Profile: Jinan Trio PharmaTech Co., Ltd. specializes in APIs & intermediates, heterocyclic compounds, and anti-tumor drugs. Our products include crizotinib, vemurafenib, afatinib, vandetanib, regorafenib, brivanib alaninate, pyridazine, imidazole, pyrazole, and oxazole. We are specialized in providing over 1000 products including molecular targeted anticancer drugs, cell signaling pathway inhibitors, pharmaceutical intermediates, and heterocyclic compounds, and quality services including custom synthesis, transfer of new drug patent and technology, technical cooperation, and process optimization.
| • Danoprevir
Synonyms: Intermune ITMN-191, ITMN B, Danoprevir [USAN:INN], UNII-911Z9PCQ5F, R7227, ITMN 191, R 7227, R05190591, R 05190591, 1001913-18-3, 1225266-12-5, 916881-67-9
InChIKey: ZVTDLPBHTSMEJZ-QIFYYAQYSA-N | ||||||||
| • Danusertib
IUPAC Name: N-[5-[(2R)-2-methoxy-2-phenylacetyl]-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazol-3-yl]-4-(4-methylpiperazin-1-yl)benzamide | CAS Registry Number: 827318-97-8 Synonyms: 5-Amido-pyrrolopyrazole 9d, UNII-M3X659D0FY, 2j50, CHEBI:536278, PHA-739358, PHA 739358, CID11442891, CID 11994441, (R)-N-(5-(2-methoxy-2-phenylacetyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)-4-(4-methylpiperazin-1-yl)benzamide, Benzamide, 4-(4-methyl-1-piperazinyl)-N-(1,4,5,6-tetrahydro-5-((2R)- methoxyphenylacetyl)pyrrolo(3,4-c)pyrazol-3-yl)-
InChIKey: XKFTZKGMDDZMJI-HSZRJFAPSA-N | ||||||||
| • DAPT
IUPAC Name: tert-butyl (2S)-2-[[(2S)-2-[[2-(3,5-difluorophenyl)acetyl]amino]propanoyl]amino]-2-phenylacetate | CAS Registry Number: 208255-80-5 Synonyms: dapt, DAPT (GSI-IX), gamma-Secretase Inhibitor IX, DAPT, GSI-IX, InSolution™ gamma-Secretase Inhibitor IX, N-[N-(3,5-Difluorophenacetyl-L-alanyl)]-S-phenylglycine t-Butyl Ester, GSIIX, S2215_Selleck, AC1NSKCB, PubChem22436, GSI IX, GSI-IX, DAPT,GSI-IX, DAPT - GSI-IX, SureCN1360313, cc-201, CHEMBL255682, QCR-29, DAPT-Supplied by Selleck Chemicals, ABP000317
InChIKey: DWJXYEABWRJFSP-XOBRGWDASA-N | ||||||||
| • Darunavir Ethanolate
IUPAC Name: [(3R,3aS,6aR)-2,3,3a,4,5,6a-hexahydrofuro[2,3-b]furan-3-yl] N-[(2S,3R)-4-[(4-aminophenyl)sulfonyl-(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl]carbamate; ethanol | CAS Registry Number: 635728-49-3 Synonyms: Prezista, Darunavir ethanolate, Prezista (TN), Darunavir ethanolate (JAN), TMC 114, LS-186602, D06478, 635728-39-1, Carbamic acid, ((1S,2R)-3-(((4-aminophenyl)sulfonyl)(2-methylpropyl)amino)-2-hydroxy-1-(phenylmethyl)propyl)-, (3R,3aS,6aR)-hexahydrofuro(2,3-b)furan-3-yl ester, compd. with ethanol
InChIKey: QWSHKNICRJHQCY-VBTXLZOXSA-N | ||||||||
| • Dasatinib
IUPAC Name: N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide | CAS Registry Number: 302962-49-8 Synonyms: Sprycel, BMS Dasatinib, Dasatinib [USAN], Dasatinib (USAN), nchembio.117-comp11, SPRYCEL (TN), BMS-354825, BMS354825, BMS 354825, CHEBI:49375, NSC732517, CID3062316, DB01254, NSC-732517, NCGC00181129-01, BCB03_000715, LS-186641, LS-187028, LS-187773, D03658
InChIKey: ZBNZXTGUTAYRHI-UHFFFAOYSA-N | ||||||||
| • Dasatinib monohydrate
IUPAC Name: N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide hydrate | CAS Registry Number: 863127-77-9 Synonyms: Dasatinib hydrate, Dasatinib hydrate (JAN), D06414
