Profile: Jinan Trio PharmaTech Co., Ltd. specializes in APIs & intermediates, heterocyclic compounds, and anti-tumor drugs. Our products include crizotinib, vemurafenib, afatinib, vandetanib, regorafenib, brivanib alaninate, pyridazine, imidazole, pyrazole, and oxazole. We are specialized in providing over 1000 products including molecular targeted anticancer drugs, cell signaling pathway inhibitors, pharmaceutical intermediates, and heterocyclic compounds, and quality services including custom synthesis, transfer of new drug patent and technology, technical cooperation, and process optimization.
| • Icotinib
Synonyms: CHEMBL2087361, Conmana, icotinib,BPI-2009H, UNII-9G6U5L461Q, BPI-2009, (1,4,7,10)Tetraoxacyclododecino(2,3-g)quinazolin-4-amine, N-(3-ethynylphenyl)-7,8,10,11,13,14-hexahydro-
InChIKey: QQLKULDARVNMAL-UHFFFAOYSA-N | ||||||||
| • Idelalisib
IUPAC Name: 5-fluoro-3-phenyl-2-[(1S)-1-(7H-purin-6-ylamino)propyl]quinazolin-4-one | CAS Registry Number: 870281-82-6 Synonyms: CAL-101, CAL 101, GS-1101, CAL101, CHEMBL2216870, CAL-101, CAL101, (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one, 5-fluoro-3-phenyl-2-((1s)-1-(9h-purin-6-ylamino)propyl)-4(3h)-quinazolinone, 5-FLUORO-3-PHENYL-2-[(1S)-1-(9H-PURIN-6-YLAMINO)PROPYL]-4(3H)-QUINAZOLINONE, S2226_Selleck, Idelalisib [USAN:INN], cc-41, SureCN356400, UNII-YG57I8T5M0, QCR-36, GS-11CAL-101, MolPort-016-633-355, BCPP000307, GS1101, BCP9000471
InChIKey: IFSDAJWBUCMOAH-HNNXBMFYSA-N | ||||||||
| • Ilomastat
IUPAC Name: (2R)-N'-hydroxy-N-[(2S)-3-(1H-indol-3-yl)-1-(methylamino)-1-oxopropan-2-yl]-2-(2-methylpropyl)butanediamide | CAS Registry Number: 142880-36-2 Synonyms: Galardin, Galardin MPI, Ilomastat [USAN], Ilomastat (USAN/INN), GM 6001, CBiol_001883, BSPBio_001079, KBioGR_000419, KBioSS_000419, BCBcMAP01_000057, KBio2_000419, KBio2_002987, KBio2_005555, KBio3_000797, KBio3_000798, CS 610, Bio1_000169, Bio1_000658, Bio1_001147, Bio2_000370
InChIKey: NITYDPDXAAFEIT-DYVFJYSZSA-N | ||||||||
| • Imatinib
IUPAC Name: 4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide | CAS Registry Number: 152459-95-5 Synonyms: Glivec, Gleevec, Imatinib mesylate, 1iep, 1xbb, sti-571, nchembio.83-comp14, Imatinib [INN:BAN], Imatinib Methansulfonate, nchembio.117-comp23, STI 571, Cgp 57148, CGP 57148B, CCRIS 9076, STI571, STOCK6S-47743, CHEBI:45783, CID5291, DB00619, DB03261
InChIKey: KTUFNOKKBVMGRW-UHFFFAOYSA-N | ||||||||
| • IMD-0354
IUPAC Name: N-[3,5-bis(trifluoromethyl)phenyl]-5-chloro-2-hydroxybenzamide | CAS Registry Number: 978-62-1 Synonyms: IKK-2 Inhibitor V, IMD 0354, CHEMBL536151, N-(3,5-Bis-trifluoromethylphenyl)-5-chloro-2-hydroxybenzamide, TCMDC-125465, N-(3,5-bis(trifluoromethyl)phenyl)-5-chloro-2-hydroxybenzamide, N-[3,5-bis(trifluoromethyl)phenyl]-5-chloro-2-hydroxybenzamide, IMD0354, Kinome_1864, AC1NO40S, I3159_SIGMA, CTK8G0277, HMS3229F11, HMS3269F13, UNII-76145IS906, IN1463, AG-H-98244, BCP9000777, NCGC00165811-01, NCGC00165811-02
InChIKey: CHILCFMQWMQVAL-UHFFFAOYSA-N | ||||||||
| • Imidazo[1,2-a]pyridin-2(3H)-one hydrochloride
IUPAC Name: 3H-imidazo[1,2-a]pyridin-2-one;hydrochloride | CAS Registry Number: 52687-85-1 Synonyms: imidazo(1,2-a)pyridin-2(3h)-one hydrochloride, PubChem23703, SureCN3306488, CTK8B8592, MolPort-003-912-125, ACN-P000818, ANW-60773, AKOS015831807, RL03941, AK-80162, KB-52554, 3H-imidazo[1,2-a]pyridin-2-one hydrochloride, A829204, I14-15855
InChIKey: YLYILEUMTDOZTJ-UHFFFAOYSA-N | ||||||||
| • Imidazo[1,2-A]Pyridin-8-Ylamine
