Profile: Jinan Trio PharmaTech Co., Ltd. specializes in APIs & intermediates, heterocyclic compounds, and anti-tumor drugs. Our products include crizotinib, vemurafenib, afatinib, vandetanib, regorafenib, brivanib alaninate, pyridazine, imidazole, pyrazole, and oxazole. We are specialized in providing over 1000 products including molecular targeted anticancer drugs, cell signaling pathway inhibitors, pharmaceutical intermediates, and heterocyclic compounds, and quality services including custom synthesis, transfer of new drug patent and technology, technical cooperation, and process optimization.
• NVP-BGT226
IUPAC Name: (Z)-but-2-enedioic acid;8-(6-methoxypyridin-3-yl)-3-methyl-1-[4-piperazin-1-yl-3-(trifluoromethyl)phenyl]imidazo[4,5-c]quinolin-2-one | CAS Registry Number: 1245537-68-1 Synonyms: BGT226, BGT-226, BGT226 maleate salt, NVPBGT226, SureCN996046, cc-443, NVP BGT 226, UNII-4YG62LG876, BGT226,NVP-BGT226, CHEBI:71953, BCP9000400, CS-0583, RL01113, HY-13334, BCP0726000185, NVP-BGT226|1245537-68-1|NVP BGT 226, 1245537-68-1 , C32H29F3N6O6 , NVP BGT226, 4-{4-[8-(6-methoxypyridin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]quinolin-1-yl]-2-(trifluoromethyl)phenyl}piperazin-1-ium (2Z)-3-carboxyacrylate, 8-(6-methoxypyridin-3-yl)-3-methyl-1-[4-(piperazin-1-yl)-3-(trifluoromethyl)phenyl]-1,3-dihydro-2H-imidazo[4,5-c]quinolin-2-one (2Z)-but-2-enedioate
InChIKey: YUXMAKUNSXIEKN-BTJKTKAUSA-N | ||||||||
• NVP-BHG712
IUPAC Name: 4-methyl-3-[(1-methyl-6-pyridin-3-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]-N-[3-(trifluoromethyl)phenyl]benzamide | CAS Registry Number: 940310-85-0 Synonyms: 940310-85-0 , NVP BHG712, 4-Methyl-3-[[1-methyl-6-(3-pyridinyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino]-N-[3-(trifluoromethyl)phenyl]benzamide, S2202_Selleck, NVPBHG712, AGN-PC-015AWW, SureCN4699731, cc-540, NVP BHG 712, QCR-258, MolPort-016-633-311, BCP9001010, CS-0469, RL05902, NCGC00249391-01, HY-13258, KB-58915, NVP-BHG712-Supplied by Selleck Chemicals, X7502, NVP-BHG712|940310-85-0|NVP BHG 712, 4-methyl-3-(1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-ylamino)-N-(3-(trifluoromethyl)phenyl)benzamide
InChIKey: ZCCPLJOKGAACRT-UHFFFAOYSA-N | ||||||||
• NVP-BKM-120
IUPAC Name: 5-(2,6-dimorpholin-4-ylpyrimidin-4-yl)-4-(trifluoromethyl)pyridin-2-amine | CAS Registry Number: 944396-07-0 Synonyms: BKM120, Buparlisib, BKM 120, NVP-BKM120, CHEMBL2017974, CHEBI:71954, BKM-120, 5-(2,6-dimorpholinopyrimidin-4-yl)-4-(trifluoromethyl)pyridin-2-amine, 5-[2,6-Di(4-morpholinyl)-4-pyrimidinyl]-4-(trifluoromethyl)-2-pyridinamine, 1202777-78-3, BKM120, BKM-120|, 5-[2,6-Di(Morpholin-4-Yl)pyrimidin-4-Yl]-4-(Trifluoromethyl)pyridin-2-Amine, Buparlisib [INN], S2247_Selleck, 3sd5, SureCN146956, QCR-4, UNII-0ZM2Z182GD, BKM 120NX, BKM120-NX
InChIKey: CWHUFRVAEUJCEF-UHFFFAOYSA-N | ||||||||
• NVP-BSK805
IUPAC Name: 4-[[2,6-difluoro-4-[3-(1-piperidin-4-ylpyrazol-4-yl)quinoxalin-5-yl]phenyl]methyl]morpholine;dihydrochloride | CAS Registry Number: 1092499-93-8 Synonyms: 1092499-93-8 pound not NVP BSK805, NVP-BSK805 2HCl, NVP-BSK805 dihydrochloride, cc-625, NVP-GSK 805, NVP-BSK805/NVPBSK805, BCP9001012, BCP0726000306, X7514, 8-(3,5-difluoro-4-(morpholinomethyl)phenyl)-2-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)quinoxaline, 8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-[1-(piperidin-4-yl)pyrazol-4-yl]quinoxaline dihydrochloride
InChIKey: NUOCAPALWRHKCU-UHFFFAOYSA-N | ||||||||
• NVP-BVU972
IUPAC Name: 6-[[6-(1-methylpyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl]quinoline | CAS Registry Number: 1185763-69-2 Synonyms: 3qti, NVPBVU972, SureCN1659100, NVP BVU972, cc-601, BVU972, BCP9000466, CS-0967, NCGC00346689-01, HY-15456, BCP0726000188, NVP-BVU972|1185763-69-2, 958025-66-6 , C20H16N6 , NVP BVU972
