Profile: Jinan Trio PharmaTech Co., Ltd. specializes in APIs & intermediates, heterocyclic compounds, and anti-tumor drugs. Our products include crizotinib, vemurafenib, afatinib, vandetanib, regorafenib, brivanib alaninate, pyridazine, imidazole, pyrazole, and oxazole. We are specialized in providing over 1000 products including molecular targeted anticancer drugs, cell signaling pathway inhibitors, pharmaceutical intermediates, and heterocyclic compounds, and quality services including custom synthesis, transfer of new drug patent and technology, technical cooperation, and process optimization.
| • Serdemetan
IUPAC Name: 1-N-[2-(1H-indol-3-yl)ethyl]-4-N-pyridin-4-ylbenzene-1,4-diamine | CAS Registry Number: 881202-45-5 Synonyms: JNJ 26854165, N1-(2-(1H-Indol-3-yl)ethyl)-N4-(pyridin-4-yl)benzene-1,4-diamine, JNJ-26854165, Serdemetan, JNJ 26854165, 881202-45-5, JNJ26854165, Serdemetan, JNJ 26854165, n-(2-(1h-indol-3-yl)ethyl)-n'-(4-pyridinyl)-1,4-benzenediamine, N-[2-(1H-INDOL-3-YL)ETHYL]-N'-(4-PYRIDINYL)-1,4-BENZENEDIAMINE, Serdemetan [INN], S1172_Selleck, AGN-PC-00CLKV, UNII-ID6YB4W3V8, SureCN3012498, cc-450, CHEMBL2137530, CTK8C1936, JNJ-26854165 (Serdemetan), ANW-67474, QC-534, AKOS016006774, CS-0166
InChIKey: CEGSUKYESLWKJP-UHFFFAOYSA-N | ||||||||
| • SGI-1776
IUPAC Name: N-[(1-methylpiperidin-4-yl)methyl]-3-[3-(trifluoromethoxy)phenyl]imidazo[1,2-b]pyridazin-6-amine | CAS Registry Number: 1025065-69-3 Synonyms: SGI-1776 free base, CHEMBL1952329, SGI1776, SGI 1776, SGI-1776, SGI1776, N-((1-methylpiperidin-4-yl)methyl)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-amine, N-[(1-methylpiperidin-4-yl)methyl]-3-[3-(trifluoromethoxy)phenyl]imidazo[1,2-b]pyridazin-6-amine, S2198_Selleck, SureCN102498, cc-574, QCR-216, MolPort-016-633-308, ABP000939, CS-0513, RL00118, NCGC00263186-01, NCGC00263186-02, HY-13287, SGI-1776-Supplied by Selleck Chemicals, X7567
InChIKey: MHXGEROHKGDZGO-UHFFFAOYSA-N | ||||||||
| • SGX-523
IUPAC Name: 6-[[6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl]quinoline | CAS Registry Number: 1022150-57-7 Synonyms: CHEMBL1236107, S1112_Selleck, SGX523, SGX 523, SGX523, SGX-523, DB08584, 6-(6-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-ylthio)quinoline, SGX523, 1022150-57-7, 3dkf, 3dkg, PubChem19151, SureCN4496422, cc-382, ABP000132, DCL000229, CS-0154, RL00113, SGX-523-Supplied by Selleck Chemicals, NCGC00263163-01, NCGC00263163-02
InChIKey: BCZUAADEACICHN-UHFFFAOYSA-N | ||||||||
| • Sitagliptin phosphate monohydrate
IUPAC Name: (3R)-3-amino-1-[3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-4-(2,4,5-trifluorophenyl)butan-1-one; phosphoric acid; hydrate | CAS Registry Number: 654671-77-9 Synonyms: Januvia, Glactiv, Tesavel, Xelevia, Januvia (TN), Sitagliptin phosphate, Sitagliptin phosphate hydrate, Sitagliptin phosphate (USAN), ONO-5435, Sitagliptin phosphate hydrate (JAN), MK-431, MK-0431, D06645
InChIKey: GQPYTJVDPQTBQC-KLQYNRQASA-N | ||||||||
| • Skepinone-L