IUPAC Name: imidazo[1,2-a]pyridin-8-amine | CAS Registry Number: 73221-18-8 Synonyms: IMIDAZO[1,2-A]PYRIDIN-8-YLAMINE, Imidazo[1,2-a]pyridin-8-amine, H-imidazo[1,2-a]pyridin-8-amine, SBB052098, PubChem22323, SureCN335977, AGN-PC-00P64E, CTK2H5980, MolPort-008-155-908, Imidazo[1,2-a]pyridin-8-ylamine;, ANW-50456, WTI-10074, ZINC34551954, AKOS006292620, AG-C-11755, AG-G-89253, MCULE-6007212180, PB32476, RP20069, 8-AMINOIMIDAZO[1,2-A]PYRIDINE
InChIKey: LKQXJYDAALZCAF-UHFFFAOYSA-N | ||||||||
| • Imidazo[2,1-b]thiazole-5-carboxylic acid
IUPAC Name: imidazo[2,1-b][1,3]thiazole-5-carboxylic acid | CAS Registry Number: 17782-81-9 Synonyms: imidazo[2,1-b][1,3]thiazole-5-carboxylic acid, SureCN269609, MolPort-008-626-706, ANW-49066, RW4012, AKOS015920176, RP23087, 5-imidazo[2,1-b]thiazolecarboxylic acid, AK-31309, BR-31309, KB-77866, W3878, A812301
InChIKey: ZGIABSKPSCMXFD-UHFFFAOYSA-N | ||||||||
| • Indole-3-acetamide
IUPAC Name: 2-(1H-indol-3-yl)acetamide | CAS Registry Number: 879-37-8 Synonyms: Indoleacetamide, indole-3-acetamide, 1H-Indole-3-acetamide, 3-Indoleacetamide, 3-Indolylacetamide, (indol-3-yl)acetamide, 2-(3-Indolyl)acetamide, 2-(1H-Indol-3-yl)acetamide, Indole-3-acetamide (8CI), Oprea1_704903, 286281_ALDRICH, CID397, NSC 1969, CHEBI:16031, CPD-237, Indole-3-acetamide (6CI,8CI), NSC1969, AIDS019635, AIDS-019635, EINECS 212-904-4
InChIKey: ZOAMBXDOGPRZLP-UHFFFAOYSA-N | ||||||||
| • Infigratinib
IUPAC Name: 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-[6-[4-(4-ethylpiperazin-1-yl)anilino]pyrimidin-4-yl]-1-methylurea | CAS Registry Number: 872511-34-7 Synonyms: NVP-BGJ398, BGJ398, BGJ 398, BGJ-398, 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-(4-(4-ethylpiperazin-1-yl)phenylamino)pyrimidin-4-yl)-1-methylurea, 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylurea, 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-((4-(4-ethylpiperazin-1-yl)phenyl)amino)pyrimidin-4-yl)-1-methylurea, NVP BGJ398, UNII-A4055ME1VK, cc-248, QCR-48, CHEBI:63451, BGJ398, NVP-BGJ398, BGJ398 (NVP-BGJ398), BGJ398 - NVP-BGJ398, FD5035, RW4152, BCP9000399, CS-0586, RL05423
InChIKey: QADPYRIHXKWUSV-UHFFFAOYSA-N | ||||||||
| • IOX2
IUPAC Name: 2-[(1-benzyl-4-hydroxy-2-oxoquinoline-3-carbonyl)amino]acetic acid | CAS Registry Number: 931398-72-0 Synonyms: SureCN8244419, IOX 2, IOX-2, cc-642, QCR-246, CS-0988, RL05859, NCGC00344625-02, HY-15468, KB-146012, IOX2|931398-72-0|IOX-2, 2-(1-benzyl-4-hydroxy-2-oxo-1,2-dihydroquinoline-3-carboxamido)acetic acid, N-[(1-BENZYL-4-HYDROXY-2-OXO-1,2-DIHYDRO-3-QUINOLINYL)CARBONYL]GLYCIN
InChIKey: CAOSCCRYLYQBES-UHFFFAOYSA-N | ||||||||
| • Ipatasertib
IUPAC Name: (2S)-2-(4-chlorophenyl)-1-[4-[(5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl]-3-(propan-2-ylamino)propan-1-one | CAS Registry Number: 1001264-89-6 Synonyms: GDC-0068, CHEMBL2177390, GDC 0068, RG 7440, SureCN191659, cc-616, GDC0068, BCP9000712, CS-0975, RG-7440, GDC-0068 (RG7440), NCGC00346714-01, HY-15186, QC-10488, BCP0726000195, GDC-0068|1001264-89-6|GDC0068|GDC 0068|RG-7440, (2s)-2-(4-Chlorophenyl)-1-{4-[(5r,7r)-7-Hydroxy-5-Methyl-6,7-Dihydro-5h-Cyclopenta[d]pyrimidin-4-Yl]piperazin-1-Yl}-3-(Propan-2-Ylamino)propan-1-One, 0RF
InChIKey: GRZXWCHAXNAUHY-NSISKUIASA-N | ||||||||
| • Isothiazalone
IUPAC Name: 1,2-thiazol-3-one | CAS Registry Number: 1003-07-2 Synonyms: 3-Isothiazolone, Isothiazol-3-one, 3(2H)-Isothiazolone, NCIOpen2_001597, NSC93489, AIDS125977, AIDS-125977, NSC 93489, NCI60_042085, TL8000042