InChIKey: RNCNPRCUHHDYPC-UHFFFAOYSA-N | ||||||||
• NVP-LDE 225
IUPAC Name: N-[6-[(2S,6R)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]-2-methyl-3-[4-(trifluoromethoxy)phenyl]benzamide | CAS Registry Number: 956697-53-3 Synonyms: Erismodegib, LDE225, NVP-LDE225, LDE 225, LDE-225, LDE225, NVP-LDE225, Sonidegib (INN), N-(6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl)-2-methyl-3-[4-(trifluoromethoxy)phenyl]benzamide, N-{6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl}-2-methyl-3-[4-(trifluoromethoxy)phenyl]benzamide, Erismodegib [INN], Erismodegib (USAN), S2151_Selleck, PubChem22446, UNII-0RLU3VTK5M, Erismodegib [USAN:INN], cc-76, SureCN554455, CHEMBL2105737, MolPort-009-194-121, LDE 225, NVP-LDE225
InChIKey: VZZJRYRQSPEMTK-CALCHBBNSA-N | ||||||||
• NVP-TAE 226
IUPAC Name: 2-[[5-chloro-2-(2-methoxy-4-morpholin-4-ylanilino)pyrimidin-4-yl]amino]-N-methylbenzamide | CAS Registry Number: 761437-28-9 Synonyms: 2-((5-Chloro-2-((2-methoxy-4-morpholinophenyl)amino)pyrimidin-4-yl)amino)-N-methylbenzamide, 2-({5-Chloro-2-[(2-Methoxy-4-Morpholin-4-Ylphenyl)amino]pyrimidin-4-Yl}amino)-N-Methylbenzamide, 2jkk, 2-[5-chloro-2-(2-methoxy-4-morpholin-4-yl-phenylamino)-pyrimidin-4-ylamino]-N-methyl-benzamide, Kinome_1212, SureCN375524, NVP-TAE226, CHEMBL458997, TAE226, CTK8B9478, CHEBI:614994, ANW-62587, AKOS016004135, CS-0594, DB07460, NCGC00346931-01, AK101877, HY-13203, NVP-TAE 226,CAS:761437-28-9, NVP-TAE 226|761437-28-9
InChIKey: UYJNQQDJUOUFQJ-UHFFFAOYSA-N | ||||||||
• NVP-TAE684
IUPAC Name: 5-chloro-2-N-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-4-N-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | CAS Registry Number: 761439-42-3 Synonyms: TAE684, NVP-TAE 684, TAE-684, 5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine, TAE684, 761439-42-3, TAE684, NVP-TAE684, GUI, S1108_Selleck, Kinome_1205, PubChem16769, cc-17, SureCN282775, AGN-PC-00RX8K, NVP TAE684, UNII-EH1713MN4K, NVP TAE 684, NVT-TAE-684, CHEMBL509032, TAE 684, CHEBI:547450
InChIKey: QQWUGDVOUVUTOY-UHFFFAOYSA-N | ||||||||
• Obatoclax Mesylate
IUPAC Name: 2-[(5Z)-5-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-4-methoxypyrrol-2-ylidene]indole;methanesulfonic acid | CAS Registry Number: 803712-79-0 Synonyms: Obatoclax mesylate, ACT06786
InChIKey: ZVAGBRFUYHSUHA-RKMKAUCSSA-N | ||||||||
• Omeprazole
IUPAC Name: 6-methoxy-2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methylsulfinyl]-1H-benzimidazole | CAS Registry Number: 73590-58-6 Synonyms: omeprazole, Prilosec, Antra, Losec, Omeprazon, Audazol, Omapren, Omepral, Parizac, Mopral, Miol, Demeprazol, Inhibitron, Ulcometion, Belmazol, Ceprandal, Dizprazol, Dudencer, Emeproton, Epirazole
InChIKey: SUBDBMMJDZJVOS-UHFFFAOYSA-N | ||||||||
• ON-01910
IUPAC Name: sodium;2-[2-methoxy-5-[[(E)-2-(2,4,6-trimethoxyphenyl)ethenyl]sulfonylmethyl]anilino]acetate | CAS Registry Number: 1225497-78-8 Synonyms: Novonex, Estybon, Rigosertib sodium, Estybon, ON-01910, ON 01910, Estybon, ON-01910, 1225497-78-8, 592542-60-4, S1362_Selleck, Rigosertib sodium (USAN), ON 01910 sodium salt, cc-628, ON-1910Na, Onc-01910, CHEMBL2013119, ON-01910Na, SyB C-1101, SyB L-1101, MolPort-016-633-202, ON 01910.Na, BCP9001024
InChIKey: VLQLUZFVFXYXQE-USRGLUTNSA-M | ||||||||
• ONX 0914; PR 957
IUPAC Name: (2S)-3-(4-methoxyphenyl)-N-[(2S)-1-(2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-yl]-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide | CAS Registry Number: 960374-59-8 Synonyms: QC-7242, (2S)-3-(4-methoxyphenyl)-N-((2S)-1-(2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-yl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