IUPAC Name: 3-(2,4-difluoroanilino)-9-[(2R)-2,3-dihydroxypropoxy]-5,6-dihydrodibenzo[3,1-[7]annulen-11-one | CAS Registry Number: 1221485-83-1 Synonyms: CHEMBL2152944, 3que, SureCN2686103, Skepinone-L|1221485-83-1, CS-0941, HY-15300, X5940, S7214,1221485-83-1, 2-(2,4-Difluorophenylamino)-7-[2R-,3-dihydroxypropoxy]-10,11-dihydro-dibenzo[a,d]-cyclohepten-5-one, 2-[(2,4-Difluorophenyl)amino]-7-{[(2r)-2,3-Dihydroxypropyl]oxy}-10,11-Dihydro-5h-Dibenzo[a,D][7]annulen-5-One, 3FF
InChIKey: HXMGCTFLLWPVFM-GOSISDBHSA-N | ||||||||
| • SL-01
IUPAC Name: benzyl N-[(2S)-4-chloro-3-oxo-1-phenylbutan-2-yl]carbamate | CAS Registry Number: 26049-94-5 Synonyms: ZPCK, Z-L-Phe chloromethyl ketone, Spectrum2_001493, Spectrum3_001809, Lopac-C-9511, Lopac0_000290, BSPBio_003397, MLS002153274, SPBio_001505, 860794_ALDRICH, KBio3_002900, CHEBI:196054, CID99625, EINECS 247-432-8, ZINC01583409, NSC 251810, NCGC00015284-01, NCGC00093742-01, NCGC00093742-02, NCGC00093742-03
InChIKey: OYHLRJGDELITAF-INIZCTEOSA-N | ||||||||
| • SL327
IUPAC Name: (Z)-3-amino-3-(4-aminophenyl)sulfanyl-2-[2-(trifluoromethyl)phenyl]prop-2-enenitrile | CAS Registry Number: 305350-87-2 Synonyms: MEK1/2 Inhibitor, SL-327, CHEMBL261237, Z-& E-alpha-(Amino-((4-aminophenyl)thio)methylene)-2-(trifluoromethyl)benzeneacetonitrile, SureCN570317, K00090, HMS3229K18, HSCI1_000044, CCG-206867, CS-0910, NCGC00092290-01, NCGC00092290-02, HY-15437, KB-80585, LS-193345, BRD-K12244279-001-01-7, SL327|305350-87-2|SL-327, (Z)-3-amino-3-(4-aminophenylthio)-2-(2-(trifluoromethyl)phenyl)acrylonitrile, |A-[Amino-(4-aminophenylthio)methylene)-2-(trifluoromethyl)phenylacetonitrile, Z-& E-a-(Amino-((4-aminophenyl)thio)methylene)-2-(trifluoromethyl)benzeneacetonitrile
InChIKey: JLOXTZFYJNCPIS-FYWRMAATSA-N | ||||||||
| • SMER3
Synonyms: indeno[2,3-b]1,2,5-oxadiazolo[3,4-e]pyrazin-5-one, BAS 01964143, AC1LC37B, SureCN7984580, Oprea1_175199, Oprea1_783821, STOCK1S-64064, MolPort-001-970-903, HMS1607O01, SBB000632, STK120842, ZINC00027763, AKOS000479457, MCULE-1070513713, KB-74322, ST000573, Indeno[1,2-b]furazano[3,4-E]pyrazin-9-one, Indeno[1,2-b]furazano[3,4-E]pyrazin-9-one,, 2-Oxa-1,3,4,10-tetraaza-cyclopenta[b]fluoren-9-one, 9H-Indeno[1,2-e][1,2,5]oxadiazolo[3,4-b]pyrazin-9-one
InChIKey: SFSSAKVWCKFRHE-UHFFFAOYSA-N | ||||||||
| • SNS-032
IUPAC Name: N-[5-[(5-tert-butyl-1,3-oxazol-2-yl)methylsulfanyl]-1,3-thiazol-2-yl]piperidine-4-carboxamide | CAS Registry Number: 345627-80-7 Synonyms: BMS-387032, BMS-387072, CID3025986, LS-186036, N-(5-(((5-(1,1-Dimethylethyl)-2-oxazolyl)methyl)thio)-2-thiazolyl)-4-piperidinecarboxamide, 4-Piperidinecarboxamide, N-(5-(((5-(1,1-dimethylethyl)-2-oxazolyl)methyl)thio)-2-thiazolyl)-
InChIKey: OUSFTKFNBAZUKL-UHFFFAOYSA-N | ||||||||
| • SNS-314 Mesylate
