Profile: Jinan Trio PharmaTech Co., Ltd. specializes in APIs & intermediates, heterocyclic compounds, and anti-tumor drugs. Our products include crizotinib, vemurafenib, afatinib, vandetanib, regorafenib, brivanib alaninate, pyridazine, imidazole, pyrazole, and oxazole. We are specialized in providing over 1000 products including molecular targeted anticancer drugs, cell signaling pathway inhibitors, pharmaceutical intermediates, and heterocyclic compounds, and quality services including custom synthesis, transfer of new drug patent and technology, technical cooperation, and process optimization.
| • N-[4-[(3-Chloro-4-fluorophenyl)amino]-7-[[(3S)-tetrahydro-3-furanyl]oxy]-6-quinazolinyl]-4-(dimethylamino)-2-butenamide
IUPAC Name: (E)-N-[4-(3-chloro-4-fluoroanilino)-7-[(3S)-oxolan-3-yl]oxyquinazolin-6-yl]-4-(dimethylamino)but-2-enamide | CAS Registry Number: 439081-18-2 Synonyms: Tovok, BIBW-2992, BIBW 2992, CID10184653, CID 10184653, 2-Butenamide, N-(4-((3-chloro-4-fluorophenyl)amino)-7-(((3S)-tetrahydro-3-furanyl)oxy)-6-quinazolinyl)-4-(dimethylamino)-, 915958-11-1
InChIKey: ULXXDDBFHOBEHA-CWDCEQMOSA-N | ||||||||
| • N-FORMYLGLYCINE ETHYL ESTER
IUPAC Name: ethyl 2-formamidoacetate | CAS Registry Number: 3154-51-6 Synonyms: Ethylformylglycine, N-Formylglycine ethyl ester, Ethyl Formamidoacetate, Ethyl N-formylglycinate, ethyl 2-formamidoacetate, 47719_ALDRICH, Glycine, N-formyl-, ethyl ester, Formamidoacetic Acid Ethyl Ester, 47719_FLUKA, MolPort-003-934-275, CID76615, NSC14440, EINECS 221-596-0, ZINC01653017, F0421, I14-1629
InChIKey: GMBCCEOJUWMBPF-UHFFFAOYSA-N | ||||||||
| • N-HYDROXY-3-[3-[(PHENYLAMINO)SULFONYL]PHENYL]-2-PROPENAMIDE
IUPAC Name: (E)-N-hydroxy-3-[3-(phenylsulfamoyl)phenyl]prop-2-enamide | CAS Registry Number: 414864-00-9 Synonyms: Belinostat, nchembio.313-comp10, Belinostat (USAN/INN), PXD101, PXD-101, PXD 101, CHEBI:535188, NSC726630, ZINC03818726, CID6918638, PX 105684, PX-105684, EC-000.2286, D08870, N-Hydroxy-3-(3-phenylsulphamoylphenyl)acrylamide, C487081, N-hydroxy-3-(3-phenylsulfamoyl-phenyl)-acrylamide, N-hydroxy-3-(3-(phenylsulfamoyl)phenyl)prop-2-enamide, 2-Propenamide, N-hydroxy-3-(3-((phenylamino)sulfonyl)phenyl)-
InChIKey: NCNRHFGMJRPRSK-MDZDMXLPSA-N | ||||||||
| • N-methyl-2-(4-methylpiperazin-1-yl)-N-(4-nitrophenyl)acetamide
IUPAC Name: N-methyl-2-(4-methylpiperazin-1-yl)-N-(4-nitrophenyl)acetamide | CAS Registry Number: 1139453-98-7 Synonyms: SureCN1361808, QC-1091, KB-79454
InChIKey: LSQRHFSGOUDQDS-UHFFFAOYSA-N | ||||||||
| • N-Methyl-3-Nitro-2-Pyridinamine
IUPAC Name: N-methyl-3-nitropyridin-2-amine | CAS Registry Number: 4093-88-3 Synonyms: n-methyl-3-nitropyridin-2-amine, N-Methyl-3-nitro-2-pyridinamine, 2-(Methylamino)-3-nitropyridine, PubChem16597, AC1LBE5W, SureCN2222503, AC1Q40Z6, CTK6I5039, methyl(3-nitro(2-pyridyl))amine, MolPort-001-757-628, N-methyl-3-nitro-pyridin-2-amine, AC1Q2086, BTB09509, 2-Pyridinamine, N-methyl-3-nitro-, ANW-60776, AR-1K7567, SBB086903, ZINC19738644, AKOS001874553, AG-B-37322
InChIKey: SILGRKFIVIVPKA-UHFFFAOYSA-N | ||||||||
| • N-Tert-Butoxycarbonyl-4-(4-Toluenesulfonyloxymethyl)Piperidine
IUPAC Name: tert-butyl 4-[(4-methylphenyl)sulfonyloxymethyl]piperidine-1-carboxylate | CAS Registry Number: 166815-96-9 Synonyms: N-Boc-4-(4-Toluenesulfonyloxymethyl)piperidine, N-TERT-BUTOXYCARBONYL-4-(4-TOLUENESULFONYLOXYMETHYL)PIPERIDINE, F2167-0074, tert-butyl 4-({[(4-methylphenyl)sulfonyl]oxy}methyl)piperidine-1-carboxylate, PubChem23416, AC1Q2LQW, AGN-PC-0CTN17, KSC532I5J, CTK4D2454, MolPort-003-823-749, ACT05192, ANW-50316, STL357534, ZINC02563761, AKOS005174069, AG-E-16214, MCULE-5860712597, AK-17106, BR-17106, KB-35282