InChIKey: MGIYRDNGCNKGJU-UHFFFAOYSA-N | ||||||||
| • Isothiazolo[5,4-b]pyridin-3(2H)-one, 1,1-dioxide
IUPAC Name: 1,1-dioxo-[1,2]thiazolo[5,4-b]pyridin-3-one | CAS Registry Number: 138417-40-0 Synonyms: Isothiazolo[5,4-b]pyridin-3(2H)-one 1,1-dioxide, ACMC-20adbx, AGN-PC-003HJU, CTK0B8283, ANW-68203, AKOS016007145, AK-80617, KB-77966, Isothiazolo[5,4-b]pyridin-3(2H)-one,1,1-dioxide, 2H,3H-1$l^{6},2,7-[1$l^{6},2]thiazolo[5,4-b]pyridine-1,1,3-trione
InChIKey: TYWYQFLITLNVEM-UHFFFAOYSA-N | ||||||||
| • Isothiazolo[5,4-c]pyridin-3(2H)-one, 1,1-dioxide
IUPAC Name: 1,1-dioxo-[1,2]thiazolo[5,4-c]pyridin-3-one | CAS Registry Number: 142141-07-9 Synonyms: Isothiazolo[5,4-c]pyridin-3(2H)-one 1,1-dioxide, AGN-PC-003Y8C, CTK8B9054, MolPort-000-884-699, ANW-61910, AKOS000282122, AK-80620, KB-77967, Isothiazolo[5,4-c]pyridin-3(2H)-one,1,1-dioxide
InChIKey: OCDUJMWEISRJAC-UHFFFAOYSA-N | ||||||||
| • Isoxazole, 4-Bromo-3-Ethoxy-5-Methyl- (9CI)
IUPAC Name: 4-bromo-3-ethoxy-5-methyl-1,2-oxazole | CAS Registry Number: 169310-98-9 Synonyms: 4-Bromo-3-ethoxy-5-methylisoxazole, 4-BROMO-3-ETHOXY-5-METHYL-ISOXAZOLE, PubChem24241, CTK8C2316, MolPort-004-789-027, ANW-68192, AKOS016007227, Isoxazole,4-bromo-3-ethoxy-5-methyl-, AK-80632, KB-77974
InChIKey: WYGNIHJIFAZCBL-UHFFFAOYSA-N | ||||||||
| • IU1
IUPAC Name: 1-[1-(4-fluorophenyl)-2,5-dimethylpyrrol-3-yl]-2-pyrrolidin-1-ylethanone | CAS Registry Number: 314245-33-5 Synonyms: CHEMBL1410015, F1142-1244, 1-(1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl)-2-(pyrrolidin-1-yl)ethanone, Usp14 inhibitor, AC1LDUCV, AC1Q2HNB, SureCN6923146, MLS001032847, MolPort-000-565-740, HMS1726C11, HMS2742M13, AKOS000811299, CCG-190730, MCULE-9620933012, QC-8208, NCGC00249377-01, SMR000363441, ST054127, MLS001032847-02, EN300-72884
InChIKey: JUWDSDKJBMFLHE-UHFFFAOYSA-N | ||||||||
| • Ixazomib
IUPAC Name: [(1R)-1-[[2-[(2,5-dichlorobenzoyl)amino]acetyl]amino]-3-methylbutyl]boronic acid | CAS Registry Number: 1072833-77-2 Synonyms: MLN2238, CHEMBL2141296, MLN 2238, MLN-2238, (R)-1-(2-(2,5-dichlorobenzamido)acetamido)-3-methylbutylboronic acid, MLN 2238, MLN2238, Ixazomib [INN], Ixazomib (USAN), S2180_Selleck, Ixazomib [USAN:INN], SureCN3742758, cc-437, CTK4A5116, MolPort-016-633-297, UNII-71050168A2, AKOS015995120, AG-I-03417, BCP9000953, RL00318, MLN2238-Supplied by Selleck Chemicals
InChIKey: MXAYKZJJDUDWDS-LBPRGKRZSA-N | ||||||||
| • JNJ-38877605
IUPAC Name: 6-[difluoro-[6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]methyl]quinoline | CAS Registry Number: 943540-75-8 Synonyms: JNJ38877605, JNJ 38877605, 6-(difluoro(6-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methyl)quinoline, JNJ-38877605, JNJ 38877605, 943540-75-8, 6-[Difluoro[6-(1-methyl-1H-pyrazol-4-yl)-1,2,4-triazolo[4,3-b]pyridazin-3-yl]methyl]quinoline, JNJ38877605, JNJ-38877605, Quinoline, 6-(difluoro(6-(1-methyl-1H-pyrazol-4-yl)-1,2,4-triazolo(4,3-b)pyridazin-3-yl)methyl)-, Quinoline, 6-[difluoro[6-(1-methyl-1H-pyrazol-4-yl)-1,2,4-triazolo[4,3-b]pyridazin-3-yl]methyl]-, S1114_Selleck, PubChem22454, cc-51, SureCN182199, UNII-15UDG410PN, QCR-226, HMS3244G09, HMS3244G10, HMS3244H09, ABP000134, RS0066, AKOS015896605
InChIKey: JRWCBEOAFGHNNU-UHFFFAOYSA-N | ||||||||
| • JNJ-7706621