InChIKey: WQAVPPWWLLVGFK-ZCKRSBOQSA-N | ||||||||
• OSI-027
IUPAC Name: 4-[(5Z)-4-amino-5-(7-methoxyindol-2-ylidene)-1H-imidazo[5,1-f][1,2,4]triazin-7-yl]cyclohexane-1-carboxylic acid | CAS Registry Number: 936890-98-1 Synonyms: OSI027, OSI 027, OSI027, OSI-027, K1146_Kinasechem, S2624_Selleck, Cyclohexanecarboxylic acid, 4-(4-amino-5-(7-methoxy-1H-indol-2-yl)imidazo(5,1-f)(1,2,4)triazin-7-yl)-, trans-, UNII-25MKH1SZ0M, cc-501, BCP9001034, CS-0257, HY-10423, OSI-027|936890-98-1|OSI 027, OSI 027, OSI-027, 936890-98-1, OSI 027, OSI-027, 936890-98-1, (+/-)-Cyclohexanecarboxylic acid, 4-(4-amino-5-(7-methoxy-1H-indol-2-yl)imidazo(5,1-f)(1,2,4)triazin-7-yl)-, trans-, (1r,4r)-4-[4-amino-5-(7-methoxy-1H-indol-2-yl)imidazo[4,3-f][1,2,4]triazin-7-yl]cyclohexane-1-carboxylic acid
InChIKey: CDNMDRUIGNHEMR-VKAVYKQESA-N | ||||||||
• OSI-420 (DESMETHYL ERLOTINIB)
IUPAC Name: 2-[4-(3-ethynylanilino)-7-(2-methoxyethoxy)quinazolin-6-yl]oxyethanol | CAS Registry Number: 183321-86-0 Synonyms: OSI-420, Free Base (Desmethyl Erlotinib), 183321-86-0 pound>>183320-51-6, CTK8F1287, BCPP000136, Desmethyl Erlotinib (CP-473420), ZINC22065493, BCP9001036, NCGC00346578-01, KB-59328, FT-0673312, FT-0673313, 2-[[4-[(3-Ethynylphenyl)amino]-7-(2-methoxyethoxy)-6-quinazolinyl]oxy]ethanol
InChIKey: KOQIAZNBAWFSQM-UHFFFAOYSA-N | ||||||||
• OSI-906
IUPAC Name: 3-[8-amino-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl]-1-methylcyclobutan-1-ol | CAS Registry Number: 867160-71-2 Synonyms: Linsitinib, Kinome_3532, OSI-906AA, OSI906, OSI-906, 867160-71-2, 3-[8-amino-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl]-1-methylcyclobutan-1-ol, cis-3-(8-amino-1-(2-phenyl-7-quinolinyl)imidazo(1,5-a)pyrazin-3-yl)-1-methylcyclobutanol, cis-3-[8-Amino-1-(2-phenyl-7-quinolinyl)imidazo[1,5-a]pyrazin-3-yl]-1-methylcyclobutanol, Linsitinib [USAN], Linsitinib (USAN/INN), SureCN400369, SureCN400734, SureCN400735, AGN-PC-00D7QU, UNII-15A52GPT8T, SureCN10255925, cc-217, CHEMBL1091644, OSI 906, QCR-128
InChIKey: PKCDDUHJAFVJJB-UHFFFAOYSA-N | ||||||||
• OSI-930
IUPAC Name: 3-(quinolin-4-ylmethylamino)-N-[4-(trifluoromethoxy)phenyl]thiophene-2-carboxamide | CAS Registry Number: 728033-96-3 Synonyms: OSI930, S1220_Selleck, OSI 930, CHEMBL1614710, OSI-930 is a multi-targeted tyrosine kinase inhibitor, 3-[(4-Quinolinylmethyl)amino]-N-[4-(trifluoromethoxy)phenyl]-2-thiophenecarboxamide, CID9868037, SureCN633719, cc-339, DCL000352, BCP9001037, CS-0174, RL04771, 3-(quinolin-4-ylmethylamino)-N-[4-(trifluoromethoxy)phenyl]thiophene-2-carboxamide, OSI-930-Supplied by Selleck Chemicals, NCGC00263159-01, HY-10204, X7484, OSI-930|728033-96-3|OSI930, 3-[(quinolin-4-ylmethyl)amino]-N-[4-(trifluoromethoxy)phenyl]thiophene-2-carboxamide
InChIKey: FGTCROZDHDSNIO-UHFFFAOYSA-N | ||||||||
• OSU-03012
IUPAC Name: 2-amino-N-[4-[5-phenanthren-2-yl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]acetamide | CAS Registry Number: 742112-33-0 Synonyms: CHEMBL1650595, OSU03012, OSU03012, OSU 03012, 742112-33-0, 2-amino-N-(4-(5-(phenanthren-2-yl)-3-(trifluoromethyl)-1H-pyrazol-1-yl)phenyl)acetamide, N/AAR-12, OSU03012, OSU-03012, S1106_Selleck, PubChem22592, PDK1 inhibitor AR-12, UNII-EX3O2Q61UV, cc-115, MolPort-009-019-120, BCPP000134, ABP000481, BCP9001039, CS-0151, RL04816, RL04817, NCGC00346490-01, HY-10547, OSU-03012-Supplied by Selleck Chemicals
InChIKey: YULUCECVQOCQFQ-UHFFFAOYSA-N | ||||||||
• Oxaliplatin
IUPAC Name: (1R,2R)-cyclohexane-1,2-diamine; oxalate; platinum(2+) | CAS Registry Number: 61825-94-3 Synonyms: oxaliplatin, oxalate, Oxalatoplatin, Oxalatoplatinum, Eloxatin, Eloxatin (TN), platinum(+2) cation, Oxaliplatinum [Latin], Oxaloplatine [French], Oxaliplatino [Spanish], Oxaloplatino [Spanish], Oxaliplatin (JAN/USAN/INN), Oxaliplatin [USAN:INN:BAN], (1R,2R)-cyclohexane-1,2-diamine, DB00526, D01790
