| • Piperazinone, 1-ethyl-5-(2-methylpropyl)-, (S)- (9CI)
IUPAC Name: (5S)-1-ethyl-5-(2-methylpropyl)piperazin-2-one | CAS Registry Number: 106576-32-3 Synonyms: (S)-1-ETHYL-5-ISOBUTYLPIPERAZIN-2-ONE, Piperazinone,1-ethyl-5-(2-methylpropyl)-, (S)- (9CI), CTK4A4642, AKOS006313912, AKOS015838643, AG-D-21090, KB-63445, AB1006570, (5S)-1-ethyl-5-(2-methylpropyl)-2-piperazinone, (5S)-1-ethyl-5-(2-methylpropyl)piperazin-2-one, A801466, I14-36810, (S)-1-Ethyl-5-(2-methylpropyl)-Piperazinone (9CI); (5S)-1-Ethyl-5-(2-Methylpropyl)piperizin-2-one
InChIKey: IIPNMKFGSRIZEK-VIFPVBQESA-N | ||||||||
| • Pyridine-2,6-Dimethanol
IUPAC Name: [6-(hydroxymethyl)pyridin-2-yl]methanol | CAS Registry Number: 1195-59-1 Synonyms: 2,6-Pyridinedimethanol, Pyridine-2,6-diyldimethanol, Oprea1_777136, 2,6-Bis-(hydroxymethyl)pyridine, 154369_ALDRICH, 2,6-Bis(hydroxymethyl)pyridine, NSC16571, EINECS 214-803-0, STK298894, ZINC00155372, P153, TL8000523, InChI=1/C7H9NO2/c9-4-6-2-1-3-7(5-10)8-6/h1-3,9-10H,4-5H
InChIKey: WWFMINHWJYHXHF-UHFFFAOYSA-N | ||||||||
| • Pyridine-2-Boronic Acid, Pinacol Ester
IUPAC Name: 2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine | CAS Registry Number: 791819-02-8 Synonyms: STK503732, ALBB-006131, Pyridine-2-boronic acid pinacol ester, P2451G1, CID11241171, 2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine, 874186-98-8
InChIKey: SOQIDYYUSMPIDR-UHFFFAOYSA-N | ||||||||
| • Pyrimido[5,4-d]pyrimidine, 2,8-dichloro-
IUPAC Name: 4,6-dichloropyrimido[5,4-d]pyrimidine | CAS Registry Number: 189747-34-0 Synonyms: 2,8-DICHLOROPYRIMIDO[5,4-D]PYRIMIDINE, AG-E-38529, PubChem14850, CTK4E0206, MolPort-000-140-430, ANW-66710, ZINC34415167, AKOS015907647, AB51062, QC-9235, RP25820, 4,6-dichloropyrimido[5,4-d]pyrimidine, AK-27444, KB-18522, Pyrimido[5,4-d]pyrimidine,2,8-dichloro-, FT-0645576, ST51054834, 4,6-bis(chloranyl)pyrimido[5,4-d]pyrimidine, A813351, 2,8-DICHLOROPYRIMIDO[5,4-D][1,3]DIAZINE
InChIKey: FVNFFJZCBGWGDZ-UHFFFAOYSA-N | ||||||||
| • Pyrrolidin-3-ylmethyl-carbamic Acid Tert-butyl Ester
IUPAC Name: tert-butyl N-(pyrrolidin-3-ylmethyl)carbamate | CAS Registry Number: 149366-79-0 Synonyms: 3-Boc-aminomethylpyrrolidine, 3-Boc-aminomethyl-pyrrolidine, 3-Bocaminomethylpyrrolidine, Tert-butyl N-(pyrrolidin-3-ylmethyl)carbamate, 3-N-Boc-Aminomethyl pyrrolidine, Pyrrolidin-3-ylmethyl-carbamic acid tert-butyl ester, 3-(Boc-Aminomethyl)pyrrolidine, AC1Q1NEM, SureCN622379, AC1N5WW3, Ambcb4036831, Jsp002830, CTK7G9248, MolPort-000-001-701, AKOS005258682, AC-2227, AG-C-19102, MCULE-8885203488, PB15798, RP04255
InChIKey: WIEJVMZWPIUWHO-UHFFFAOYSA-N | ||||||||
| • Risperidone Chloride HCL