IUPAC Name: 4-[[5-amino-1-(2,6-difluorobenzoyl)-1,2,4-triazol-3-yl]amino]benzenesulfonamide | CAS Registry Number: 443797-96-4 Synonyms: JNJ7706621, JNJ 7706621, JNJ7706621, 443797-96-4, 4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)benzenesulfonamide, 4-[[5-Amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]benzenesulfonamide, JNJ7706621, JNJ-7706621, 3ama, 4-((5-Amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-yl)amino)benzenesulfonamide, 4-[[5-amino-1-(2,6-difluorobenzoyl)-1,2,4-triazol-3-yl]amino]benzenesulfonamide, 4-{[5-amino-1-(2,6-difluorobenzoyl)-1,2,4-triazol-3-yl]amino}benzenesulfonamide, RWJ-387252, S1249_Selleck, Kinome_3748, PubChem22455, AC1NS9N9, SureCN1060773, UNII-74GK72DON8, cc-474, CHEMBL191003, CTK1D4880
InChIKey: KDKUVYLMPJIGKA-UHFFFAOYSA-N | ||||||||
| • JNK-IN-8
IUPAC Name: 3-[[(E)-4-(dimethylamino)but-2-enoyl]amino]-N-[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide | CAS Registry Number: 1410880-22-6 Synonyms: CHEMBL2216824, CS-0601, HY-13319, JNK-IN-8|1410880-22-6, S4901,1410880-22-6
InChIKey: GJFCSAPFHAXMSF-UXBLZVDNSA-N | ||||||||
| • KI8751
IUPAC Name: 1-(2,4-difluorophenyl)-3-[4-(6,7-dimethoxyquinolin-4-yl)oxy-2-fluorophenyl]urea | CAS Registry Number: 228559-41-9 Synonyms: Ki8751, Ki 8751, Ki-8751, Ki8751, S1363_Selleck, AGN-PC-006NWD, SureCN1249562, cc-604, CHEMBL178455, CTK8E8844, CHEBI:399423, MolPort-021-804-894, HMS3269O17, Ki-8751, ABP001020, Ki8751-Supplied by Selleck Chemicals, BCP9000009, CS-0190, NCGC00167768-01, NCGC00167768-02, HY-12038
InChIKey: LFKQSJNCVRGFCC-UHFFFAOYSA-N | ||||||||
| • KRN-633
IUPAC Name: 1-[2-chloro-4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-3-propylurea | CAS Registry Number: 286370-15-8 Synonyms: KRN 633, CHEMBL406381, KRN633, S1557_Selleck, K00589a, VEGF Receptor Tyrosine Kinase Inhibitor III, KRN633, KRN633, KRN-633, KRN 633, N-(2-Chloro-4-((6,7-dimethoxy-4-quinazolinyl)oxy)phenyl)-N′-propylurea, 1-(2-chloro-4-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-propylurea, CID9549295, SureCN1249684, cc-528, MolPort-016-633-236, DCL000355, FD7289, CS-0220, RL02972, KRN 633-Supplied by Selleck Chemicals, NCGC00346548-01, HY-12060
InChIKey: VPBYZLCHOKSGRX-UHFFFAOYSA-N | ||||||||
| • KU-0060648
IUPAC Name: 2-(4-ethylpiperazin-1-yl)-N-[4-(2-morpholin-4-yl-4-oxochromen-8-yl)dibenzothiophen-1-yl]acetamide;trihydrochloride | CAS Registry Number: 881375-00-4
InChIKey: UPQYIHWLJGXREE-UHFFFAOYSA-N | ||||||||
| • KU-0063794
IUPAC Name: [5-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-morpholin-4-ylpyrido[2,3-d]pyrimidin-7-yl]-2-methoxyphenyl]methanol | CAS Registry Number: 938440-64-3 Synonyms: Ku-0063794, KU0063794, KU-63794, KU 0063794, KU0063794, 938440-64-3, KU0063794, KU-0063794, S1226_Selleck, PubChem22475, cc-34, SureCN290211, UNII-81HJG228AB, CHEMBL1078983, CHEBI:716942, MolPort-018-493-667, ACT06824, ABP000901, RS0068, AKOS005145564, BCP9000821, CS-0065
InChIKey: RFSMUFRPPYDYRD-CALCHBBNSA-N | ||||||||
| • KU-55933
IUPAC Name: 2-morpholin-4-yl-6-thianthren-1-ylpyran-4-one | CAS Registry Number: 587871-26-9 Synonyms: nchembio.63-comp3, nchembio800-comp3, nchembio800_comp3, ATM Kinase Inhibitor, CHEBI:472228, AIDS284437, AIDS-284437, 2-Morpholin-4-yl-6-thianthren-1-yl-pyran-4-one, CID5278396, EC-000.1920, 2-Morpholin-4-yl-6-thianthren-1-ylpyran-4-one, C495818, 2-Morpholino-6-(thianthren-1-yl)-4H-pyran-4-one, CU-00000000010-1, 4H-Pyran-4-one, 2-(4-morpholinyl)-6-(1-thianthrenyl)-
InChIKey: XRKYMMUGXMWDAO-UHFFFAOYSA-N | ||||||||
| • KU-57788