InChIKey: ZROHGHOFXNOHSO-BNTLRKBRSA-L | ||||||||
• OXAZOLE, 2-CHLORO-
IUPAC Name: 2-chloro-1,3-oxazole | CAS Registry Number: 95458-77-8 Synonyms: Oxazole, 2-chloro-, 2-Chlorooxazole, 2-CHLORO-OXAZOLE, SureCN317377, AGN-PC-00ME2Y, CTK3I6009, AKOS006288793, AG-H-92848, FT-0645180
InChIKey: SSXYKBHZZRYLLY-UHFFFAOYSA-N | ||||||||
• OXAZOLE,5-(CHLOROMETHYL)-
IUPAC Name: 5-(chloromethyl)-1,3-oxazole | CAS Registry Number: 172649-57-9 Synonyms: 5-(Chloromethyl)oxazole, OXAZOLE, 5-(CHLOROMETHYL)-, AGN-PC-00ORQJ, SureCN7442697, CTK8C2828, ANW-69074, RB3366, AKOS006286857, AB42450, 5-(CHLOROMETHYL)-1,3-OXAZOLE, AK-48287, KB-243840, FT-0084326, FT-0660245
InChIKey: UJLHZLUVPVJDQI-UHFFFAOYSA-N | ||||||||
• Oxazole-2-Carbaldehyde
IUPAC Name: 1,3-oxazole-2-carbaldehyde | CAS Registry Number: 65373-52-6 Synonyms: Oxazole-2-carbaldehyde, 2-Oxazolecarboxaldehyde, 1,3-oxazole-2-carbaldehyde, SBB052295, zlchem 772, PubChem17600, AGN-PC-002JTD, OXAZOLE-2-CARBOXALDEHYDE, 1,3-Oxazole-2-carboxaldehyde;, CTK2F2741, ZLD0231, MolPort-004-747-047, ACT06108, WTI-10543, ZINC02530178, 1,3-OXAZOLE-2-CARBOXALDEHYDE, AKOS006342976, AB14413, AG-B-76909, AG-G-46050
InChIKey: TYHOSUCCUICRLM-UHFFFAOYSA-N | ||||||||
• OXAZOLO[4,5-C]PYRIDIN-2-AMINE
IUPAC Name: [1,3]oxazolo[4,5-c]pyridin-2-amine | CAS Registry Number: 114498-55-4 Synonyms: Oxazolo[4,5-c]pyridin-2-amine, ACMC-20adcd, AGN-PC-000U7Q, CTK0H3203, MolPort-004-757-684, ANW-68219, AKOS016007039, AG-D-34817, QC-4947, Oxazolo[4,5-c]pyridin-2-amine (9CI), AK-80598, BD236979, KB-79732
InChIKey: FJHYVYMTPVSYDO-UHFFFAOYSA-N | ||||||||
• Oxazolo[4,5-c]pyridine, 7-bromo-2-ethyl-
IUPAC Name: 7-bromo-2-ethyl-[1,3]oxazolo[4,5-c]pyridine | CAS Registry Number: 118685-69-1 Synonyms: 7-Bromo-2-ethyloxazolo[4,5-c]pyridine, CTK8C2335, ANW-68217, AKOS016007061, AK-80600, KB-79734, Oxazolo[4,5-c]pyridine,7-bromo-2-ethyl-
InChIKey: AMHXDXSOKYQXFX-UHFFFAOYSA-N | ||||||||
• Oxazolo[4,5-c]pyridine, 7-bromo-2-methyl-
IUPAC Name: 7-bromo-2-methyl-[1,3]oxazolo[4,5-c]pyridine | CAS Registry Number: 116081-17-5 Synonyms: 7-Bromo-2-methyloxazolo[4,5-c]pyridine, CTK8C2336, ANW-68218, AKOS016007060, AK-80599, BD236980, KB-79735, Oxazolo[4,5-c]pyridine,7-bromo-2-methyl-
InChIKey: LACXEYMKTOJZHX-UHFFFAOYSA-N | ||||||||
• P 22077
IUPAC Name: 1-[5-(2,4-difluorophenyl)sulfanyl-4-nitrothiophen-2-yl]ethanone | CAS Registry Number: 1247819-59-5 Synonyms: CHEMBL2159498, SureCN2680945, QC-8199, 1-(5-(2,4-difluorophenylthio)-4-nitrothiophen-2-yl)ethanone
InChIKey: RMAMGGNACJHXHO-UHFFFAOYSA-N | ||||||||
• P-Methoxyacetanilide
IUPAC Name: N-(4-methoxyphenyl)acetamide | CAS Registry Number: 51-66-1 Synonyms: p-Acetanisidide, Metacetin, Methacetin, p-Acetanisidine, Aceto-p-anisidide, Acetyl-p-anisidine, p-Methoxyacetanilide, N-Acetyl-p-anisidine, 4'-Methoxyacetanilide, N-(4-Methoxyphenyl)acetamide, N-Acetyl-p-methoxyaniline, Acetanilide, 4'-methoxy-, 4-METHOXYACETANILIDE, Acetamide, N-(4-methoxyphenyl)-, WLN: 1VMR DO1, ARONIS003521, NSC 4687, EINECS 200-114-2, NSC4687, BRN 0387887
InChIKey: XVAIDCNLVLTVFM-UHFFFAOYSA-N | ||||||||
• P-TOLUENESULFONYL-L-ARGININE METHYL ESTER HCL
IUPAC Name: methyl 5-(diaminomethylideneamino)-2-[(4-methylphenyl)sulfonylamino]pentanoate | CAS Registry Number: 901-47-3 Synonyms: Probes1_000325, Probes2_000471, CBDivE_015738, CHEBI:380054, MolPort-001-813-207, NSC80683, CID416661, Arginine, N(2)-p-toluenesulfonyl-, methyl ester, p-TOLUENESULFONYL-L-ARGININE METHYL ESTER HCl, 5-Guanidino-2-(toluene-4-sulfonylamino)-pentanoic acid methyl ester