InChIKey: DARTVAOOTJKHQW-UHFFFAOYSA-N | ||||||||
| • N2,N2-dimethyl-2,6-Pyridinediamine
IUPAC Name: 6-N,6-N-dimethylpyridine-2,6-diamine | CAS Registry Number: 63763-86-0 Synonyms: 2-N,2-N-dimethylpyridine-2,6-diamine, SCHEMBL1097604, 2-amino-6-dimethylaminopyridine, 6-dimethylamino-2-amino pyridine, MolPort-027-633-159, QFUOHXVQTQKZRB-UHFFFAOYSA-N, AKOS006338873, NE16310, SC-87667, DB-073392
InChIKey: QFUOHXVQTQKZRB-UHFFFAOYSA-N | ||||||||
| • N2-METHYL-PYRIDINE-2,3-DIAMINE
IUPAC Name: 2-N-methylpyridine-2,3-diamine | CAS Registry Number: 5028-20-6 Synonyms: N2-Methylpyridine-2,3-diamine, N2-Methyl-2,3-pyridinediamine, SureCN2947216, 2-N-methylpyridine-2,3-diamine, CTK4J2385, (3-amino(2-pyridyl))methylamine, MolPort-003-726-662, N~2~-methylpyridine-2,3-diamine, ANW-60988, SBB079410, STL155428, ZINC19770005, AKOS005202681, AG-L-23423, MCULE-8846074671, QC-1009, AK-74048, KB-85745, BB 0257209, FT-0681483
InChIKey: COANMWJRJDRXNS-UHFFFAOYSA-N | ||||||||
| • N2-methylpyridine-2,3-diamine
IUPAC Name: 2-N-methylpyridine-2,3-diamine
InChIKey: COANMWJRJDRXNS-UHFFFAOYSA-N | ||||||||
| • Nafamostat mesylate
IUPAC Name: (6-carbamimidoylnaphthalen-2-yl) 4-(diaminomethylideneamino)benzoate; methanesulfonic acid | CAS Registry Number: 82956-11-4 Synonyms: Futhan, Nafamstat, Ronastat, nafamostat mesilate, Nafamstat Mesilate, Ronastat (TN), Nafamostat mesilate (JAN), Nafamostat mesylate (USAN), FUT-175, CID5311180, D01670, 6-Amidino-2-naphthyl-4-guanidinobenzoate Dimethanesulfonate
InChIKey: SRXKIZXIRHMPFW-UHFFFAOYSA-N | ||||||||
| • Navitoclax
IUPAC Name: 4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-morpholin-4-yl-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide | CAS Registry Number: 923564-51-6 Synonyms: ABT-263, ABT 263, CHEBI:608147, 1000696-69-4, 4-(4-{[2-(4-chlorophenyl)-5,5-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-N-({4-({(1R)-3-morpholin-4-yl-1-[(phenylsulfanyl)methyl]propyl}amino)-3-[(trifluoromethyl)sulfonyl]phenyl}sulfonyl)benzamide, Benzamide, 4-(4-((2-(4-chlorophenyl)-5,5-dimethyl-1-cyclohexen-1-yl)methyl)-1-piperazinyl)-N-((4-(((1R)-3-(4-morpholinyl)-1-((phenylthio)methyl)propyl)amino)-3-((trifluoromethyl)sulfonyl)phenyl)sulfonyl)-
InChIKey: JLYAXFNOILIKPP-KXQOOQHDSA-N | ||||||||
| • Necrostatin-1
IUPAC Name: 5-(1H-indol-3-ylmethyl)-3-methyl-2-sulfanylideneimidazolidin-4-one | CAS Registry Number: 4311-88-0 Synonyms: MTH-DL-Tryptophan, MTH-trp, Nec-1, nchembio.83-comp1, nchembio711-1, methyl-thiohydantoin-tryptophan, Oprea1_645908, CBDivE_006695, Bio-0868, N9037_SIGMA, Necroptotic Inhibitor, Nec-1, methylthiohydantoin-DL-tryptophan, CHEBI:430803, MolPort-002-131-513, IN1207, CID2828334, NCGC00092372-01, NCGC00092372-02, 5-(Indol-3-ylmethyl)-(2-thio-3-methyl)hydantoin, 5-(indol-3-ylmethyl)-3-methyl-2-thio-Hydantoin
InChIKey: TXUWMXQFNYDOEZ-UHFFFAOYSA-N | ||||||||
| • Nedaplatin
IUPAC Name: azanide; 2-hydroxyacetic acid; platinum(2+) | CAS Registry Number: 95734-82-0 Synonyms: Aqupla, Nedaplatin [INN], Aqupla (TN), CGDP-II, Nedaplatin (JAN/INN), C2H6N2O3Pt, cis-Diammine(glycolato)platinum, CCRIS 4088, cis-Diammine (glycolato)platinum, cis-Diammine(glycolato)platinum(II), NSC 375101D, cis-diammine(glycolato)platinum II, (Glycolato-O,O')diammineplatinum(II), NSC-375101D, (glycolato-O,O')diammineplatinum II, 254-S, NCGC00181152-01, LS-117704, C12862, cis-Diammine(glycolato-O(sup 1),O(sup 2))platinum