InChIKey: XHXFZZNHDVTMLI-UHFFFAOYSA-N | ||||||||
| • DBEQ
IUPAC Name: 2-N,4-N-dibenzylquinazoline-2,4-diamine | CAS Registry Number: 177355-84-9 Synonyms: DBeQ, N,N'-dibenzylquinazoline-2,4-diamine, JRF12, JRF-12, N2,N4-dibenzylquinazoline-2,4-diamine, SMR002239188, AC1LDWFN, 2,4-dibencilaminoquinazoline, Oprea1_067556, Oprea1_526582, MLS003568133, MLS006012041, JRF 12, CHEMBL1624459, SCHEMBL12175837, STOCK3S-86339, MolPort-002-593-377, KUC105555N, CCG-24030, KSC-16-67
InChIKey: QAIMUUJJAJBPCL-UHFFFAOYSA-N | ||||||||
| • Decitabine
IUPAC Name: 4-amino-1-[(2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-1,3,5-triazin-2-one | CAS Registry Number: 2353-33-5 Synonyms: Dezocitidine, Dacogen, 5-Aza-2'-deoxycytidine, AzadC, 5-Azadeoxycytidine, 5-aza-CdR, 5-aza-dC, Dacogen (TN), 2'-Deoxy-5-azacytidine, 5A2dc, 5-aza-2-deoxycytidine, 5-AZAdC, NCGC_5ADOC, Decitabine (USAN/INN), MolMap_000063, MLS001332587, MLS001332588, A3656_SIGMA, 5-Aza-2′-Deoxycytidine, 5-Deoxy-2′-azacytidine
InChIKey: XAUDJQYHKZQPEU-KVQBGUIXSA-N | ||||||||
| • Degrasyn
IUPAC Name: (E)-3-(6-bromopyridin-2-yl)-2-cyano-N-[(1S)-1-phenylbutyl]prop-2-enamide | CAS Registry Number: 856243-80-6 Synonyms: WP1130, CHEMBL1923233, WP 1130, WP-1130, WP 1130, WP-1130, 856243-80-6, (S,E)-3-(6-bromopyridin-2-yl)-2-cyano-N-(1-phenylbutyl)acrylamide, WP1130 - Adooq Bioscience, QCR-21, CS-0483, HY-13264, KB-81491, X7509, WP1130|856243-80-6|WP 1130|WP-1130, (2E)-3-(6-bromopyridin-2-yl)-2-cyano-N-[(1S)-1-phenylbutyl]prop-2-enamide
InChIKey: LIDOPKHSVQTSJY-VMEIHUARSA-N | ||||||||
| • Delanzomib
IUPAC Name: [(1R)-1-[[(2R,3S)-3-hydroxy-2-[(6-phenylpyridine-2-carbonyl)amino]butanoyl]amino]-3-methylbutyl]boronic acid | CAS Registry Number: 847499-27-8 Synonyms: BCP9000508, RL05207, ((1r)-1-(((2s,3r)-3-hydroxy-2-(((6-phenylpyridin-2-yl)carbonyl)amino)-1-oxobutyl)amino)-3-methylbutyl)boronic acid; cep 18770
InChIKey: SJFBTAPEPRWNKH-ZOCIIQOWSA-N | ||||||||
| • Dequalinium chloride
IUPAC Name: 1-[10-(4-amino-2-methylquinolin-1-ium-1-yl)decyl]-2-methylquinolin-1-ium-4-amine dichloride | CAS Registry Number: 522-51-0 Synonyms: dequalinium chloride, Dequafungan, Dequavagyn, Phylletten, Polycidine, Decamine, Decaminum, Dekuarin, Dequadin, Dequavet, Eriosept, Grocreme, Labosept, Optipect, Danical, Decabis, Decosan, Dekadin, Dekamin, Erosept
InChIKey: LTNZEXKYNRNOGT-UHFFFAOYSA-N | ||||||||
| • Desmethyl Erlotinib
IUPAC Name: 2-[4-(3-ethynylanilino)-7-(2-methoxyethoxy)quinazolin-6-yl]oxyethanol | CAS Registry Number: 183321-86-0 Synonyms: OSI-420, Free Base (Desmethyl Erlotinib), 183321-86-0 pound>>183320-51-6, CTK8F1287, BCPP000136, Desmethyl Erlotinib (CP-473420), ZINC22065493, BCP9001036, NCGC00346578-01, KB-59328, FT-0673312, FT-0673313, 2-[[4-[(3-Ethynylphenyl)amino]-7-(2-methoxyethoxy)-6-quinazolinyl]oxy]ethanol
InChIKey: KOQIAZNBAWFSQM-UHFFFAOYSA-N | ||||||||
| • Deuterated Atazanivir-D3-2
IUPAC Name: methyl N-[(2S)-1-[2-[(2S,3S)-2-hydroxy-4-phenyl-3-[[(2S)-4,4,4-trideuterio-2-(methoxycarbonylamino)-3,3-bis(trideuteriomethyl)butanoyl]amino]butyl]-2-[(4-pyridin-2-ylphenyl)methyl]hydrazinyl]-3,3-dimethyl-1-oxobutan-2-yl]carbamate | CAS Registry Number: 1092540-51-6