InChIKey: FKMJXALNHKIDOD-UHFFFAOYSA-N | ||||||||
• P005091
IUPAC Name: 1-[5-(2,3-dichlorophenyl)sulfanyl-4-nitrothiophen-2-yl]ethanone | CAS Registry Number: 882257-11-6 Synonyms: CHEMBL2159495, ZINC00125366, SureCN2681288, AC1ME173, MolPort-002-906-122, KM03205, QC-8200, 1-(5-(2,3-dichlorophenylthio)-4-nitrothiophen-2-yl)ethanone, 1-[5-(2,3-dichlorophenyl)sulfanyl-4-nitrothiophen-2-yl]ethanone, 1-{5-[(2,3-dichlorophenyl)thio]-4-nitro-2-thienyl}ethan-1-one
InChIKey: LKZLGMAAKNEGCH-UHFFFAOYSA-N | ||||||||
• PAC 1; 4-BENZYL-1-PIPERAZINEACETIC ACID [[2-HYDROXY-3-(2-ALLYL)PHENYL]METHYLENE]HYDRAZIDE
IUPAC Name: 2-(4-benzylpiperazin-1-yl)-N'-[(Z)-(6-oxo-5-prop-2-enylcyclohexa-2,4-dien-1-ylidene)methyl]acetohydrazide | CAS Registry Number: 315183-21-2 Synonyms: PAC-1, Procaspase-3 Activator, PAC-1, PAC 1 pound not Procaspase activating compound 1, 315183-21-2, (4-Benzylpiperazino)acetic acid-(3-allyl-2-hydroxybenzylidene)hydrazide, PAC 1, Procaspase-3 Activator, PAC-1 pound notPAC1, AC1OA9GH, cc-276, CHEMBL591429, Procaspase activating compound 1, STOCK3S-22963, MolPort-002-580-634, NSC743444, BCP9001044, NSC-743444, NCGC00167785-02, BCP0726000262, X5905, 2-(4-benzylpiperazin-1-yl)-N'-[(1E)-[2-hydroxy-3-(prop-2-en-1-yl)phenyl]methylidene]acetohydrazide
InChIKey: XSGXRYNZNGUGEJ-PGMHBOJBSA-N | ||||||||
• Paclitaxel
Synonyms: paclitaxel, Yewtaxan, TAXOL, Plaxicel, Paxceed, Taxol A, Abraxane, Ebetaxel, Capxol, Paxene, Onxol, TaxAlbin, LipoPac, Genetaxyl, Nanotaxel, Paclical, Pacligel, Anzatax, Genaxol, Genexol
InChIKey: RCINICONZNJXQF-MZXODVADSA-N | ||||||||
• PALBOCICLIB ISETHIONATE
IUPAC Name: 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7-one;2-hydroxyethanesulfonic acid | CAS Registry Number: 827022-33-3 Synonyms: Palbociclib Isethionate, AGN-PC-009X4E, Palbociclib Isethionate [USAN}, CHEMBL2364621, PD 0332991 (Palbociclib) Isethionate, PF-0008066573, PD 0332991-0054, PD-03329910054, PF-00080665-73, S1579,827022-33-3, 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7-one;2-hydroxyethanesulfonic acid
InChIKey: LYYVFHRFIJKPOV-UHFFFAOYSA-N | ||||||||
• Palomid 529
IUPAC Name: 8-(1-hydroxyethyl)-2-methoxy-3-[(4-methoxyphenyl)methoxy]benzo[c]chromen-6-one | CAS Registry Number: 914913-88-5 Synonyms: Palomid529, Palomid-529, P-529, P529, Palomid 529, P529, P529, 914913-88-5, 8-(1-hydroxyethyl)-2-methoxy-3-[(4-methoxyphenyl)methoxy]benzo[c]chromen-6-one, S2238_Selleck, AGN-PC-00JIQP, Palomid 529,P529, SureCN290034, SureCN7860257, UNII-XV9409EWG4, cc-513, Palomid 529 - P529, QCR-215, BCPP000131, BCP9001049, CS-0258, RL05762
InChIKey: YEAHTLOYHVWAKW-UHFFFAOYSA-N | ||||||||
• Pazopanib
IUPAC Name: 5-[[4-[(2,3-dimethylindazol-6-yl)-methylamino]pyrimidin-2-yl]amino]-2-methylbenzenesulfonamide | CAS Registry Number: 444731-52-6 Synonyms: GW786034, UNII-7RN5DR86CK, CHEBI:71219, NCGC00188865-01, GW 78603, Pazopanib [INN], DSSTox_CID_28659, DSSTox_RID_82929, DSSTox_GSID_48733, 790713-33-6, Kinome_3790, CHEMBL477772, 5-(4-((2,3-dimethyl-2H-indazol-6-yl)(methyl)amino)pyrimidin-2-ylamino)-2-methylbenzenesulfonamide, 5-[[4-[(2,3-Dimethyl-2H-indazol-6-yl)(methyl)amino]pyrimidin-2-yl]amino]-2-methylbenzenesulfonamide, Benzenesulfonamide, 5-[[4-[(2,3-dimethyl-2H-indazol-6-yl)methylamino]-2-pyrimidinyl]amino]-2-methyl-, CAS-444731-52-6, AKOS005145819, 5-[[4-[(2,3-dimethylindazol-6-yl)-methyl-amino]pyrimidin-2-yl]amino]-2-methyl-benzenesulfonamide, ST51053493, pazopanibum
InChIKey: CUIHSIWYWATEQL-UHFFFAOYSA-N | ||||||||
• PCI-32765