InChIKey: KLNFSAOEKUDMFA-UHFFFAOYSA-N | ||||||||
| • Neflamapimod
IUPAC Name: 5-(2,6-dichlorophenyl)-2-(2,4-difluorophenyl)sulfanylpyridazino[6,1-f]pyrimidin-6-one | CAS Registry Number: 209410-46-8 Synonyms: VX-745, CID3038525, 5-(2,6-Dichlorophenyl)-2-((2,4-difluorophenyl)thio)-6H-pyrimido(1,6-b)pyridazin-6-one, 6H-Pyrimido(1,6-b)pyridazin-6-one, 5-(2,6-dichlorophenyl)-2-((2,4-difluorophenyl)thio)-
InChIKey: VEPKQEUBKLEPRA-UHFFFAOYSA-N | ||||||||
| • Neratinib
IUPAC Name: (E)-N-[4-[3-chloro-4-(pyridin-2-ylmethoxy)anilino]-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)but-2-enamide | CAS Registry Number: 698387-09-6 Synonyms: HKI-272, HKI 272, Neratinib(HKI-272), Neratinib, HKI-272, 698387-09-6, HKI272, HKI 272, HKI-272,, (2E)-N-[4-[[3-chloro-4-[(pyridin-2-yl)methoxy]phenyl]amino]-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)but-2-enamide, HKI272, S2150_Selleck, Neratinib HKI 272, PubChem22399, Neratinib (INN/USAN), UNII-JJH94R3PWB, Neratinib - HKI-272, cc-32, SureCN571762, JSPY-st000262, CHEMBL180022, QCR-104, CHEBI:399120, MolPort-006-069-389
InChIKey: JWNPDZNEKVCWMY-VQHVLOKHSA-N | ||||||||
| • Niclosamide
IUPAC Name: 5-chloro-N-(2-chloro-4-nitrophenyl)-2-hydroxybenzamide | CAS Registry Number: 50-65-7 Synonyms: niclosamide, Niclocide, Bayluscid, Devermine, Dichlosale, Helmiantin, Tredemine, Cestocid, Devermin, Mansonil, Phenasal, Radeverm, Vermitid, Vermitin, Atenase, Fenasal, Iomesan, Iomezan, Sagimid, Yomesan
InChIKey: RJMUSRYZPJIFPJ-UHFFFAOYSA-N | ||||||||
| • Nicotinylchloride
IUPAC Name: pyridine-3-carbonyl chloride | CAS Registry Number: 10400-19-8 Synonyms: Nicotinoyl chloride, 3-Pyridinecarbonyl chloride, MolPort-001-781-839, CID82604, EINECS 233-863-9, SBB005806, ZINC02539499, I02-0326, 20260-53-1
InChIKey: ATBIAJXSKNPHEI-UHFFFAOYSA-N | ||||||||
| • Nilotinib
IUPAC Name: 4-methyl-N-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]benzamide | CAS Registry Number: 641571-10-0 Synonyms: AMN107, AMN 107, CHEBI:52172, AMN-107, TL8004531, 4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]benzamide, 4-Methyl-3-((4-(3-pyridinyl)-2-pyrimidinyl)amino)-N-(5-(4-methyl-1H-imidazol-1-yl)-3-(trifluoromethyl)phenyl)benzamide, 4-Methyl-3-(4-(3-pyridinyl)-2-pyrimidinyl)amino)-N-[5-(4-methyl-1H-imidazol-1-yl)-3-(trifluoromethyl)phenyl]benzamide, 4-Methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]-N-[5-(4-methyl-1H-imidazol-1-yl)-3-(trifluoromethyl)phenyl]benzamide, Benzamide, 4-methyl-N-((3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-3-(4-(3-pyridinyl)-2-pyrimidinyl)amino)-, Benzamide, 4-methyl-N-(3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-3-(4-(3-pyridinyl)-2-pyrimidinyl)amino)-, benzamide, 4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]-, Benzamide, 4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]- (9CI), NIL
InChIKey: HHZIURLSWUIHRB-UHFFFAOYSA-N | ||||||||
| • Nimodipine
IUPAC Name: 5-O-(2-methoxyethyl) 3-O-propan-2-yl 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate | CAS Registry Number: 66085-59-4 Synonyms: nimodipine, Nimotop, Periplum, Admon, Remontal, Brainal, Kenesil, Calnit, Modus, Nimodipin Hexal, NimodipinISIS, Nimodipin ISIS, Nimodipin-ISIS, Nimodipino Bayvit, Nimotop(TM), nchembio.79-comp6, Nimodipinum [INN-Latin], Nimodipino [INN-Spanish], Spectrum_001880, SpecPlus_000716
InChIKey: UIAGMCDKSXEBJQ-UHFFFAOYSA-N | ||||||||
| • Nintedanib