IUPAC Name: 3-(2-chloroethyl)-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one | CAS Registry Number: 63234-80-0 Synonyms: 3-(2-chloroethyl)-6,7,8,9-tetrahydro-2-methyl-4h-pyrido[1,2-a]pyrimidin-4-one, 3-(2-chloroethyl)-2-methyl-6,7,8,9-tetrahydro-4h-pyrido[1,2-a]pyrimidin-4-one, 3-(2-chloroethyl)-6,7,8,9-tetrahydro-2-methyl-4H-pyrido(1,2a)pyrimidine-4-one, 3-(2-Chloro-ethyl)-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one, 3-2(2-Chloroethyl)-6,7,8,9-tetrahydro-2-methyl-4H-Pyrido[1,2-a]Pyrimdin-4-one, 3-(2-chloroethyl)-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one, 3-(2-chloroethyl)-2-methyl-6,7,8,9-tetrahydro-4h-pyridino(1,2-a)-pyrimidine-4-one, 3-(2-chloroethyl)-6,7,8,9-tetrahydro-2-methyl-4h-pyridino[1,2-a]pyrimidine-4-one, 3-(2-chloroethyl)-6,7,8,9-tetrahydro-2-methyl-4h-pyrido(1,2-a)pyrimidin-4-one, 3-(2-chloroethyl)-2-methyl-6,7,8,9-tetrahydro-4h-pyrido(1,2-a)pyrimidin-4-one, 4H-Pyrido(1,2-a)pyrimidin-4-one, 3-(2-chloroethyl)-6,7,8,9-tetrahydro-2-methyl-, 4H-PYRIDO[1,2-A]PYRIMIDIN-4-ONE, 3-(2-CHLOROETHYL)-6,7,8,9-TETRAHYDRO-2-METHYL-, PubChem20773, AC1MC7SG, ACMC-209ne8, SureCN460865, UNII-2089CR1AQN, Risperidone impurity L [EP], RISPERIDONE INTERMEDIATE, Piperidopyrimidinone intermediate
InChIKey: CMWCQQUYLPYOMY-UHFFFAOYSA-N | ||||||||
| • Squaric Acid
IUPAC Name: 3,4-dihydroxycyclobut-3-ene-1,2-dione | CAS Registry Number: 2892-51-5 Synonyms: Squaric acid, Quadratic acid, Cyclobutenedione, dihydroxy-, Dihydroxycyclobutenedione, 3,4-Dihydroxy-3-cyclobutene-1,2-dione, CCRIS 6793, WLN: L4VVTJ CQ DQ, 3-Cyclobutene-1,2-dione, 3,4-dihydroxy-, 1,2-Dihydroxycyclobutene-3,4-dione, 1,2-Diketo-3,4-dihydroxycyclobutene, 123447_ALDRICH, 3,4-Dihydroxy-cyclobutene-1,2-dione, EINECS 220-761-4, NSC624671, AIDS160322, NSC 125692, AIDS-160322, BRN 0774275, Cyclobutenedione, dihydroxy- (8CI), NSC125692
InChIKey: PWEBUXCTKOWPCW-UHFFFAOYSA-N | ||||||||
| • Tert-Butyl 3-Oxoazetidine-1-Carboxylate
IUPAC Name: tert-butyl 3-oxoazetidine-1-carboxylate | CAS Registry Number: 398489-26-4 Synonyms: 1-Boc-3-azetidinone, 1-Boc-azetidin-3-one, C-3186K, TL8002873
InChIKey: VMKIXWAFFVLJCK-UHFFFAOYSA-N | ||||||||
| • (1,3-Dimethyl-1H-pyrazol-5-yl)methanol
IUPAC Name: (2,5-dimethylpyrazol-3-yl)methanol | CAS Registry Number: 57012-20-1 Synonyms: ZINC00158736, CID2776363, CC 12509, H09018
InChIKey: GUJDKMVLHCJODO-UHFFFAOYSA-N | ||||||||
| • (1,3-Dimethyl-1H-Pyrazol-5-Yl)methylamine
IUPAC Name: (2,5-dimethylpyrazol-3-yl)methanamine | CAS Registry Number: 499770-63-7 Synonyms: STK349283, (2,5-dimethylpyrazol-3-yl)methanamine, CC12513, CID1257670, (1,3-Dimethyl-1H-pyrazol-5-yl)methanamine, 1-(1,3-dimethyl-1H-pyrazol-5-yl)methanamine, H09019