IUPAC Name: 8-dibenzothiophen-4-yl-2-morpholin-4-ylchromen-4-one | CAS Registry Number: 503468-95-9 Synonyms: NU7441, NU 7441, KU57788, NU-7441, NU7441(KU-57788), SureCN600096, AGN-PC-006VBM, cc-207, CHEMBL188678, CTK8F0292, CHEBI:415023, HMS3265K11, HMS3265K12, HMS3265L11, HMS3265L12, ABP000502, DNC005258, RS0029, BCP9000823, NU-7432
InChIKey: JAMULYFATHSZJM-UHFFFAOYSA-N | ||||||||
| • KU60019
IUPAC Name: 2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-N-[5-(6-morpholin-4-yl-4-oxopyran-2-yl)-9H-thioxanthen-2-yl]acetamide | CAS Registry Number: 925701-49-1 Synonyms: KU-60019, ku60019, KU 60019, S1570_Selleck, cc-509, MolPort-016-633-240, CS-0221, RL05828, NCGC00229735-01, NCGC00229735-02, NCGC00229735-03, HY-12061, KB-53044, KU-60019-Supplied by Selleck Chemicals, X7426, KU-60019|925701-49-1|KU 60019, KU60019,KU 60019,925701-49-1, pound molweight:547.66512) , KU60019 , KU 60019 , 925701-49-1, 2-((2S,6R)-2,6-dimethylmorpholino)-N-(5-(6-morpholino-4-oxo-4H-pyran-2-yl)-9H-thioxanthen-2-yl)acetamide, 2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-{5-[6-(morpholin-4-yl)-4-oxopyran-2-yl]-9H-thioxanthen-2-yl}acetamide
InChIKey: SCELLOWTHJGVIC-BGYRXZFFSA-N | ||||||||
| • KW-2449
IUPAC Name: [4-[(E)-2-(1H-indazol-3-yl)ethenyl]phenyl]-piperazin-1-ylmethanone | CAS Registry Number: 1000669-72-6 Synonyms: KW2449, KW 2449, CHEMBL1908397, 1000669-72-6 , KW 2449, KW-2449, KW 2449, KW2449, S2158_Selleck, SureCN1596894, cc-533, MolPort-016-633-288, BCP9000826, CS-0231, RL00013, KW 2449-Supplied by Selleck Chemicals, HY-10339, KB-78038, X7371, KW-2449|1000669-72-6|KW2449, [4-[2-(1H-Indazol-3-yl)ethenyl]phenyl]-1-piperazinylmethanone, 3-[(E)-2-[4-(piperazine-1-carbonyl)phenyl]ethenyl]-1H-indazole, (E)-(4-(2-(1H-indazol-3-yl)vinyl)phenyl)(piperazin-1-yl)methanone
InChIKey: YYLKKYCXAOBSRM-JXMROGBWSA-N | ||||||||
| • KW-2478
IUPAC Name: 2-[2-ethyl-3,5-dihydroxy-6-[3-methoxy-4-(2-morpholin-4-ylethoxy)benzoyl]phenyl]-N,N-bis(2-methoxyethyl)acetamide | CAS Registry Number: 819812-04-9 Synonyms: 819812-04-9 pound not KW2478 pound not KW 2478, UNII-QY50S617NM, cc-326, BCPP000191, BCP9000825, KW 2478, QC-7253, RL05131, NCGC00346685-01, BCP0726000279, KB-145989, 2-(2-ethyl-3,5-dihydroxy-6-(3-methoxy-4-(2-morpholinoethoxy)benzoyl)phenyl)-N,N-bis(2-methoxyethyl)acetamide, 2-(2-ethyl-3,5-dihydroxy-6-{3-methoxy-4-[2-(morpholin-4-yl)ethoxy]benzoyl}phenyl)-N,N-bis(2-methoxyethyl)acetamide, 2-ethyl-3,5-dihydroxy-n,n-bis(2-methoxyethyl)-6-(3-methoxy-4-(2-(4-morpholinyl)ethoxy)benzoyl)benzeneacetamide
InChIKey: VFUXSYAXEKYYMB-UHFFFAOYSA-N | ||||||||
| • Lactacystin
IUPAC Name: (2R)-2-acetamido-3-[(3S,4R)-3-hydroxy-2-[(1S)-1-hydroxy-2-methylpropyl]-4-methyl-5-oxopyrrolidine-2-carbonyl]sulfanylpropanoic acid | CAS Registry Number: 133343-34-7 Synonyms: lactacystin, NChemBio.2007.16-comp4, C15H24N2O7S, CHEBI:606509, Bio1_000949, CID3034764, LS-172867, L-Cysteine, N-acetyl-, (2R,3S,4R)-3-hydroxy-2-(1-hydroxy-2-methylpropyl)-4-methyl-5-oxo-2-pyrrolidinecarboxylate (ester), L-Cysteine, N-acetyl-, 3-hydroxy-2-(1-hydroxy-2-methylpropyl)-4-methyl-5-oxo-2-pyrrolidinecarboxylate (ester), (2R-(2alpha,2(S*),3alpha,4alpha))-, (R)-2-acetamido-3-((3S,4R)-3-hydroxy-2-((S)-1-hydroxy-2-methylpropyl)-4-methyl-5-oxopyrrolidine-2-carbonylthio)propanoic acid
InChIKey: DAQAKHDKYAWHCG-WVDSPMRNSA-N | ||||||||
| • Lapatinib