IUPAC Name: methyl (3Z)-3-[[4-[methyl-[2-(4-methylpiperazin-1-yl)acetyl]amino]anilino]-phenylmethylidene]-2-oxo-1H-indole-6-carboxylate | CAS Registry Number: 656247-17-5 Synonyms: Vargatef, BIBF-1120, BIBF1120, 928326-83-4, BIBF 1120, Vargatef, BIBF1120, (Z)-methyl 3-((4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenylamino)(phenyl)methylene)-2-oxoindoline-6-carboxylate, S1010_Selleck, BIBF1120,Vargatef, PubChem20543, Bibf1120 - Vargatef, Nintedanib (USAN/INN), Vargatef, BIBF 1120, cc-88, SureCN431006, CHEMBL502835, QCR-43, CHEBI:622730, RS0107, AKOS005145820
InChIKey: XZXHXSATPCNXJR-ZIADKAODSA-N | ||||||||
| • Nithiamide
IUPAC Name: N-(5-nitro-1,3-thiazol-2-yl)acetamide | CAS Registry Number: 140-40-9 Synonyms: Aminitrozole, Nitazole, Tricogen, Tritheon, Gynofon, Nitasol, Acinitrazole, Ametoterina, Aminitrazol, Aminitrozol, Tricosteril, Lavoflagin, Trichlorad, Trichocid, Trichoman, Trichorad, Trichoral, Tricolaval, Trikolaval, Pleocide
InChIKey: UJRRDDHEMZLWFI-UHFFFAOYSA-N | ||||||||
| • Nitrendipine
IUPAC Name: 3-O-ethyl 5-O-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate | CAS Registry Number: 39562-70-4 Synonyms: nitrendipine, Baypress, Bayotensin, Nidrel, Nitrendimerck, Baylotensin, Nitregamma, Nitrendepat, Nitrendidoc, Nitrendipin, Nitrepress, Tensogradal, Vastensium, Balminil, Baypresol, Jutapress, Nitrensal, Trendinol, Gericin, Niprina
InChIKey: PVHUJELLJLJGLN-UHFFFAOYSA-N | ||||||||
| • Nitromalonaldehyde Sodium
IUPAC Name: 2-nitropropanedial | CAS Registry Number: 34461-00-2 Synonyms: MolPort-001-781-578, CID313475, NSC152527, NSC191937, NSC227850, STT-00282693, 609-32-5
InChIKey: WQDQLOXQQUFECI-UHFFFAOYSA-N | ||||||||
| • Nocodazole
IUPAC Name: methyl N-[6-(thiophene-2-carbonyl)-1H-benzimidazol-2-yl]carbamate | CAS Registry Number: 31430-18-9 Synonyms: nocodazole, Oncodazole, Nocodazolum, Nocidazole, Nocodazol, Prestwick_359, nchembio.63-comp4, nchembio.100-comp7, nchembio.90-comp11, Nocodazol [INN-Spanish], Nocodazolum [INN-Latin], Tocris-1228, Nocodazole (USAN/INN), Nocodazole [USAN:INN], Prestwick0_000100, Prestwick1_000100, Prestwick2_000100, Prestwick3_000100, Spectrum3_001768, Spectrum4_001060
InChIKey: KYRVNWMVYQXFEU-UHFFFAOYSA-N | ||||||||
| • Nodinitib-1
IUPAC Name: 1-(4-methylphenyl)sulfonylbenzimidazol-2-amine | CAS Registry Number: 799264-47-4 Synonyms: ML130, BAS 07162070, 1-(Toluene-4-sulfonyl)-1H-benzoimidazol-2-ylamine, SMR000523991, Noditinib-1, ZINC00807071, AC1LLPTT, SureCN10107599, MLS001201458, MLS002639479, CHEMBL1412853, MolPort-002-008-875, HMS2819O03, CCG-25324, AKOS000641831, MCULE-7249710756, FT-0673025, 1-(4-methylphenyl)sulfonylbenzimidazol-2-amine, MLS-0350096.0001, MLS-0350096.0002
InChIKey: SRFABRWQVPCPRG-UHFFFAOYSA-N | ||||||||
| • NSC 405020
IUPAC Name: 3,4-dichloro-N-pentan-2-ylbenzamide | CAS Registry Number: 7497-07-6 Synonyms: ST50721491, NSC405020, AC1L85MV, MolPort-001-510-886, STK029746, 3,4-dichloro-N-pentan-2-ylbenzamide, AKOS003260207, LS41106, MCULE-6949455563, NSC-405020, 3,4-dichloro-N-(pentan-2-yl)benzamide, (3,4-dichlorophenyl)-N-(methylbutyl)carboxamide
InChIKey: ARDYECYBETXQFD-UHFFFAOYSA-N | ||||||||
| • NSC 66811
IUPAC Name: 7-[anilino(phenyl)methyl]-2-methylquinolin-8-ol | CAS Registry Number: 6964-62-1 Synonyms: NSC-66811, 7-(anilino(phenyl)methyl)-2-methyl-8-quinolinol, 7-(Anilino(phenyl)-methyl)-2-methyl-8-quinolinol, 2-methyl-7-[phenyl(phenylamino)methyl]quinolin-8-ol, NSC66811, AC1L6NIN, AC1Q79MP, SureCN1241576, CHEMBL210778, CTK5D0724, AR-1H2750, DNC006772, AKOS003020553, AG-K-29451, VU0452053-1, 7-[anilino(phenyl)methyl]-2-methylquinolin-8-ol, 2-methyl-7-(phenyl-phenylamino)methyl) quinolin-8-ol, 8-Quinolinol,2-methyl-7-[phenyl(phenylamino)methyl]-, S4923,NSC66811,6964-62-1, 2-METHYL-7-[PHENYL(PHENYLAMINO)METHYL]-8-QUINOLINOL