InChIKey: DAOWQCXPMWGSBW-UHFFFAOYSA-N | ||||||||
| • (2-Ethoxycarbonylphenyl)boronic acid
IUPAC Name: (2-ethoxycarbonylphenyl)boronic acid | CAS Registry Number: 380430-53-5 Synonyms: 2-Ethoxycarbonylphenylboronic acid, BM200
InChIKey: QZKVVOXAEBCLPZ-UHFFFAOYSA-N | ||||||||
| • (2-Methylthio)phenylboronic Acid
IUPAC Name: (2-methylsulfanylphenyl)boronic acid | CAS Registry Number: 168618-42-6 Synonyms: 2-(Methylthio)phenylboronic acid, 2-Methylthiophenylboronic acid, 521248_ALDRICH, BM209, ST5408309, TL8001305
InChIKey: QXBWTYBCNFKURT-UHFFFAOYSA-N | ||||||||
| • (2R,4S)-4-fluoropyrrolidine-2-carboxylic acid
IUPAC Name: (2R,4S)-4-fluoropyrrolidine-2-carboxylic acid | CAS Registry Number: 131176-02-8 Synonyms: AG-D-63262, D-Proline, 4-fluoro-,(4S)-, 4-Fluoro-pyrrolidine-2-carboxylic acid, AC1ODYYA, trans-4-Fluoro-D-proline, SureCN900297, Jsp001877, CTK4B7124, MolPort-000-140-560, ANW-56554, AKOS005063934, AC-2248, RP20042, AK-29824, KB-01285, U345, TL8000738, FT-0601716, B-1564, I11-0112
InChIKey: ZIWHMENIDGOELV-IUYQGCFVSA-N | ||||||||
| • (2S,4R)-4-Fluoropyrrolidine-2-carboxylic acid
IUPAC Name: (2S,4R)-4-fluoropyrrolidine-2-carboxylic acid | CAS Registry Number: 21156-44-5 Synonyms: (2S,4R)-4-fluoropyrrolidine-2-carboxylic acid, trans-4-Fluoro-l-proline, 2507-61-1, (2S, 4R)-4-Fluoroproline, SBB066761, AG-E-55212, PubChem18392, SureCN305909, AC1Q71AA, TRANS-4-FLUOROPROLINE, R-4-FLUORO-L-PROLINE, Jsp004327, TRANS H-PRO(4-F)-OH, CHEMBL1232810, CTK4E5982, H-TRANS-4-FLUORO-PRO-OH, TRANS-4-FLUORO-L-PRO-OH, (4R)-4-FLUOR-L-PROLIN, MolPort-000-140-558, Proline, 4-fluoro-,trans- (8CI)
InChIKey: ZIWHMENIDGOELV-DMTCNVIQSA-N | ||||||||
| • (2S,4S)-4-Fluoropyrrolidine-2-carboxylic acid
IUPAC Name: (2S,4S)-4-fluoropyrrolidine-2-carboxylic acid | CAS Registry Number: 6745-32-0 Synonyms: (2S,4S)-4-fluoropyrrolidine-2-carboxylic acid, cis-4-Fluoroproline, cis-4-Fluoro-L-proline, 2438-57-5, AG-G-55024, (2S,4S)-4-fluoro-2-pyrrolidinecarboxylic acid, (2S,4S)-4-fluoranylpyrrolidine-2-carboxylic acid, 4-Fluoro-pyrrolidine-2-carboxylic acid, PubChem18395, SureCN661917, AC1Q71AC, S-4-FLUORO-L-PROLINE, H-CIS-PRO(4-F)-OH, L-Proline, 4-fluoro-, cis-, CIS-4-FLUORO-L-PRO-OH, H-CIS-4-FLUORO-PRO-OH, CTK5C6182, (4S)-4-FLUOR-L-PROLIN, MolPort-000-140-559, (2S,4S)-4-FLUOROPROLINE
InChIKey: ZIWHMENIDGOELV-IMJSIDKUSA-N | ||||||||
| • (3-Aminomethylphenyl)boronic acid hydrochloride
IUPAC Name: [3-(aminomethyl)phenyl]boronic acid hydrochloride | CAS Registry Number: 352525-94-1 Synonyms: A1260G1, 3-Aminomethylphenylboronic acid hydrochloride