InChIKey: AXRYRYVKAWYZBR-HMLRVIJPSA-N | ||||||||
| • Deuterated Atazanivir-D3-3
IUPAC Name: methyl N-[(2S)-4,4,4-trideuterio-1-[[(2S,3S)-3-hydroxy-1-phenyl-4-[(4-pyridin-2-ylphenyl)methyl-[[(2S)-4,4,4-trideuterio-2-(methoxycarbonylamino)-3,3-bis(trideuteriomethyl)butanoyl]amino]amino]butan-2-yl]amino]-1-oxo-3,3-bis(trideuteriomethyl)butan-2-yl]carbamate | CAS Registry Number: 1092540-52-7
InChIKey: AXRYRYVKAWYZBR-AAPVVJSESA-N | ||||||||
| • Dexamethasone
IUPAC Name: (8S,9R,10S,11S,13S,14S,16R,17R)-9-fluoro-11,17-dihydroxy-17-(2-hydroxyacetyl)-10,13,16-trimethyl-6,7,8,11,12,14,15,16-octahydrocyclopenta[a]phenanthren-3-one | CAS Registry Number: 50-02-2 Synonyms: dexamethasone, Dexamethazone, Decadron, Maxidex, Desametasone, Desamethasone, Prednisolone F, Deltafluorene, Mediamethasone, Cortisumman, Dexadeltone, Dexapolcort, Fortecortin, Gammacorten, Hexadecadrol, Millicorten, Superprednol, Visumetazone, Aphtasolon, Decaspray
InChIKey: UREBDLICKHMUKA-CXSFZGCWSA-N | ||||||||
| • Diethyl 1,1-cyclopropanedicarboxylate
IUPAC Name: diethyl cyclopropane-1,1-dicarboxylate | CAS Registry Number: 1559-02-0 Synonyms: Diethyl cyclopropane-1,1-dicarboxylate, 147710_ALDRICH, NSC21376, EINECS 216-321-6, ZINC00162383, 1,1-Cyclopropanedicarboxylic acid, diethyl ester, AI3-05554, ST5406551
InChIKey: KYYUCZOHNYSLFV-UHFFFAOYSA-N | ||||||||
| • Diethyl 1-amino-3-methyl-1H-pyrrole-2,4-dicarboxylate
IUPAC Name: diethyl 1-amino-3-methylpyrrole-2,4-dicarboxylate | CAS Registry Number: 427878-69-1 Synonyms: 1-Amino-3-methyl-1H-pyrrole-2,4-dicarboxylic acid diethyl ester, AGN-PC-00ACFA, SureCN3690592, CTK1D3031, ANW-68714, AKOS016005803, AB56193, QC-1050, AK-68152, KB-217728, diethyl 1-amino-3-methylpyrrole-2,4-dicarboxylate, ETHYL 1-AMINO-3-METHYLPYRROLE-2,4-DICARBOXYLATE, 1H-Pyrrole-2,4-dicarboxylic acid, 1-amino-3-methyl-, diethyl ester, 1-AMINO-3-METHYL-1H-PYRROLE-2,4-DICARBOXYLIC ACID, 2,4-DIETHYL ESTER, 1H-PYRROLE-2,4-DICARBOXYLIC ACID, 1-AMINO-3-METHYL-, 2,4-DIETHYL ESTER
InChIKey: WADSUPVZUARTPO-UHFFFAOYSA-N | ||||||||
| • diethyl cyclopropane-1,1-dicarboxylate
IUPAC Name: diethyl cyclopropane-1,1-dicarboxylate
InChIKey: KYYUCZOHNYSLFV-UHFFFAOYSA-N | ||||||||
| • Dimethyl 5-Bromopyridine-2,3-Dicarboxylate
IUPAC Name: 5-bromopyridine-2,3-dicarboxylic acid | CAS Registry Number: 98555-51-2 Synonyms: 5-BROMOPYRIDINE-2,3-DICARBOXYLIC ACID, 5-bromo-pyridine-2,3-dicarboxylic acid, 5-bromo-2,3-pyridinedicarboxylic acid, SureCN617721, AGN-PC-00PE21, CTK3I6250, MolPort-000-927-991, ALBB-013878, ANW-50093, AKOS004114717, QC-1015, RL06117, 2,3-Pyridinedicarboxylicacid, 5-bromo-, 2,3-Pyridinedicarboxylic acid, 5-bromo-, AK-40088, BR-40088, KB-42541, WT-130303, AM20061808, BB 0257738
InChIKey: WDDREAGLVSBXOG-UHFFFAOYSA-N | ||||||||
| • Dinaciclib
IUPAC Name: 2-[(2S)-1-[3-ethyl-7-[(1-oxidopyridin-1-ium-3-yl)methylamino]pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-2-yl]ethanol | CAS Registry Number: 779353-01-4 Synonyms: SCH-727965, SCH727965, Dinaciclib (USAN/INN), SureCN12048446, cc-241, Dinaciclib (SCH727965), CHEMBL2103840, DCL001081, NSC747135, CS-0541, MK-7965, NSC-727135, NSC-747135, RL05018, SCH 727965, HY-10492, KB-76642, SCH 727965,SCH727965, Dinaciclib, Y0347, D09604