InChIKey: WEENRMPCSWFMTE-UHFFFAOYSA-N | ||||||||
| • NSC632839
IUPAC Name: (3E,5E)-3,5-bis[(4-methylphenyl)methylidene]piperidin-4-one;hydrochloride | CAS Registry Number: 157654-67-6 Synonyms: NSC-632839, MLS002701647, AC1NS0DO, S4922,NSC632839,157654-67-6, 4-Piperidinone,5-bis[(4-methylphenyl)methylene]-, hydrochloride, (3E,5E)-3,5-bis[(4-methylphenyl)methylidene]piperidin-4-one hydrochloride, 3,5-BIS[(4-METHYLPHENYL)METHYLENE]-4-PIPERIDONE HYDROCHLORIDE
InChIKey: ZOKZLTXPTLIWOJ-BYCVLTJGSA-N | ||||||||
| • NU 7026
IUPAC Name: 2-morpholin-4-ylbenzo[h]chromen-4-one | CAS Registry Number: 154447-35-5 Synonyms: NU7026, DNA-PK Inhibitor II, 2-(Morpholin-4-yl)-benzo[h]chromen-4-one, 2-morpholino-4H-benzo[h]chromen-4-one, LY293646, DNA-Dependent Protein Kinase Inhibitor II, LY-293646, SureCN610237, cc-674, CHEMBL104468, CTK0E7833, CHEBI:270938, MolPort-009-019-548, HMS3229C11, DNC000625, DNC001049, DNC003945, HSCI1_000223, IN1364, AKOS015994580
InChIKey: KKTZALUTXUZPSN-UHFFFAOYSA-N | ||||||||
| • NU6027
IUPAC Name: 6-(cyclohexylmethoxy)-5-nitrosopyrimidine-2,4-diamine | CAS Registry Number: 220036-08-8 Synonyms: 4-cyclohexylmethoxy-5-nitrosopyrimidine-2,6-diamine, 6-CYCLOHEXYLMETHYLOXY-5-NITROSO-PYRIMIDINE-2,4-DIAMINE, 6-(cyclohexylmethoxy)-5-nitrosopyrimidine-2,4-diamine, NW1, 1e1x, AC1L9FZU, MLS001074890, N4411_SIGMA, AC1Q53K2, CHEMBL303958, CTK0J6897, HMS2234C12, HMS3263D06, AR-1G2051, DNC004110, NSC707616, DB08312, LP01212, NSC-707616, NCGC00165844-01
InChIKey: DGWXOLHKVGDQLN-UHFFFAOYSA-N | ||||||||
| • Nutlin-3a
IUPAC Name: 4-[(4S,5R)-4,5-bis(4-chlorophenyl)-2-(4-methoxy-2-propan-2-yloxyphenyl)-4,5-dihydroimidazole-1-carbonyl]piperazin-2-one | CAS Registry Number: 675576-98-4 Synonyms: nutlin-3A, Nutlin 3a, nutlin 3, Nutlin-3a chiral, SureCN1155752, UNII-L7C92IOE65, cc-452, CHEMBL191334, S8059,(-)-Nutlin-3, CHEBI:417700, MolPort-009-019-256, DNC006637, BCP9001003, CS-0296, RL04569, HY-10029, Nutlin-3a chiral|675576-98-4|Nutlin 3a, 2-Piperazinone, 4-(((4S,5R)-4,5-bis(4-chlorophenyl)-4,5-dihydro-2-(4-methoxy-2-(1-methylethoxy)phenyl)-1H-imidazol-1-yl)carbonyl)-
InChIKey: BDUHCSBCVGXTJM-WUFINQPMSA-N | ||||||||
| • Nutlin-3b
IUPAC Name: 4-[(4R,5S)-4,5-bis(4-chlorophenyl)-2-(4-methoxy-2-propan-2-yloxyphenyl)-4,5-dihydroimidazole-1-carbonyl]piperazin-2-one | CAS Registry Number: 675576-97-3 Synonyms: nutlin-3B, CHEMBL2152332, CHEBI:46742, nutlin 3, Nutlin3, UNII-FJA1772CVW, SureCN13233382, Nutlin-3b|675576-97-3, BCP9001004, CS-0295, CS-0727, Nutlin-3|548472-68-0|Nutlin3, NCGC00263124-01, HY-15335, HY-50696, 2-Piperazinone, 4-(((4R,5S)-4,5-bis(4-chlorophenyl)-4,5-dihydro-2-(4-methoxy-2-(1-methylethoxy)phenyl)-1H-imidazol-1-yl)carbonyl)-, cis-4-{[4,5-bis(4-chlorophenyl)-2-(2-isopropoxy-4-methoxyphenyl)-4,5-dihydroimidazol-1-yl]carbonyl}piperazin-2-one, rel-4-{[(4R,5S)-4,5-bis(4-chlorophenyl)-2-{2-[(propan-2-yl)oxy]-4-methoxyphenyl}-4,5-dihydro-1H-imidazol-1-yl]carbonyl}piperazin-2-one
InChIKey: BDUHCSBCVGXTJM-IZLXSDGUSA-N | ||||||||
| • NVP-ADW742
IUPAC Name: 5-(3-phenylmethoxyphenyl)-7-[3-(pyrrolidin-1-ylmethyl)cyclobutyl]pyrrolo[2,3-d]pyrimidin-4-amine | CAS Registry Number: 475488-23-4 Synonyms: ADW742, NVP-ADW742, S1088_Selleck, Kinome_2540, SureCN95142, SureCN1983470, SureCN1983472, cc-532, ADW742, CHEMBL399021, CHEBI:513409, MolPort-016-633-174, GSK 552602A, DNC001052, BCP9001005, CS-0450, RL03774, NCGC00346485-01, HY-10252, NVP-ADW742-Supplied by Selleck Chemicals, X7472