IUPAC Name: N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[(2-methylsulfonylethylamino)methyl]furan-2-yl]quinazolin-4-amine | CAS Registry Number: 231277-92-2 Synonyms: Tykerb, Lapatinib [INN], 1xkk, Lapatinib Ditosylate, nchembio866-comp20, Lapatinib tosilate hydrate, GW572016, CHEBI:49603, GSK 572016, GW 572016, CID208908, DB01259, NCGC00167507-01, LS-187029, LS-187771, FMM, N-{3-CHLORO-4-[(3-FLUOROBENZYL)OXY]PHENYL}-6-[5-({[2-(METHYLSULFONYL)ETHYL]AMINO}METHYL)-2-FURYL]-4-QUINAZOLINAMINE, 4-Quinazolinamine, N-(3-chloro-4-((3-fluorophenyl)methoxy)phenyl)-6-(5-(((2-(methylsulfonyl)ethyl)amino)methyl)-2-furanyl)-, N-(3-chloro-4-((3-fluorophenyl)methoxy)phenyl)-6-(5-(((2-(methylsulfonyl)ethyl)amino)methyl)-2-furanyl)-4-quinazolinamine, N-(3-Chloro-4-((3-fluorophenyl)methoxy)phenyl)-6-(5-((2-methylsulfonylethylamino)methyl)-2-furyl)quinazolin-4-amine
InChIKey: BCFGMOOMADDAQU-UHFFFAOYSA-N | ||||||||
| • LDN-57444
IUPAC Name: [[5-chloro-1-[(2,5-dichlorophenyl)methyl]-2-oxoindol-3-ylidene]amino] acetate | CAS Registry Number: 668467-91-2 Synonyms: AGN-PC-015JWF, CTK8E7168, IN1021, [(Z)-[5-chloro-1-[(2,5-dichlorophenyl)methyl]-2-oxoindol-3-ylidene]amino] acetate
InChIKey: OPQRFPHLZZPCCH-UHFFFAOYSA-N | ||||||||
| • LDN193189
IUPAC Name: 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | CAS Registry Number: 1062368-24-4 Synonyms: LDN 193189, LDN-193189, 4-(6-(4-(piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinoline, 4-{6-[4-(piperazin-1-yl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl}quinoline, S2618_Selleck, SureCN456393, UNII-W69H5YQU9O, cc-233, CHEMBL513147, CHEBI:588756, BCP9000845, CS-0669, DM 3189, DM-3189, EX-8677, RL00282, NCGC00249389-01, HY-12071, KB-78111, X7510
InChIKey: CDOVNWNANFFLFJ-UHFFFAOYSA-N | ||||||||
| • Lenalidomide
IUPAC Name: 3-(7-amino-3-oxo-1H-isoindol-2-yl)piperidine-2,6-dione | CAS Registry Number: 191732-72-6 Synonyms: Revlimid, Revimid, Revamid, IMiD3, Revlimid (TN), IMiD3 cpd, Lenalidomide [USAN], Lenalidomide (USAN/INN), CDC 501, CC-5013, Celgene brand of lenalidomide, Thalidomide analog CC-5013, STOCK6S-54938, CC 5013, ENMD-0997, IMID-5013, CDC-501, CDC-5013, CC5013, CID216326
InChIKey: GOTYRUGSSMKFNF-UHFFFAOYSA-N | ||||||||
| • Lenvatinib
IUPAC Name: 4-[3-chloro-4-(cyclopropylcarbamoylamino)phenoxy]-7-methoxyquinoline-6-carboxamide | CAS Registry Number: 417716-92-8 Synonyms: CID9823820, E7080, 4-[3-chloro-4-(cyclopropylcarbamoylamino)phenoxy]-7-methoxy-quinoline-6-carboxamide, 6-Quinolinecarboxamide, 4-(3-chloro-4- (((cyclopropylamino)carbonyl)amino)phenoxy)-7-methoxy-, 942407-57-0
InChIKey: WOSKHXYHFSIKNG-UHFFFAOYSA-N | ||||||||
| • Letrozole
IUPAC Name: 4-[(4-cyanophenyl)-(1,2,4-triazol-1-yl)methyl]benzonitrile | CAS Registry Number: 112809-51-5 Synonyms: letrozole, Femara, Letrozol, Femera, F?mara, Femara (TN), Letrozole [USAN:INN], Prestwick0_001025, Prestwick1_001025, Prestwick2_001025, Prestwick3_001025, Novartis Brand of Letrozole, Letrozole (JAN/USP/INN), BSPBio_001209, MLS000759455, MLS001424038, SPBio_003070, CGS 20267, CGS-20267, BPBio1_001331
InChIKey: HPJKCIUCZWXJDR-UHFFFAOYSA-N | ||||||||
| • Lexibulin
IUPAC Name: 1-ethyl-3-[2-methoxy-4-[5-methyl-4-[[(1S)-1-pyridin-3-ylbutyl]amino]pyrimidin-2-yl]phenyl]urea | CAS Registry Number: 917111-44-5 Synonyms: CYT997, LEXIBULIN, CYT-997, CYT 997, Lexibulin [INN], Lexibulin (USAN), S2195_Selleck, Lexibulin [USAN:INN], SureCN1122311, UNII-2GTU230HA1, cc-400, CHEMBL552212, MolPort-016-633-306, CYT997-Supplied by Selleck Chemicals, BCP9000572, CYT9970000, QC-8216, RL05776, NCGC00346574-01, X7569
InChIKey: MTJHLONVHHPNSI-IBGZPJMESA-N | ||||||||
| • Linagliptin