InChIKey: PIMQWRZWLQKKBJ-SFHVURJKSA-N | ||||||||
| • Divalproex Sodium
IUPAC Name: sodium; 2-propylpentanoate; 2-propylpentanoic acid | CAS Registry Number: 76584-70-8 Synonyms: Depakote, Epival, Delepsine, Sprinkle, Valparin, Valcote, Epilex, Valproate semisodium, Divalproate, Valdisoval, Depakote ER, Cereb, Depakine chrono, DIVALPROEX SODIUM, Sodium divalproate, 2-propylpentanoate, Depakote (TN), SODIUM, Abbott 50711, 2-Propylpentanoic acid
InChIKey: MSRILKIQRXUYCT-UHFFFAOYSA-M | ||||||||
| • Docetaxel
Synonyms: docetaxel, Taxotere, Docetaxol, Docetaxel anhydrous, nchembio853-comp8, Docetaxel, Trihydrate, nchembio.2007.34-comp7, 01885_FLUKA, XRP-6976L, ANX-514, SDP-014, DB01248, NSC-628503, RP-56976, SL-00678, C11231, TXL, (2alpha,5beta,7beta,10beta,13alpha)-4-(acetyloxy)-13-({(2R,3S)-3-[(tert-butoxycarbonyl)amino]-2-hydroxy-3-phenylpropanoyl}oxy)-1,7,10-trihydroxy-9-oxo-5,20-epoxytax-11-en-2-yl benzoate, (2aR,4S,4aS,6R,9S,11S,12S,12aR,12bS)-12b-(acetyloxy)-12-(benzoyloxy)-2a,3,4,4a,5,6,9,10,11,12,12a,12b-dodecahydro-4,6,11-trihydroxy-4a,8,13,13-tetramethyl-5-oxo-7,11-methano-1H-cyclodeca[3,4]benz[1,2-b]oxet-9-yl (aR,bS)-b-[[(1,1-dimethylethoxy)carbonyl]amino]-a-hydroxybenzenepropanoate
InChIKey: ZDZOTLJHXYCWBA-VCVYQWHSSA-N | ||||||||
| • Doramapimod
IUPAC Name: 1-[5-tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]urea | CAS Registry Number: 285983-48-4 Synonyms: nchembio.162-comp7, BIRB-796, 1kv2, UNII-HO1A8B3YVV, Doramapimod (USAN/INN), BIRB 796, CID156422, DB03044, D03736, 1-(5-TERT-BUTYL-2-P-TOLYL-2H-PYRAZOL-3-YL)-3-[4-(2-MORPHOLIN-4-YL-ETHOXY)-NAPHTHALEN-1-YL]-UREA, B96, 1-(3-(1,1-dimethylethyl)-1-(4-methylphenyl)-1H-pyrazol-5-yl)-3-(4-(2-(morpholin-4-yl)ethoxy)naphthalen-1-yl)urea, 1-(5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl)-3(4-(2-morpholin-4-yl-ethoxy)naphthalen-1-yl)urea, 1-[5-tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]urea, Urea, N-(3-(1,1-dimethylethyl)-1-(4-methylphenyl)-1H-pyrazol-5-yl)-N'-(4-(2-(4-morpholinyl)ethoxy)-1-naphthalenyl)-
InChIKey: MVCOAUNKQVWQHZ-UHFFFAOYSA-N | ||||||||
| • Dorsomorphin dihydrochloride
IUPAC Name: 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine;dihydrochloride | CAS Registry Number: 1219168-18-9 Synonyms: Dorsomorphin 2HCl, 6-[4-[2-(1-PIPERIDINYL)ETHOXY]PHENYL]-3-(4-PYRIDINYL)-PYRAZOLO[1,5-A]PYRIMIDINE DIHYDROCHLORIDE, SureCN2119244, CTK8F9363, FD5027, MCULE-9260462246, QC-11168, S7306,BML-275,Compound C,1219168-18-9
InChIKey: RJDVIJJQKMGPMV-UHFFFAOYSA-N | ||||||||
| • Dovitinib
IUPAC Name: 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1,3-dihydrobenzimidazol-2-ylidene]quinolin-2-one | CAS Registry Number: 405169-16-6 Synonyms: Kinome_1513, SureCN172687, SureCN949705, SureCN9975396, SureCN10330209, CTK4I3259, AG-F-43728, NCGC00249685-01, NCGC00249685-02, 196472-EP2270000A1, 2(1H)-Quinolinone,4-amino-5-fluoro-3-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-, 4-amino-5-fluoro-3-[6-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-quinolin-2-one, 2(1H)-Quinolinone,4-amino-5-fluoro-3-[5-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]- (9CI);4-Amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]quinolin-2(1H)-one;Dovitinib, 4-AMINO-5-FLUORO-3-[6-(4-METHYLPIPERAZIN-1-YL)-1H-BENZIMIDAZOL-2-YL]QUINOLIN-2(1H)-ONE