InChIKey: LSFLAQVDISHMNB-UHFFFAOYSA-N | ||||||||
| • NVP-AEW541
IUPAC Name: 7-[3-(azetidin-1-ylmethyl)cyclobutyl]-5-(3-phenylmethoxyphenyl)pyrrolo[2,3-d]pyrimidin-4-amine | CAS Registry Number: 475489-16-8 Synonyms: AEW-541, AEW541, AEW 541, 475488-34-7, SureCN94862, AGN-PC-009VBF, SureCN1441421, SureCN1987652, NVP AEW541, cc-535, NVP-AEW 541, UNII-97QB5037VR, CTK4J0098, BCPP000146, DCL000364, AG-F-61825, BCP9001006, CS-0448, PB19343, RL03775
InChIKey: AECDBHGVIIRMOI-UHFFFAOYSA-N | ||||||||
| • NVP-BHG712
IUPAC Name: 4-methyl-3-[(1-methyl-6-pyridin-3-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]-N-[3-(trifluoromethyl)phenyl]benzamide | CAS Registry Number: 940310-85-0 Synonyms: 940310-85-0 , NVP BHG712, 4-Methyl-3-[[1-methyl-6-(3-pyridinyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino]-N-[3-(trifluoromethyl)phenyl]benzamide, S2202_Selleck, NVPBHG712, AGN-PC-015AWW, SureCN4699731, cc-540, NVP BHG 712, QCR-258, MolPort-016-633-311, BCP9001010, CS-0469, RL05902, NCGC00249391-01, HY-13258, KB-58915, NVP-BHG712-Supplied by Selleck Chemicals, X7502, NVP-BHG712|940310-85-0|NVP BHG 712, 4-methyl-3-(1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-ylamino)-N-(3-(trifluoromethyl)phenyl)benzamide
InChIKey: ZCCPLJOKGAACRT-UHFFFAOYSA-N | ||||||||
| • NVP-BSK805
IUPAC Name: 4-[[2,6-difluoro-4-[3-(1-piperidin-4-ylpyrazol-4-yl)quinoxalin-5-yl]phenyl]methyl]morpholine;dihydrochloride | CAS Registry Number: 1092499-93-8 Synonyms: 1092499-93-8 pound not NVP BSK805, NVP-BSK805 2HCl, NVP-BSK805 dihydrochloride, cc-625, NVP-GSK 805, NVP-BSK805/NVPBSK805, BCP9001012, BCP0726000306, X7514, 8-(3,5-difluoro-4-(morpholinomethyl)phenyl)-2-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)quinoxaline, 8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-[1-(piperidin-4-yl)pyrazol-4-yl]quinoxaline dihydrochloride
InChIKey: NUOCAPALWRHKCU-UHFFFAOYSA-N | ||||||||
| • NVP-BVU972
IUPAC Name: 6-[[6-(1-methylpyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl]quinoline | CAS Registry Number: 1185763-69-2 Synonyms: 3qti, NVPBVU972, SureCN1659100, NVP BVU972, cc-601, BVU972, BCP9000466, CS-0967, NCGC00346689-01, HY-15456, BCP0726000188, NVP-BVU972|1185763-69-2, 958025-66-6 , C20H16N6 , NVP BVU972
InChIKey: RNCNPRCUHHDYPC-UHFFFAOYSA-N | ||||||||
| • NVP-TAE 226
IUPAC Name: 2-[[5-chloro-2-(2-methoxy-4-morpholin-4-ylanilino)pyrimidin-4-yl]amino]-N-methylbenzamide | CAS Registry Number: 761437-28-9 Synonyms: 2-((5-Chloro-2-((2-methoxy-4-morpholinophenyl)amino)pyrimidin-4-yl)amino)-N-methylbenzamide, 2-({5-Chloro-2-[(2-Methoxy-4-Morpholin-4-Ylphenyl)amino]pyrimidin-4-Yl}amino)-N-Methylbenzamide, 2jkk, 2-[5-chloro-2-(2-methoxy-4-morpholin-4-yl-phenylamino)-pyrimidin-4-ylamino]-N-methyl-benzamide, Kinome_1212, SureCN375524, NVP-TAE226, CHEMBL458997, TAE226, CTK8B9478, CHEBI:614994, ANW-62587, AKOS016004135, CS-0594, DB07460, NCGC00346931-01, AK101877, HY-13203, NVP-TAE 226,CAS:761437-28-9, NVP-TAE 226|761437-28-9
InChIKey: UYJNQQDJUOUFQJ-UHFFFAOYSA-N | ||||||||
| • NVP-TAE 684
IUPAC Name: 5-chloro-2-N-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-4-N-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | CAS Registry Number: 761439-42-3 Synonyms: NVP-TAE684, TAE684, TAE-684, 5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine, TAE684, 761439-42-3, TAE684, NVP-TAE684, GUI, S1108_Selleck, Kinome_1205, PubChem16769, cc-17, SureCN282775, AGN-PC-00RX8K, NVP TAE684, UNII-EH1713MN4K, NVP TAE 684, NVT-TAE-684, CHEMBL509032, TAE 684, CHEBI:547450