IUPAC Name: 1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | CAS Registry Number: 936563-96-1 Synonyms: Ibrutinib, PCI 32765, CHEBI:76612, PCI32765, UNII-1X70OSD4VX, ibrutinibum, CRA-032765, Imbruvica (TN), Ibrutinib (USAN), IMBRUVICA, SureCN201859, 1X70OSD4VX, PCI-32765 (Ibrutinib), CHEMBL1873475, AMX10219, EX-5960, QC-4573, NCGC00187912-01, NCGC00187912-02, NCGC00187912-03
InChIKey: XYFPWWZEPKGCCK-GOSISDBHSA-N | ||||||||
• PD 0325901
IUPAC Name: N-[(2R)-2,3-dihydroxypropoxy]-3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzamide | CAS Registry Number: 391210-10-9 Synonyms: nchembio.282-comp3, CHEBI:553228, ZINC03938683, CID9826528, PD-0325901, PD325901, PD 325901, PD-325901, PD0325901, C506614, (R)-(-)-N-(2,3-dihydroxy-propoxy)-3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-benzamide, N-[((R)-2,3-dihydroxypropyl)oxy]-3,4-difluoro-2-[(2-fluoro-4-iodophenyl)amino]benzamide, N-[(2R)-2,3-dihydroxypropoxy]-3,4-difluoro-2-[(2-fluoro-4-iodo-phenyl)amino]benzamide, N-{[(2R)-2,3-dihydroxypropyl]oxy}-3,4-difluoro-2-[(2-fluoro-4-iodophenyl)amino]benzamide, 4BM, 870474-62-7
InChIKey: SUDAHWBOROXANE-SECBINFHSA-N | ||||||||
• PD 173074
IUPAC Name: 1-tert-butyl-3-[2-[4-(diethylamino)butylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea | CAS Registry Number: 219580-11-7 Synonyms: PD173074, PD-173074, CHEBI:63448, 1-tert-butyl-3-[2-{[4-(diethylamino)butyl]amino}-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea, FGF/VEGF Receptor Tyrosine Kinase Inhibitor, PD173074, PD173074, 219580-11-7, 2fgi, 1-(tert-Butyl)-3-(2-((4-(diethylamino)butyl)amino)-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl)urea, 1-t-Butyl-3-(6-(3,5-dimethoxyphenyl)-2-(4-diethylaminobutylamino)-pyrido[2,3-d]pyrimidin-7-yl)urea, 1-tert-butyl-3-(2-(4-(diethylamino)butylamino)-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl)urea, 1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-urea, PD1, 1-tert-butyl-3-[2-[4-(diethylamino)butylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea, S1264_Selleck, PubChem22593, SureCN177946, AC1L1BE8, UNII-A4TLL8634Y, JSPY-st000263, cc-523
InChIKey: DXCUKNQANPLTEJ-UHFFFAOYSA-N | ||||||||
• PD0332991
IUPAC Name: 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7-one;hydrochloride | CAS Registry Number: 827022-32-2 Synonyms: PD 0332991 HCl, Palbociclib HCl, Palbociclib hydrochloride, AGN-PC-008ZCE, SureCN2076416, PD0332991 hydrochloride, cc-424, PD 0332991 hydrochloride, HY-50767A, CS-1327, RL05143, X7620, Palbociclib hydrochloride|827022-32-2|PD0332991 hydrochloride|PD 0332991 hydrochloride, 6-acetyl-8-cyclopentyl-5-methyl-2-((5-(1-piperazinyl)-2-pyridinyl)amino)pyrido(2,3-d)pyrimidin-7(8h)-one hydrochloride, 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7-one;hydrochloride, 6-acetyl-8-cyclopentyl-5-methyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}pyrido[2,3-d]pyrimidin-7-one hydrochloride
InChIKey: STEQOHNDWONVIF-UHFFFAOYSA-N | ||||||||
• PD318088
IUPAC Name: 5-bromo-N-(2,3-dihydroxypropoxy)-3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzamide | CAS Registry Number: 391210-00-7 Synonyms: PD 318088, PD-318088, S1568_Selleck, AGN-PC-01LTJY, C16H13BrF3IN2O4, cc-457, MolPort-006-168-845, BCPP000120, BCP9001066, CS-0222, RL03489, NCGC00346552-01, HY-12062, PD318088-Supplied by Selleck Chemicals, X7397, PD 318088, 391210-00-7, PD318088|391210-00-7|PD-318088, 5-bromo-N-(2,3-dihydroxypropoxy)-3,4-difluoro-2-(2-fluoro-4-iodophenylamino)benzamide, 5-BROMO-N-(2,3-DIHYDROXYPROPOXY)-3,4-DIFLUORO-2-[(2-FLUORO-4-IODOPHENYL)AMINO]-, 5-bromo-N-[(2R)-2,3-dihydroxypropoxy]-3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzamide
InChIKey: XXSSGBYXSKOLAM-UHFFFAOYSA-N | ||||||||
• Pelitinib