InChIKey: KCOYQXZDFIIGCY-UHFFFAOYSA-N | ||||||||
| • Doxycycline hydrochloride
IUPAC Name: (2Z,4S,4aR,5S,5aR,6R)-2-[amino(hydroxy)methylidene]-4-(dimethylamino)-5,10,11,12a-tetrahydroxy-6-methyl-4a,5,5a,6-tetrahydro-4H-tetracene-1,3,12-trione hydrochloride | CAS Registry Number: 10592-13-9 Synonyms: Doxycycline hyclate, Prestwick_1072, MLS002154032, CID6420082, SMR001233359
InChIKey: VLUQVUWDECWBTL-WGDOXZFCSA-N | ||||||||
| • Duvelisib
IUPAC Name: 8-chloro-2-phenyl-3-[(1S)-1-(7H-purin-6-ylamino)ethyl]isoquinolin-1-one | CAS Registry Number: 1201438-56-3 Synonyms: IPI-145, Duvelisib [USAN], SureCN153543, UNII-610V23S0JI, IPI145, CHEMBL3039502, INK-1197, IPI-145 (INK1197), CS-0888, HY-17044, QC-10232, IPI-145|1201438-56-3|IPI145, S7028,INK1197,1201438-56-3, (S)-3-(1-(7H-purin-6-ylamino)ethyl)-8-chloro-2-phenylisoquinolin-1(2H)-one, 1(2H)-Isoquinolinone, 8-chloro-2-phenyl-3-((1S)-1-(9H-purin-6-ylamino)ethyl)-, 8-Chloro-2-phenyl-3-((1S)-1-(7H-purin-6-ylamino)ethyl)isoquinolin-1(2H)-one
InChIKey: SJVQHLPISAIATJ-ZDUSSCGKSA-N | ||||||||
| • E-Maleimidocapronic Acid Hydrazide
IUPAC Name: 6-(2,5-dioxopyrrol-1-yl)hexanehydrazide | CAS Registry Number: 81186-33-6 Synonyms: 6-Maleimidocaproic acid hydrazide, 6-Maleimidocaproicacidhydrazide(EMCH), AG-H-26219, PubChem11841, 6-(2,5-dioxopyrrol-1-yl)hexanehydrazide, AC1N5ED1, SureCN1064498, CTK3E6282, e-Maleimidocaproic acid hydrazide, ZINC06691778, AKOS016014324, 6-MALEIMIDOCAPROIC ACIDHYDRAZIDE, AK129117, KB-199511, A9985, FT-0604082, FT-0670912, 6-(2,5-dioxo-2H-pyrrol-1(5H)-yl)hexanehydrazide, 6-(2,5-Dioxo-2,5-dihydro-1H-pyrrol-1-yl)hexanehydrazide, 1H-Pyrrole-1-hexanoicacid, 2,5-dihydro-2,5-dioxo-, hydrazide
InChIKey: FYWVFGAAKATOHN-UHFFFAOYSA-N | ||||||||
| • E7080 (CAS: 17716-92-8) | ||||||||
| • Elesclomol
IUPAC Name: 1-N',3-N'-bis(benzenecarbonothioyl)-1-N',3-N'-dimethylpropanedihydrazide | CAS Registry Number: 488832-69-5 Synonyms: UNII-6UK191M53P, NSC174939, STA 4783, STA-4783, CID300471, NCI60_001429, N'1,N'3-dimethyl-N'1,N'3-bis(phenylcarbonothioyl)propanedihydrazide, Propanedioic acid, bis[2-methyl-2-(phenylthioxomethyl)hydrazide]
InChIKey: BKJIXTWSNXCKJH-UHFFFAOYSA-N | ||||||||
| • EMCS
IUPAC Name: (2,5-dioxopyrrolidin-1-yl) 6-(2,5-dioxopyrrol-1-yl)hexanoate | CAS Registry Number: 55750-63-5 Synonyms: Nmicos, BICL222, 568600_ALDRICH, 63177_FLUKA, N-Succinimidyl 6-maleimidocaproate, N-(epsilon-Maleimidocaproyloxy)succinimide, CID5091655, 6-Maleimidocaproic acid N-succinimidyl ester, 6-Maleimidohexanoic acid N-hydroxysuccinimide ester, 1H-Pyrrole-2,5-dione, 1-(6-((2,5-dioxo-1-pyrrolidinyl)oxy)-6-oxohexyl)-
InChIKey: VLARLSIGSPVYHX-UHFFFAOYSA-N | ||||||||
| • ENMD-2076
IUPAC Name: (2S,3S)-2,3-dihydroxybutanedioic acid; 6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine | CAS Registry Number: 1291074-87-7 Synonyms: ENMD-2076 Tartrate, ENMD-2076 L-(+)-Tartaric acid, CS-0210, HY-10987, A4129, ENMD-2076 Tartrate|1291074-87-7|ENMD2076
InChIKey: KGWWHPZQLVVAPT-PCWHHUEVSA-N | ||||||||
| • ENMD-2076