InChIKey: QQWUGDVOUVUTOY-UHFFFAOYSA-N | ||||||||
| • Obatoclax Mesylate
IUPAC Name: 2-[(5Z)-5-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-4-methoxypyrrol-2-ylidene]indole;methanesulfonic acid | CAS Registry Number: 803712-79-0 Synonyms: Obatoclax mesylate, ACT06786
InChIKey: ZVAGBRFUYHSUHA-RKMKAUCSSA-N | ||||||||
| • Omeprazole
IUPAC Name: 6-methoxy-2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methylsulfinyl]-1H-benzimidazole | CAS Registry Number: 73590-58-6 Synonyms: omeprazole, Prilosec, Antra, Losec, Omeprazon, Audazol, Omapren, Omepral, Parizac, Mopral, Miol, Demeprazol, Inhibitron, Ulcometion, Belmazol, Ceprandal, Dizprazol, Dudencer, Emeproton, Epirazole
InChIKey: SUBDBMMJDZJVOS-UHFFFAOYSA-N | ||||||||
| • Omipalisib
IUPAC Name: 2,4-difluoro-N-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamide | CAS Registry Number: 1086062-66-9 Synonyms: GSK2126458, GSK 2126458, GSK-2126458, 2,4-Difluoro-N-[2-methoxy-5-[4-(4-pyridazinyl)-6-quinolinyl]-3-pyridinyl]benzenesulfonamide, 2,4-difluoro-N-(2-methoxy-5-(4-(pyridazin-4-yl)quinolin-6-yl)pyridin-3-yl)benzenesulfonamide, GSK212, GSK 212, GSK-212, 2,4-difluoro-N-{2-methoxy-5-[4-(pyridazin-4-yl)quinolin-6-yl]pyridin-3-yl}benzenesulfonamide, PubChem22430, cc-65, SureCN623194, UNII-1X8F5A3NA0, GSK-458, 3l08, ABP000103, AKOS015904655, CS-0085, QC-7243, RL00368
InChIKey: CGBJSGAELGCMKE-UHFFFAOYSA-N | ||||||||
| • ON-01910
IUPAC Name: sodium;2-[2-methoxy-5-[[(E)-2-(2,4,6-trimethoxyphenyl)ethenyl]sulfonylmethyl]anilino]acetate | CAS Registry Number: 1225497-78-8 Synonyms: Novonex, Estybon, Rigosertib sodium, Estybon, ON-01910, ON 01910, Estybon, ON-01910, 1225497-78-8, 592542-60-4, S1362_Selleck, Rigosertib sodium (USAN), ON 01910 sodium salt, cc-628, ON-1910Na, Onc-01910, CHEMBL2013119, ON-01910Na, SyB C-1101, SyB L-1101, MolPort-016-633-202, ON 01910.Na, BCP9001024
InChIKey: VLQLUZFVFXYXQE-USRGLUTNSA-M | ||||||||
| • Onalespib
IUPAC Name: (2,4-dihydroxy-5-propan-2-ylphenyl)-[5-[(4-methylpiperazin-1-yl)methyl]-1,3-dihydroisoindol-2-yl]methanone | CAS Registry Number: 912999-49-6 Synonyms: AT13387, AT-13387, SureCN382780, AGN-PC-00IPH6, UNII-Q7Y33N57ZZ, CHEMBL1214827, BCP9000333, CS-0969, NCGC00346674-01, AT 13387, HY-14463, BCP0726000186, AT13387|912999-49-6|AT-13387, AT-13387;AT13387;AT 13387;912999-49-6, (2,4-Dihydroxy-5-isopropylphenyl)-(5-(4-methylpiperazin-1-ylmethyl)-1,3-dihydroisoindol-2-yl)methanone, (2,4-dihydroxy-5-propan-2-ylphenyl)-[5-[(4-methylpiperazin-1-yl)methyl]-1,3-dihydroisoindol-2-yl]methanone, Methanone, (1,3-dihydro-5-((4-methyl-1-piperazinyl)methyl)-2H-isoindol-2-yl)(2,4-dihydroxy-5-(1-methylethyl)phenyl)-
InChIKey: IFRGXKKQHBVPCQ-UHFFFAOYSA-N | ||||||||
| • ONX-0914
IUPAC Name: (2S)-3-(4-methoxyphenyl)-N-[(2S)-1-(2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-yl]-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide | CAS Registry Number: 960374-59-8 Synonyms: QC-7242, (2S)-3-(4-methoxyphenyl)-N-((2S)-1-(2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-yl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
InChIKey: WQAVPPWWLLVGFK-ZCKRSBOQSA-N | ||||||||
| • Oprozomib