IUPAC Name: 8-[(3R)-3-aminopiperidin-1-yl]-7-but-2-ynyl-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]purine-2,6-dione | CAS Registry Number: 668270-12-0 Synonyms: Ondero, CHEBI:499873, BI-1356-BS, BI 1356, BI-1356, CID10096344, CID 10096344, (R)-8-(3-Amino-piperidin-1-yl)-7-but-2-ynyl-3-methyl-1-(4-methyl-quinazolin-2-ylmethyl)-3,7-dihydro-purine-2,6-dione, (R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-methyl-1-((4-methylquinazolin-2-yl)methyl)-1H-purine-2,6(3H,7H)-dione, 1H-Purine-2,6-dione, 8-((3R)-3-amino-1-piperidinyl)-7-(2-butynyl)-3,7-dihydro-3-methyl-1-((4-methyl-2-quinazolinyl)methyl)-
InChIKey: LTXREWYXXSTFRX-QGZVFWFLSA-N | ||||||||
| • Linifanib
IUPAC Name: 1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-5-methylphenyl)urea | CAS Registry Number: 796967-16-3 Synonyms: ABT-869, ABT 869, CHEBI:471147, CID11485656, EC-000.2119, N-(4-(3-Amino-1H-indazol-4-yl)phenyl)-N'-(2-fluoro-5-methylphenyl)urea, 1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-(2-fluoro-5-methylphenyl)urea, N-(4-(3-Amino-1H-indazol-4-yl)phenyl)-N1-(2-fluoro-5-methylphenyl)urea, N-[4-(3-amino-1H-indazol-4-yl)phenyl]-N'-(2-fluoro-5-methylphenyl)urea, Urea, N-(4-(3-amino-1H-indazol-4-yl)phenyl)-N'-(2-fluoro-5-methylphenyl)-
InChIKey: MPVGZUGXCQEXTM-UHFFFAOYSA-N | ||||||||
| • Linsitinib
IUPAC Name: 3-[8-amino-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl]-1-methylcyclobutan-1-ol | CAS Registry Number: 867160-71-2 Synonyms: OSI-906, Kinome_3532, OSI-906AA, OSI906, OSI-906, 867160-71-2, 3-[8-amino-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl]-1-methylcyclobutan-1-ol, cis-3-(8-amino-1-(2-phenyl-7-quinolinyl)imidazo(1,5-a)pyrazin-3-yl)-1-methylcyclobutanol, cis-3-[8-Amino-1-(2-phenyl-7-quinolinyl)imidazo[1,5-a]pyrazin-3-yl]-1-methylcyclobutanol, Linsitinib [USAN], Linsitinib (USAN/INN), SureCN400369, SureCN400734, SureCN400735, AGN-PC-00D7QU, UNII-15A52GPT8T, SureCN10255925, cc-217, CHEMBL1091644, OSI 906, QCR-128
InChIKey: PKCDDUHJAFVJJB-UHFFFAOYSA-N | ||||||||
| • Lobaplatin
IUPAC Name: [2-(aminomethyl)cyclobutyl]methanamine; 2-oxidopropanoate; platinum(2+) | CAS Registry Number: 135558-11-1 Synonyms: Lobaplatin [INN], Lobaplatine [INN-French], Lobaplatinum [INN-Latin], Lobaplatino [INN-Spanish], D 19466, cis-(trans-1,2-Cyclobutanebis(methylamine))((S)-lactato-O(sup 1),O(sup 1))platinum, Platinum, (1,2-cyclobutanedimethanamine-N,N')(2-hydroxypropanoato(2-)-O1,O2)-, (SP-4-3-(S),(trans))-, Platinum, (rel-(1R,2R)-1,2-cyclobutanedimethanamine-kappaN,kappaN')((2S)-2-(hydroxy-kappa-O)propanoato(2-)-kappaO)-, (SP-4-3)-
InChIKey: RLXPIABKJFUYFG-UHFFFAOYSA-M | ||||||||
| • Lomeguatrib
IUPAC Name: 6-[(4-bromothiophen-2-yl)methoxy]-7H-purin-2-amine | CAS Registry Number: 192441-08-0 Synonyms: PaTrin 2, Lomeguatrib [INN], UNII-S79265T71M, CHEBI:316928, 6-(4-Bromothenyloxy)-7H-purin-2-amine, CID3025944, LS-184193, 6-((4-bromo-2-thienyl)methoxy)purin-2-amine, 6-((4-Bromo-2-thienyl)methoxyl)purin-2-amine, C521206, 6-(4-Bromo-thiophen-2-ylmethoxy)-9H-purin-2-ylamine, 793035-44-6
InChIKey: JUJPKFNFCWJBCX-UHFFFAOYSA-N | ||||||||
| • Loperamide hydrochloride
IUPAC Name: 4-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-N,N-dimethyl-2,2-di(phenyl)butanamide hydrochloride | CAS Registry Number: 34552-83-5 Synonyms: Imodium, Loperamide HCl, Dissenten, Fortasec, Suprasec, Lopemid, Lopemin, Loperyl, Imosec, Tebloc, Imodium A-D, Maalox Antidiarrheal, BLOX, BREK, Prestwick_302, Imodium (TN), IMODIUM ADVANCED, C29H33ClN2O2.HCl, MLS000069779, MLS001148627
InChIKey: PGYPOBZJRVSMDS-UHFFFAOYSA-N | ||||||||