IUPAC Name: 6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine | CAS Registry Number: 934353-76-1 Synonyms: ENMD 2076, ENMD2076, 6-(4-METHYL-1-PIPERAZINYL)-N-(5-METHYL-1H-PYRAZOL-3-YL)-2-[(1E)-2-PHENYLETHENYL]-4-PYRIMIDINAMINE, SureCN597664, UNII-J6U9WP10T7, SureCN10122872, cc-471, CHEMBL482968, CHEBI:620121, DCL001071, HY-10987A, CS-0836, RL05865, ENMD-2076|934353-76-1|ENMD2076, (E)-N-(5-Methyl-1H-pyrazol-3-yl)-6-(4-methylpiperazin-1-yl)-2-styrylpyrimidin-4-amine, 4-Pyrimidinamine, 6-(4-methyl-1-piperazinyl)-N-(5-methyl-1H-pyrazol-3-yl)-2-((1E)-2-phenylethenyl)-
InChIKey: BLQYVHBZHAISJM-CMDGGOBGSA-N | ||||||||
| • Entacapone
IUPAC Name: (E)-2-cyano-3-(3,4-dihydroxy-5-nitrophenyl)-N,N-diethylprop-2-enamide | CAS Registry Number: 130929-57-6 Synonyms: Comtan, ENTACAPONE, Entacaponum, Comtess, Entacapona, Comtan (TN), Entacaponum [INN-Latin], Entacapona [INN-Spanish], Entacapone [USAN:INN], BIDD:GT0026, Entacapone (JAN/USAN/INN), UNII-4975G9NM6T, OR-611, CHEBI:4798, COM-998, MolPort-003-847-054, OR 611, C14H15N3O5, HMS2089O16, AC-393
InChIKey: JRURYQJSLYLRLN-BJMVGYQFSA-N | ||||||||
| • Enzalutamide
IUPAC Name: 4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluoro-N-methylbenzamide | CAS Registry Number: 915087-33-1 Synonyms: MDV3100, MDV-3100, MDV 3100, 4-(3-(4-cyano-3-(trifluoromethyl)phenyl)-5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl)-2-fluoro-N-methylbenzamide, XTANDI, UNII-93T0T9GKNU, CHEBI:68534, MDV-3100, 915087-33-1, MDV-3100, MDV3100, 4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluoro-N-methylbenzamide, 4-{3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl}-2-fluoro-N-methylbenzamide, 4-{3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl}-2-fluoro-N-methylbenzamide, Xtandi (TN), S1250_Selleck, PubChem19320, MDV3100 Enzalutamide, AGN-PC-00QCRK, Enzalutamide (JAN/USAN), MDV3100 (Enzalutamide), 93T0T9GKNU
InChIKey: WXCXUHSOUPDCQV-UHFFFAOYSA-N | ||||||||
| • Enzastaurin
IUPAC Name: 3-(1-methylindol-3-yl)-4-[1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]indol-3-yl]pyrrole-2,5-dione | CAS Registry Number: 170364-57-5 Synonyms: UNII-UC96G28EQF, CHEBI:183217, CID176167, LY317615, 1H-Pyrrole-2,5-dione, 3-(1-methyl-1H-indol-3-yl)-4-(1-(1-(2-pyridinylmethyl)-4-piperidinyl)-1H-indol-3-yl)-, 3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-pyridin-2-ylmethyl-piperidin-4-yl)-1H-indol-3-yl]-pyrrole-2,5-dione, 3-(1-methyl-1H-indol-3-yl)-4-{1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-indol-3-yl}-1H-pyrrole-2,5-dione
InChIKey: AXRCEOKUDYDWLF-UHFFFAOYSA-N | ||||||||
| • Epothilone A
IUPAC Name: (1R,5S,6S,7R,10S,14S,16S)-6,10-dihydroxy-5,7,9,9-tetramethyl-14-[(E)-1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-13,17-dioxabicyclo[14.1.0]heptadecane-8,12-dione | CAS Registry Number: 152044-53-6 Synonyms: (-)-Epothilone A, Epoa, EP, Epothilones, Epo A, Epothilon A, Epothilone-A, Epothilone A [MI], S1297_Selleck, AC1L9MD2, cc-632, E3656_SIGMA, UNII-51E07YBX96, CHEMBL329993, MolPort-016-633-197, (1S,3S,7S,10R,11S,12S,16R)-7,11-dihydroxy-8,8,10,12-tetramethyl-3-[(1E)-1-methyl-2-(2-methyl-4-thiazolyl)ethenyl]-4,17-dioxabicyclo[14.1.0]heptadecane-5,9-dione, LMPK04000040, NSC684362, BCP9000654, NSC-684362
InChIKey: HESCAJZNRMSMJG-KKQRBIROSA-N | ||||||||
| • Epothilone B