IUPAC Name: N-[(2S)-3-methoxy-1-[[(2S)-3-methoxy-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]-2-methyl-1,3-thiazole-5-carboxamide | CAS Registry Number: 935888-69-0 Synonyms: ONX-0912, Oprozomib [USAN], Oprozomib (USAN/INN), UNII-MZ37792Y8J, CHEMBL2103884, ONX 0912, PR-047, QC-9273, NCGC00345799-01, D10318, L-Serinamide, O-methyl-N-((2-methyl-5-thiazolyl)carbonyl)-L-seryl-O-methyl-N-((1S)-2- ((2R)-2-methyl-2-oxiranyl)-2-oxo-1-(phenylmethyl)ethyl)-, N-((S)-3-methoxy-1-((S)-3-methoxy-1-((S)-1-((R)-2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-2-methylthiazole-5-carboxamide, O-Methyl-N-((2-methylthiazol-5-yl)carbonyl)-L-seryl-O-methyl-N-((1S)-1-benzyl-2-((2R)- 2-methyloxiran-2-yl)-2-oxoethyl)-L-serinamide
InChIKey: SWZXEVABPLUDIO-WSZYKNRRSA-N | ||||||||
| • Orantinib
IUPAC Name: 3-[2,4-dimethyl-5-[(E)-(2-oxo-1H-indol-3-ylidene)methyl]-1H-pyrrol-3-yl]propanoic acid | CAS Registry Number: 252916-29-3 Synonyms: TSU68, TSU 68, SU6668, CID5995546, NSC 702827, SU 6668, SU-6668, 3-(4-(2-Carboxyethyl)-3,5-dimethylpyrrol-2-methylidenyl)-2-indolinone, 3-(2,4-Dimethyl-5-(2-oxo-1,2-dihydroindol-3-ylidenemethyl)-1H-pyrrol-3-yl)propionic acid, 1H-Pyrrole-3-propanoic acid, 5-((1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-2,4-dimethyl-, 245036-27-5, 3-(2,4-Dimethyl-5-((2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl)-1H-pyrrol-3-yl)propionic acid, 3-{2,4-dimethyl-5-[(E)-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-1H-pyrrol-3-yl}propanoic acid, 5-((1,2-Dihydro-2-oxo-3H-indol-3-ylidene)methyl)-2,4-dimethyl-1H-pyrrole-3-propanoic acid
InChIKey: NHFDRBXTEDBWCZ-NTEUORMPSA-N | ||||||||
| • OSI-027
IUPAC Name: 4-[(5Z)-4-amino-5-(7-methoxyindol-2-ylidene)-1H-imidazo[5,1-f][1,2,4]triazin-7-yl]cyclohexane-1-carboxylic acid | CAS Registry Number: 936890-98-1 Synonyms: OSI027, OSI 027, OSI027, OSI-027, K1146_Kinasechem, S2624_Selleck, Cyclohexanecarboxylic acid, 4-(4-amino-5-(7-methoxy-1H-indol-2-yl)imidazo(5,1-f)(1,2,4)triazin-7-yl)-, trans-, UNII-25MKH1SZ0M, cc-501, BCP9001034, CS-0257, HY-10423, OSI-027|936890-98-1|OSI 027, OSI 027, OSI-027, 936890-98-1, OSI 027, OSI-027, 936890-98-1, (+/-)-Cyclohexanecarboxylic acid, 4-(4-amino-5-(7-methoxy-1H-indol-2-yl)imidazo(5,1-f)(1,2,4)triazin-7-yl)-, trans-, (1r,4r)-4-[4-amino-5-(7-methoxy-1H-indol-2-yl)imidazo[4,3-f][1,2,4]triazin-7-yl]cyclohexane-1-carboxylic acid
InChIKey: CDNMDRUIGNHEMR-VKAVYKQESA-N | ||||||||
| • OSI-930
IUPAC Name: 3-(quinolin-4-ylmethylamino)-N-[4-(trifluoromethoxy)phenyl]thiophene-2-carboxamide | CAS Registry Number: 728033-96-3 Synonyms: OSI930, S1220_Selleck, OSI 930, CHEMBL1614710, OSI-930 is a multi-targeted tyrosine kinase inhibitor, 3-[(4-Quinolinylmethyl)amino]-N-[4-(trifluoromethoxy)phenyl]-2-thiophenecarboxamide, CID9868037, SureCN633719, cc-339, DCL000352, BCP9001037, CS-0174, RL04771, 3-(quinolin-4-ylmethylamino)-N-[4-(trifluoromethoxy)phenyl]thiophene-2-carboxamide, OSI-930-Supplied by Selleck Chemicals, NCGC00263159-01, HY-10204, X7484, OSI-930|728033-96-3|OSI930, 3-[(quinolin-4-ylmethyl)amino]-N-[4-(trifluoromethoxy)phenyl]thiophene-2-carboxamide
InChIKey: FGTCROZDHDSNIO-UHFFFAOYSA-N | ||||||||
| • Osu03012
IUPAC Name: 2-amino-N-[4-[5-phenanthren-2-yl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]acetamide | CAS Registry Number: 742112-33-0 Synonyms: OSU-03012, CHEMBL1650595, OSU03012, OSU03012, OSU 03012, 742112-33-0, 2-amino-N-(4-(5-(phenanthren-2-yl)-3-(trifluoromethyl)-1H-pyrazol-1-yl)phenyl)acetamide, N/AAR-12, OSU03012, OSU-03012, S1106_Selleck, PubChem22592, PDK1 inhibitor AR-12, UNII-EX3O2Q61UV, cc-115, MolPort-009-019-120, BCPP000134, ABP000481, BCP9001039, CS-0151, RL04816, RL04817, NCGC00346490-01, HY-10547
InChIKey: YULUCECVQOCQFQ-UHFFFAOYSA-N |