InChIKey: NPTBTFRGCBFYPZ-UHFFFAOYSA-N | ||||||||
| • (3-Boc-aminophenyl)bronoic acid
IUPAC Name: [3-(butoxycarbonylamino)phenyl]boronic acid | CAS Registry Number: 380430-68-2 Synonyms: 3-Butoxycarbonylaminophenylboronic acid
InChIKey: XESUEUMDUBPYNR-UHFFFAOYSA-N | ||||||||
| • (3-Bromomethylphenyl)boronic acid neopentyl glycol ester
IUPAC Name: 2-[3-(bromomethyl)phenyl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane | CAS Registry Number: 143805-78-1 Synonyms: B1862G1, (3-Bromomethylphenyl)boronic acid pinacol ester
InChIKey: WUIYGXGXVOHAFW-UHFFFAOYSA-N | ||||||||
| • (3-Formyl-1-indolyl)acetic acid
IUPAC Name: 2-(3-formylindol-1-yl)acetate | CAS Registry Number: 138423-98-0 Synonyms: ZINC00254469, CID3544186
InChIKey: ZUUGBTJTGRTIFK-UHFFFAOYSA-M | ||||||||
| • (4-Aminophenyl)piperidin-1-ylmethanone
IUPAC Name: (4-aminophenyl)-piperidin-1-ylmethanone | CAS Registry Number: 42837-37-6 Synonyms: nchembio.87-comp30, TimTec1_002611, Oprea1_328484, Oprea1_777979, ARONIS015991, 4-(1-Piperidinylcarbonyl)aniline, MolPort-000-140-746, 4-(piperidin-1-ylcarbonyl)aniline, Piperidine, 1-(4-aminobenzoyl)-, ALBB-000064, (4-Amino-phenyl)-piperidin-1-yl-methanone, CID577812, STK299342, ZINC00045801, BAS 03421360, 4-(piperidin-1-ylcarbonyl)phenylamine, BBV-026093, NCGC00173934-01, (4-aminophenyl)(piperidin-1-yl)methanone, EU-0067488
InChIKey: FQEGZNLIOFLYNI-UHFFFAOYSA-N | ||||||||
| • (6-Methyl-Pyridin-2-Yl)-Carbamic Acid Tert-Butyl Ester
IUPAC Name: tert-butyl N-(6-methylpyridin-2-yl)carbamate | CAS Registry Number: 205676-84-2 Synonyms: tert-Butyl (6-methylpyridin-2-yl)carbamate, 90101-22-7, 2-(Boc-Amino)-6-Picoline, tert-Butyl 6-methylpyridin-2-ylcarbamate, Tert-butyl N-(6-methylpyridin-2-yl)carbamate, 2-Amino-6-methylpyridine, 2-BOC protected, (6-METHYL-(PYRIDIN-2-YL))-CARBAMIC ACID TERT-BUTYL ESTER, CARBAMIC ACID, (6-METHYL-2-PYRIDINYL)-, 1,1-DIMETHYLETHYL ESTER, 2-BOC protected, SureCN533505, AGN-PC-007OXA, CTK4E4554, MolPort-000-140-097, ANW-48000, ZINC15021499, AKOS005255287, AB42387, AG-E-50877, OR14770, RP04685
InChIKey: XSVAARVWQDEAEL-UHFFFAOYSA-N | ||||||||
| • (r )-2-aminomethyl-pyrrolidine-1-carboxylic Acid Tert-butyl Ester
IUPAC Name: tert-butyl 2-(aminomethyl)pyrrolidine-1-carboxylate | CAS Registry Number: 259537-92-3 Synonyms: (R)-1-Boc-2-(aminomethyl)pyrrolidine, FS011276
InChIKey: SOGXYCNKQQJEED-UHFFFAOYSA-N | ||||||||
| • (R)-1-Boc-2-cyanopyrrolidine