IUPAC Name: (1R,5S,6S,7R,10S,14S,16S)-6,10-dihydroxy-1,5,7,9,9-pentamethyl-14-[(E)-1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-13,17-dioxabicyclo[14.1.0]heptadecane-8,12-dione | CAS Registry Number: 152044-54-7 Synonyms: Patupilone, (-)-Epothilone B, Epothilon B, EpoB, nchembio853-comp4, E2656_SIGMA, EPO 906, EPO906, EPO-906, CHEBI:252995, CID448013, LMPK04000041, NSC684363, NCGC00181131-01, LS-62193, C12154, 4,17-Dioxabicyclo(1410)heptadecane-5,9-dione, 7,11-dihydroxy-8,8,10,12,16-pentamethyl-3-((1E)-1-methyl-2-(2-methyl-4-thiazolyl)ethenyl)-, (1S,3S,7S,10R,11S,12S,16R)-, 4,17-Dioxabicyclo(1410)heptadecane-5,9-dione, 7,11-dihydroxy-8,8,10,12,16-pentamethyl-3-(1-methyl-2-(2-methyl-4-thiazolyl)ethenyl)-, (1S-(1R*,3R*(E),7R*,10S*,11R*,12R*,16S*))-, EPB, (1S,3S,7S,10R,11S,12S,16R)-7,11-Dihydroxy-8,8,10,12,16-pentamethyl-3-((1E)-1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl)-4,17-dioxabicyclo(14.1.0)heptadecane-5,9-dione
InChIKey: QXRSDHAAWVKZLJ-PVYNADRNSA-N | ||||||||
| • Epoxomicin
IUPAC Name: (2S,3S)-2-[[(2S,3S)-2-[acetyl(methyl)amino]-3-methylpentanoyl]amino]-N-[(2S,3R)-3-hydroxy-2-[[4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]butanoyl]-3-methylpentanamide | CAS Registry Number: 134381-21-8 Synonyms: epoxomicin, CHEBI:447838, MolPort-006-822-455, CID3035402, CID 3035402, C078846, (2S,3S)-2-[(2S,3S)-2-(acetyl-methyl-amino)-3-methyl-pentanoylamino]-3-methyl-pentanoic acid {(2S,3R)-3-hydroxy-2-[3-methyl-1-((R)-2-methyl-oxiranecarbonyl)-butylamino]-butyryl}-amide, L-Threoninamide, N-acetyl-N-methyl-L-isoleucyl-L-isoleucyl-N-((1S)-3-methyl-1-(((2R)-2-methyloxiranyl)carbonyl)butyl)-, N-Acetyl-N-methyl-L-isoleucyl-L-isoleucyl-N-(3-methyl-1-((2-methyloxiranyl)carbonyl)butyl)-L-threoninamide
InChIKey: ZWCBKZGIPPDRLY-TXLQCSLMSA-N | ||||||||
| • EPZ004777
IUPAC Name: 1-[3-[[(2R,3S,4R,5R)-5-(4-aminopyrrolo[2,3-d]pyrimidin-7-yl)-3,4-dihydroxyoxolan-2-yl]methyl-propan-2-ylamino]propyl]-3-(4-tert-butylphenyl)urea | CAS Registry Number: 1338466-77-5 Synonyms: CHEMBL2169919, 0QK, 7-{5-[(3-{[(4-Tert-Butylphenyl)carbamoyl]amino}propyl)(Propan-2-Yl)amino]-5-Deoxy-Beta-D-Ribofuranosyl}-7h-Pyrrolo[2,3-D]pyrimidin-4-Amine, SureCN9274416, EPZ 004777, KB-76812, S7032,1338466-77-5, 1-(3-((((2R,3S,4R,5R)-5-(4-Amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl)(isopropyl)amino)propyl)-3-(4-(tert-butyl)phenyl)urea
InChIKey: WXRGFPHDRFQODR-ICLZECGLSA-N | ||||||||
| • EPZ005687
IUPAC Name: 1-cyclopentyl-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[4-(morpholin-4-ylmethyl)phenyl]indazole-4-carboxamide | CAS Registry Number: 1396772-26-1 Synonyms: SureCN12684069, CS-1215, EPZ 005687, HY-15555, KB-145937, EPZ005687|1396772-26-1|EPZ 005687, S7004,EPZ 005687,1396772-26-1
InChIKey: ZOIBZSZLMJDVDQ-UHFFFAOYSA-N | ||||||||
| • Erlotinib
IUPAC Name: N-(3-ethynylphenyl)-6,7-bis(2-methoxyethoxy)quinazolin-4-amine | CAS Registry Number: 183321-74-6 Synonyms: Tarceva, erlotinib HCl, Erlotinib [INN], Erlotinib(Tarceva), nchembio866-comp3, OSI-774, STOCK6S-52681, CID176870, DB00530, NCGC00164574-01, BCB03_000783, CP 358774, CP-358774, LS-184395, CP 358,774, CP-358,774, K00241, C400278, N-(3-Ethynylphenyl)-6,7-bis(2-methoxyethoxy)quinazolin-4-amine, 4-Quinazolinamine, N-(3-ethynylphenyl)-6,7-bis(2-methoxyethoxy)-