| • Lopinavir
IUPAC Name: (2S)-N-[(2S,4S,5S)-5-[[2-(2,6-dimethylphenoxy)acetyl]amino]-4-hydroxy-1,6-di(phenyl)hexan-2-yl]-3-methyl-2-(2-oxo-1,3-diazinan-1-yl)butanamide | CAS Registry Number: 192725-17-0 Synonyms: Aluviran, Kaletra, Koletra, Aluvia, Mixture Name, 1mui, ABT-378, Component of Kaletra, 2o4s, 2q5k, ABT 378, Lopinavir (JAN/USAN/INN), Lopinavir [USAN:INN:BAN], ABT-378, LOPINAVIR, RS-346, AIDS032937, C37H48N4O5, AIDS-032937, ABT 157378, DB01601
InChIKey: KJHKTHWMRKYKJE-SUGCFTRWSA-N | ||||||||
| • Luminespib
IUPAC Name: (5Z)-N-ethyl-5-(4-hydroxy-6-oxo-3-propan-2-ylcyclohexa-2,4-dien-1-ylidene)-4-[4-(morpholin-4-ylmethyl)phenyl]-2H-1,2-oxazole-3-carboxamide | CAS Registry Number: 747412-49-3 Synonyms: NVP-AUY922, VER-52296, AUY-922, AUY922 (NVP-AUY922), AUY922, VER-52296, 747412-49-3, 5-(2,4-dihydroxy-5-isopropylphenyl)-N-ethyl-4-(4-(morpholinomethyl)phenyl)isoxazole-3-carboxamide, 5-[2,4-DIHYDROXY-5-ISOPROPYLPHENYL]-N-ETHYL-4-[4-(4-MORPHOLINYLMETHYL)PHENYL]-3-ISOXAZOLECARBOXAMIDE, PubChem19135, UNII-C6V1DAR5EB, cc-237, NVP-AUY 922, AUY922,NVP-AUY922, QCR-179, BCPP000145, AUY922 - NVP-AUY922, VER52296, ABP000836, VER 52296, AKOS015966502, BCP9001007
InChIKey: SWDZPNJZKUGIIH-QQTULTPQSA-N | ||||||||
| • LY-364947
IUPAC Name: 4-(5-pyridin-2-yl-1H-pyrazol-4-yl)quinoline | CAS Registry Number: 396129-53-6 Synonyms: 4-(3-PYRIDIN-2-YL-1H-PYRAZOL-4-YL)QUINOLINE, TbetaR-I Inhibitor, ALK5 Inhibitor I, TGF-beta RI Kinase Inhibitor, LY364947, Transforming Growth Factor-beta Type I Receptor Kinase Inhibitor, LY 364947, [3-(Pyridin-2-yl)-4-(4-quinonyl)]-1H-pyrazole, PY1, 4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)quinoline, 4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline, HTS 466284, HTS-466284, 1py5, AC1L9LFY, Peakdale1_000394, SureCN373665, Ambpe3000655, cc-654, L6293_SIGMA
InChIKey: IBCXZJCWDGCXQT-UHFFFAOYSA-N | ||||||||
| • LY-411575
IUPAC Name: (2S)-2-[[(2S)-2-(3,5-difluorophenyl)-2-hydroxyacetyl]amino]-N-[(7S)-5-methyl-6-oxo-7H-benzo[d][1]benzazepin-7-yl]propanamide | CAS Registry Number: 209984-57-6 Synonyms: LY411575, LY 411575, 209984-57-6 pound not LY 411575 pound not LY-411575, SureCN33171, cc-581, CHEMBL392068, CHEBI:499634, BCP9000887, CS-0309, RL02594, NCGC00346841-01, HY-50752, LS-193033, LY-411575|209984-57-6|LY 411575, (2S)-2-[(2S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido]-N-[(10S)-8-methyl-9-oxo-8-azatricyclo[9.4.0.0^{2,7}]pentadeca-1(11),2(7),3,5,12,14-hexaen-10-yl]propanamide, ly 411575;(as)-n-((1s)-2-(((7s)-6,7-dihydro-5-methyl-6-oxo-5h-dibenz(b,d)azepin-7-yl)amino)-1-methyl-2-oxoethyl)-3,5-difluoro-alpha-hydroxybenzeneacetamide, M/A
InChIKey: ULSSJYNJIZWPSB-CVRXJBIPSA-N | ||||||||
| • LY2090314
Synonyms: Kinome_3681, SureCN633455, UNII-822M3GYM67, CHEMBL362558, CHEBI:411715, LY-2090314
InChIKey: HRJWTAWVFDCTGO-UHFFFAOYSA-N | ||||||||
| • LY2109761
IUPAC Name: 4-[2-[4-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)quinolin-7-yl]oxyethyl]morpholine | CAS Registry Number: 700874-71-1 Synonyms: LY 2109761, 700874-71-1 pound not LY-2109761 pound not LY 2109761, 4-(2-(4-(2-(pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)quinolin-7-yloxy)ethyl)morpholine, Dihydropyrrolopyrazole, 15d, AGN-PC-00DI8T, SureCN3737735, cc-120, CHEMBL260015, ACN-S001851, ABP001002, BCP9000868, CS-0571, QC-7261, RL04685, NCGC00242598-01, NCGC00242598-03, HY-12075, KB-53445, LY-2109761, LY2109761,CAS:700874-71-1
InChIKey: IHLVSLOZUHKNMQ-UHFFFAOYSA-N |