IUPAC Name: (E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)but-2-enamide | CAS Registry Number: 257933-82-7 Synonyms: EKB-569, Pelitinib (USAN/INN), WAY-EKB 569, WAY-EKB-569, CHEBI:38927, EKB 569, NSC729742, CID6445562, WAY-172569, D05399, (2E)-N-(4-((3-chloro-4-fluorophenyl)amino)-3-cyano-7-ethoxy-6-quinolinyl)-4-(dimethylamino)-2-butenamide, (2E)-N-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamide, (E)-N-[4-(3-Chloro-4-fluoroanilino)-cyano-7-ethoxyquinolin-6-yl]-4-(dimethlyamino)but-2-enamide,, 2-Butenamide, N-(4-((3-chloro-4-fluorophenyl)amino)-3-cyano-7-ethoxy-6-quinolinyl)-4-(dimethylamino)-, (2E)-, 2-Butenamide, N-[4-(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl-4-(dimethylamino)-, (E)-,, 4-Dimethylaminobut-2-enoic Acid, [4-(3-Chloro-4-fluoro phenylamino)-3-cyano-7-ethoxyquinoline-6-yl]amide
InChIKey: WVUNYSQLFKLYNI-AATRIKPKSA-N | ||||||||
• Pemetrexed
IUPAC Name: (2R)-2-[[4-[2-(2-amino-4-oxo-1,7-dihydropyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]amino]pentanedioic acid | CAS Registry Number: 137281-23-3 Synonyms: Alimta, Pemetrexed disodium, Pemetrexed [INN:BAN], UNII-04Q9AIZ7NO, HSDB 7316, C20H21N5O6, CID60843, LY231514, DB00642, LY 231514, LY 231,514, LS-172988, LY-231514, LY-231,514, L-Glutamic acid, N-(4-(2-(2-amino-4,7-dihydro-4-oxo-1H-pyrrolo(2,3-d)pyrimidin-5-yl)ethyl)benzoyl)-, N-(4-(2-(2-Amino-3,4-dihydro-4-oxo-7H-pyrrolo(2,3-d)pyrimdin-5-yl)ethyl)benzoyl)glutamic acid, (2R)-2-[[4-[2-(2-amino-4-oxo-1,7-dihydropyrrolo[4,5-e]pyrimidin-5-yl)ethyl]benzoyl]amino]pentanedioic acid, MTA
InChIKey: WBXPDJSOTKVWSJ-CYBMUJFWSA-N | ||||||||
• Pendimethalin
IUPAC Name: 3,4-dimethyl-2,6-dinitro-N-pentan-3-ylaniline | CAS Registry Number: 40487-42-1 Synonyms: Penoxaline, PENDIMETHALIN, Prowl, Pendimethaline, Tendimethalin, Phenoxalin, Herbadox, Penoxalin, Accotab, Penoxyn, Sipaxol, Stomp, Wayup, Wax Up, Way Up, Go-Go-San, SWGC, Stomp 330D, Stomp 330E, Caswell No. 454BB
InChIKey: CHIFOSRWCNZCFN-UHFFFAOYSA-N | ||||||||
• Pentanamide, 2-[[(4-Chlorophenyl)sulfonyl][[2-Fluoro-4-(1,2,4-Oxadiazol-3-Yl)phenyl]methyl]amino]-5,5,5-Trifluoro-, (2R)-
IUPAC Name: (2R)-2-[(4-chlorophenyl)sulfonyl-[[2-fluoro-4-(1,2,4-oxadiazol-3-yl)phenyl]methyl]amino]-5,5,5-trifluoropentanamide | CAS Registry Number: 1146699-66-2 Synonyms: BMS-708163, Avagacestat, BMS 708163, BMS-708163-01, BMS708163, Avagacestat (USAN), Avagacestat [USAN], BMS708163, 1146699-66-2, BMS708163, BMS-708163, S1262_Selleck, Avagacestat [USAN:INN], SureCN310019, UNII-TQ44WWY45Q, cc-297, CHEMBL1090771, BCPP000327, (2R)-2-[N-[(4-CHLOROPHENYL)SULFONYL]-N-[2-FLUORO-4-(1,2,4-OXADIAZOL-3-YL)BENZYL]AMINO]-5,5,5-TRIFLUOROPENTANAMIDE, AKOS005146523, AKOS016016280, BCP9000429
InChIKey: XEAOPVUAMONVLA-QGZVFWFLSA-N | ||||||||
• Perifosine
IUPAC Name: (1,1-dimethylpiperidin-1-ium-4-yl) octadecyl phosphate | CAS Registry Number: 157716-52-4 Synonyms: Perifosine [INN], NKA17, KRX-0401, CID148177, NSC639966, NSC 639966, NSC-639966, D 21266, D-21266, octadecyl-(1,1-dimethyl-4-piperidylio)phosphate, C105905, 4-((Hydroxy(octadecyloxy)phosphinyl)oxy)-1,1-dimethylpiperidinium inner salt, Piperidinium, 4-((hydroxy(octadecyloxy)phosphinyl)oxy)-1,1-dimethyl-, inner salt, Piperidinium, 4-[[hydroxy(octadecyloxy)phosphinyl]oxy]-1,1-dimethyl-, inner salt
InChIKey: SZFPYBIJACMNJV-UHFFFAOYSA-N | ||||||||
• PF 4708671
IUPAC Name: 2-[[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl]-6-(trifluoromethyl)-1H-benzimidazole | CAS Registry Number: 1255517-76-0 Synonyms: PF-4708671, 2-((4-(5-Ethylpyrimidin-4-yl)piperazin-1-yl)methyl)-5-(trifluoromethyl)-1H-benzo[d]imidazole, 2-{[4-(5-Ethylpyrimidin-4-Yl)piperazin-1-Yl]methyl}-5-(Trifluoromethyl)-1h-Benzimidazole, 5FI, CHEMBL2134202, HMS3263P20, CCG-222583, QC-8396, NCGC00263134-01, FT-0673656, S2163,PF4708671,PF-04708671,1255517-76-0, 2-[[4-(5-ethyl-4-pyrimidinyl)-1-piperazinyl]methyl]-6-(trifluoromethyl)-1H-benzimidazole