IUPAC Name: tert-butyl (2R)-2-cyanopyrrolidine-1-carboxylate | CAS Registry Number: 228244-20-0 Synonyms: (R)-1-N-BOC-2-CYANO-PYRROLIDINE, (R)-N-BOC-2-pyrrolidinonitrile, tert-butyl (2R)-2-cyanopyrrolidine-1-carboxylate, AG-E-65769, (R)-(+)-1-Boc-2-pyrrolidinecarbonitrile, AC1MBUDD, PubChem18389, (R)-tert-butyl 2-cyanopyrrolidine-1-carboxylate, SureCN2896482, 647233_ALDRICH, CTK4F0279, MolPort-000-140-607, ANW-47294, OR4611, ZINC00404034, AKOS005258740, AB25300, AC-2244, AK-29021, BR-29021
InChIKey: MDMSZBHMBCNYNO-MRVPVSSYSA-N | ||||||||
| • (R)-1-Boc-2-ethylpiperazine
IUPAC Name: tert-butyl (2R)-2-ethylpiperazine-1-carboxylate | CAS Registry Number: 393781-70-9 Synonyms: (R)-1-Boc-2-Ethyl-piperazine, (R)-1-Boc-2-ethylPiperazine, (R)-tert-butyl 2-ethylpiperazine-1-carboxylate, tert-Butyl-2(R)-ethyl-1-piperazinecarboxylate, tert-Butyl (2R)-2-ethylpiperazine-1-carboxylate, SBB056112, AG-F-39142, (S)-1-Boc-2-ethyl-piperazine, 1-Piperazinecarboxylic acid, 2-ethyl-, 1,1-dimethylethyl ester, (2R)-, PubChem18340, PubChem18343, SureCN337351, Jsp006835, CTK4I1301, MolPort-000-140-573, RS-11, ANW-49208, AKOS005258565, AKOS015910195, AC-2205
InChIKey: CTCGRXDGXGUOTE-SECBINFHSA-N | ||||||||
| • (R)-1-Boc-2-isopropyl-piperazine
IUPAC Name: tert-butyl (2R)-2-propan-2-ylpiperazine-1-carboxylate | CAS Registry Number: 674792-04-2 Synonyms: (R)-1-Boc-2-isopropylpiperazine, (R)-tert-butyl 2-isopropylpiperazine-1-carboxylate, (R)-1-Boc- 2-isopropyl-piperazine, SBB056113, tert-Butyl (2R)-2-isopropylpiperazine-1-carboxylate, AG-G-55169, (R)-2-ISOPROPYL-PIPERAZINE-1-CARBOXYLIC ACID TERT-BUTYL ESTER, 1-Piperazinecarboxylic acid, 2-(1-methylethyl)-, 1,1-dimethylethyl ester, (2R)-, SureCN3618472, CTK5C6229, MolPort-000-140-577, BH133, ANW-52377, FC0178, AKOS005258579, AB42213, RP05471, AC-17376, AK-30116, BL002244
InChIKey: NZTWGWFHWJARJX-JTQLQIEISA-N | ||||||||
| • (R)-1-Boc-3-((dimethylamino)methyl)pyrrolidine
IUPAC Name: tert-butyl (3R)-3-[(dimethylamino)methyl]pyrrolidine-1-carboxylate | CAS Registry Number: 859027-48-8 Synonyms: AG-H-46454, PubChem18382, SureCN3568388, CTK5F5942, MolPort-000-140-601, AKOS015850673, AKOS015910632, AC-2237, RP05473, AK-30138, KB-02742, S919, AB1005738, TL8005596, FT-0084103, FT-0601701, ST51055051, A841484, R-1-BOC-3-DIMETHYLAMINOMETHYL-PYRROLIDINE, I14-3968
InChIKey: SVFCKPUIJBZBQS-SNVBAGLBSA-N | ||||||||
| • (R)-1-Boc-3-ethyl-piperazine
IUPAC Name: tert-butyl (3R)-3-ethylpiperazine-1-carboxylate | CAS Registry Number: 438050-08-9 Synonyms: (R)-1-Boc-3-Ethylpiperazine, (R)-tert-butyl 3-ethylpiperazine-1-carboxylate, (R)-1-Boc- 3-ethyl-piperazine, AG-F-54567, SureCN2799343, PS-RS-12, CTK4I7748, MolPort-000-140-580, ANW-58040, AKOS007930665, AKOS015910030, AC-2209, RP04921, AK-29250, BL002248, KB-63134, AB1005781, TL8003068, BB 0261541, FT-0084000
InChIKey: DXJOJUNLMJMJSN-SECBINFHSA-N |