InChIKey: AAKJLRGGTJKAMG-UHFFFAOYSA-N | ||||||||
| • Erlotinib hydrochloride
IUPAC Name: N-(4-ethynylphenyl)-6,7-bis(2-methoxyethoxy)quinazolin-4-amine hydrochloride | CAS Registry Number: 183319-69-9 Synonyms: Tarceva, Tarceva (TN), Erlotinib hydrochloride (JAN/USAN), CID11954378, D04023
InChIKey: OMDIKDVVYHAXGO-UHFFFAOYSA-N | ||||||||
| • ETHANETHIOAMIDE,N-(4-METHOXYPHENYL)-
IUPAC Name: N-(4-methoxyphenyl)ethanethioamide | CAS Registry Number: 5310-18-9 Synonyms: p-Acetanisidide, thio-, N-(4-Methoxyphenyl)thioacetamide, MolPort-006-827-184, CID3034157, Ethanethioamide, N-(4-methoxyphenyl)-
InChIKey: WZNUJVLBHDEJDY-UHFFFAOYSA-N | ||||||||
| • Ethanone, 1-(4-bromo-2-hydroxyphenyl)-
IUPAC Name: 1-(4-bromo-2-hydroxyphenyl)ethanone | CAS Registry Number: 30186-18-6 Synonyms: 1-(4-bromo-2-hydroxyphenyl)ethanone, 4-Bromo-2-Hydroxyacetophenone, 4'-Bromo-2'-hydroxyacetophenone, acetophenone,2-hydroxy-4-bromo, 1-(4-bromo-2-hydroxyphenyl) ethanone, 1-(4-Bromo-2-hydroxyphenyl)ethan-1-one, PubChem19929, SureCN55915, KSC916A5D, CTK8B6051, MolPort-000-481-985, 1-acetyl-4-bromo-2-hydroxybenzene, ANW-52314, RW3109, STK820367, WTI-10111, ZINC02585998, AKOS002229507, AB15427, MCULE-2030152556
InChIKey: LQCMMXGKEGWUIM-UHFFFAOYSA-N | ||||||||
| • Ethanone, 1-(4-chloro-6-methyl-2-pyridinyl)-
IUPAC Name: 1-(4-chloro-6-methylpyridin-2-yl)ethanone | CAS Registry Number: 339586-00-4 Synonyms: 1-(4-Chloro-6-methylpyridin-2-yl)ethanone, AGN-PC-01X5EK, SureCN6550051, CTK8B8674, ANW-61011, AKOS016003429, AB66887, AK-68368, KB-76852, Ethanone,1-(4-chloro-6-methyl-2-pyridinyl)-, 1-(4-CHLORO-6-METHYL-2-PYRIDINYL)-ETHANONE, 1-(4-CHLORO-6-METHYLPYRIDIN-2-YL)ETHAN-1-ONE, ETHANONE, 1-(4-CHLORO-6-METHYL-2-PYRIDINYL)-
InChIKey: NLXINSLPJMHYKN-UHFFFAOYSA-N | ||||||||
| • Ethanone, 1-(6-chloro-5-nitro-3-pyridinyl)-
IUPAC Name: 1-(6-chloro-5-nitropyridin-3-yl)ethanone | CAS Registry Number: 127356-40-5 Synonyms: 1-(6-Chloro-5-nitropyridin-3-yl)ethanone, AGN-PC-002GMP, CTK8B8839, ANW-61442, AKOS016002981, AB60285, AK-41546, KB-76865, 5-ACETYL-2-CHLORO-3-NITROPYRIDINE, Ethanone,1-(6-chloro-5-nitro-3-pyridinyl)-, 1-(6-CHLORO-5-NITRO-3-PYRIDINYL)ETHANONE, 1-(6-CHLORO-5-NITROPYRIDIN-3-YL)ETHAN-1-ONE, ETHANONE, 1-(6-CHLORO-5-NITRO-3-PYRIDINYL)-
InChIKey: UZUVOPNXKQOJKI-UHFFFAOYSA-N | ||||||||
| • ETHANONE,1-(3-AMINO-4-METHYLPHENYL)-
IUPAC Name: 1-(3-amino-4-methylphenyl)ethanone | CAS Registry Number: 17071-24-8 Synonyms: MolPort-002-462-083, NSC380875, CID342914, ZINC01591218
InChIKey: MCQYTLIHRDCHHT-UHFFFAOYSA-N | ||||||||
| • ETHANONE,1-(3-HYDROXY-PYRIDIN-4-YL)-
IUPAC Name: 1-(3-hydroxypyridin-4-yl)ethanone | CAS Registry Number: 30152-05-7 Synonyms: 1-(3-Hydroxypyridin-4-yl)ethanone, SureCN1798009, CTK8B4165, MolPort-004-770-875, 1-(3-hydroxy-4-pyridinyl)ethanone, ANW-44165, AKOS015999719, Ethanone,1-(3-hydroxy-4-pyridinyl)-, AK-68365, KB-76847
InChIKey: REYSBWKWFPSDDR-UHFFFAOYSA-N | ||||||||
| • ETHANONE,1-(3-METHOXY-PYRIDIN-2-YL)-
IUPAC Name: 1-(3-methoxypyridin-2-yl)ethanone | CAS Registry Number: 379227-03-9 Synonyms: 1-(3-Methoxypyridin-2-yl)ethanone, SureCN5928881, CTK8C2292, MolPort-004-771-598, ANW-68154, AKOS016007064, AK-80679, BD237050, KB-213933
InChIKey: IGYMEVBVNSGNSD-UHFFFAOYSA-N |