InChIKey: FBLPQCAQRNSVHB-UHFFFAOYSA-N | ||||||||
• PF-00299804; Dacomitinib
IUPAC Name: (E)-N-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]-4-piperidin-1-ylbut-2-enamide | CAS Registry Number: 1110813-31-4 Synonyms: Dacomitinib, PF299804, PF-299804, 1110813-31-4 pound not PF 299804 pound not PF-299804, (2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-7-methoxy-6-quinazolinyl]-4-(1-piperidinyl)-2-butenamide, (2e)-N-{4-[(3-Chloro-4-Fluorophenyl)amino]-7-Methoxyquinazolin-6-Yl}-4-(Piperidin-1-Yl)but-2-Enamide, Dacomitinib [USAN], SureCN33147, Dacomitinib (USAN/INN), cc-194, UNII-2XJX250C20, CHEMBL2110732, QCR-174, PF-299, CS-0500, RL00451, HY-13272, KB-76397, PF 299804, Y0338
InChIKey: LVXJQMNHJWSHET-AATRIKPKSA-N | ||||||||
• PF-04217903
IUPAC Name: 2-[4-[3-(quinolin-6-ylmethyl)triazolo[4,5-b]pyrazin-5-yl]pyrazol-1-yl]ethanol | CAS Registry Number: 956905-27-4 Synonyms: PF 04217903, CHEMBL2001019, PF04217903, aka PF-04217903, PF04217903, 956905-27-4, 1159490-85-3, PF-04217903, PF04217903, 3zxz, 2-(4-(1-(Quinolin-6-ylmethyl)-1H-(1,2,3)triazolo(4,5-b)pyrazin-6-yl)-1H-pyrazol-1-yl)ethanol, 2-(4-(1-(quinolin-6-ylmethyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)-1H-pyrazol-1-yl)ethanol, S1094_Selleck, Kinome_3829, PubChem19150, PubChem22335, UNII-CYJ9ATV1IJ, SureCN93550, AGN-PC-01LTWA, cc-599, QCR-189, MolPort-016-633-176
InChIKey: PDMUGYOXRHVNMO-UHFFFAOYSA-N | ||||||||
• PF-04691502
IUPAC Name: 2-amino-8-[4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7-one | CAS Registry Number: 1013101-36-4 Synonyms: CHEMBL1234354, PF04691502, PF 04691502, 1013101-36-4 pound not PF04691502 pound not PF 04691502, 2-amino-8-((1r,4r)-4-(2-hydroxyethoxy)cyclohexyl)-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8H)-one, PubChem24348, SureCN1381425, SureCN1381431, SureCN1984896, SureCN10092210, SureCN13976989, cc-350, QCR-137, AKOS005266645, CS-0919, NCGC00346659-01, HY-15177, BCP0726000275, PF-4691502, X7464
InChIKey: XDLYKKIQACFMJG-UHFFFAOYSA-N | ||||||||
• PF-04929113?SNX5422?
IUPAC Name: [4-[2-carbamoyl-5-[6,6-dimethyl-4-oxo-3-(trifluoromethyl)-5,7-dihydroindazol-1-yl]anilino]cyclohexyl] 2-aminoacetate | CAS Registry Number: 908115-27-5 Synonyms: SNX-5422, SNX5422, SNX 5422, PF04929113, PF 04929113, PF-04929113, SNX-5422, PF-04929113, 908115-27-5, cc-40, SureCN1220790, SureCN1220791, UNII-BF52J69Q8T, BCPP000065, ABP000737, DCL000231, CS-0272, RL05706, NCGC00346640-01, HY-10213, PF-4929113, X7589
InChIKey: AVDSOVJPJZVBTC-UHFFFAOYSA-N | ||||||||
• PF-5274857
IUPAC Name: 1-[4-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]piperazin-1-yl]-3-methylsulfonylpropan-1-one | CAS Registry Number: 1373615-35-0 Synonyms: 1-(4-(5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl)piperazin-1-yl)-3-(methylsulfonyl)propan-1-one, SureCN2715391, cc-682, CS-1206, QC-1145, RL01646, NCGC00346696-01, HY-13459, KB-145934, PF5274857, Y0361, PF-5274857|1373615-35-0|PF5274857
InChIKey: BBVNTTZIOTWDSV-UHFFFAOYSA-N | ||||||||
• PF-562271
IUPAC Name: benzenesulfonic acid;N-methyl-N-[3-[[[2-[(2-oxo-1,3-dihydroindol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | CAS Registry Number: 939791-38-5 Synonyms: CHEMBL2430359, PF 562271, PF-00562271, cc-23, RS0038s, PF-562,271, Methanesulfonamide, N-(3-(((2-((2,3-dihydro-2-oxo-1H-indol-5-yl)amino)-5- (trifluoromethyl)-4-pyrimidinyl)amino)methyl)-2-pyridinyl)-N-methyl-, benzenesulfonate (1:1), Methanesulfonamide, N-[3-[[[2-[(2,3-dihydro-2-oxo-1H-indol-5-yl)amino]-5-(trifluoromethyl)-4-pyrimidinyl]amino]methyl]-2-pyridinyl]-N-methyl-, benzenesulfonate (1:1)
InChIKey: LKLWTLXTOVZFAE-UHFFFAOYSA-N |