IUPAC Name: 1-(3-chlorophenyl)-3-[5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl]urea;methanesulfonic acid | CAS Registry Number: 1146618-41-8 Synonyms: SNS-314, SNS314, SNS-314 Mesylate, CHEMBL518051, SNS 314, S1154_Selleck, UNII-KGW32FDY3U, cc-347, SNS314, MolPort-016-633-186, AKOS015904656, CS-0113, RL00570, HY-12003, X7391, SNS-314 Mesylate-Supplied by Selleck Chemicals, I14-17005, SNS-314|1146618-41-8|SNS314|SNS 314, 1-(3-chlorophenyl)-3-[5-(2-{thieno[3,2-d]pyrimidin-4-ylamino}ethyl)-1,3-thiazol-2-yl]urea mesylate, N-(3-Chlorophenyl)-N'-[5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-2-thiazolyl]urea methanesulfonate (1:1), Urea, N-(3-chlorophenyl)-N'-(5-(2-(thieno(3,2-d)pyrimidin-4-ylamino)ethyl)-2-thiazolyl)-, methanesulfonate (1:1)
InChIKey: FYCODPVDEFFWSR-UHFFFAOYSA-N | ||||||||
| • SNX2112
IUPAC Name: 4-[6,6-dimethyl-4-oxo-3-(trifluoromethyl)-5,7-dihydroindazol-1-yl]-2-[(4-hydroxycyclohexyl)amino]benzamide | CAS Registry Number: 908112-43-6 Synonyms: SNX-2112, SNX 2112, CHEMBL560895, SNX 2112, SNX2112, 908112-43-6, HIE, PF-04928473, UNII-10C9P3FFOW, SureCN1219380, SureCN1219382, SureCN1221195, SureCN12685879, cc-397, CHEMBL561224, DNC014879, CS-0481, RL05705, NCGC00346633-01, HY-10214, BCP0726000309, FT-0660383
InChIKey: ZFVRYNYOPQZKDG-UHFFFAOYSA-N | ||||||||
| • sodium 2-(2-aminophenyl)-2-hydroxyacetate
IUPAC Name: sodium;2-(2-aminophenyl)-2-hydroxyacetate | CAS Registry Number: 39588-85-7 Synonyms: Sodium 2-(2-aminophenyl)-2-hydroxyacetate, SureCN9191810, CTK8C2290, ANW-68151, AKOS016007083, AK-80682, KB-259744
InChIKey: DMLZRJSMMIQZIZ-UHFFFAOYSA-M | ||||||||
| • Sodium 2-(2-aminophenyl)-2-oxoacetate
IUPAC Name: sodium;2-(2-aminophenyl)-2-oxoacetate | CAS Registry Number: 17617-34-4 Synonyms: CTK8C2312, ANW-68188, AKOS016007258, AK-80636, KB-259745
InChIKey: XCFAFIKPWWFZPL-UHFFFAOYSA-M | ||||||||
| • Sodium 4-aminosalicylate dihydrate
IUPAC Name: 4-amino-2-hydroxybenzoic acid | CAS Registry Number: 6018-19-5 Synonyms: Aminosalicylic acid, 4-Aminosalicylic acid, Pamisyl, Rezipas, Parasalicil, Parasalindon, Gabbropas, Paramycin, Aminopar, Deapasil, Ferrosan, Pasnodia, Entepas, Pamacyl, Parasal, Pasalon, Pasdium, Pasolac, Propasa, Aminox
InChIKey: WUBBRNOQWQTFEX-UHFFFAOYSA-N | ||||||||
| • Sonidegib
IUPAC Name: N-[6-[(2S,6R)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]-2-methyl-3-[4-(trifluoromethoxy)phenyl]benzamide | CAS Registry Number: 956697-53-3 Synonyms: Erismodegib, LDE225, NVP-LDE225, LDE 225, LDE-225, NVP-LDE 225, LDE225, NVP-LDE225, Sonidegib (INN), N-(6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl)-2-methyl-3-[4-(trifluoromethoxy)phenyl]benzamide, N-{6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl}-2-methyl-3-[4-(trifluoromethoxy)phenyl]benzamide, Erismodegib [INN], Erismodegib (USAN), S2151_Selleck, PubChem22446, UNII-0RLU3VTK5M, Erismodegib [USAN:INN], cc-76, SureCN554455, CHEMBL2105737, MolPort-009-194-121
InChIKey: VZZJRYRQSPEMTK-CALCHBBNSA-N | ||||||||
| • Sorafenib
IUPAC Name: 4-[4-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-N-methylpyridine-2-carboxamide | CAS Registry Number: 284461-73-0 Synonyms: Nexavar, sorafenibum, Sorafenib tosylate, Sorafenib [INN], nchembio.117-comp17, STOCK6S-50043, CHEBI:50924, K00597a, BAY 43-9006, BAY 439006, DB00398, NSC-724772, BAY-43-0006, BAY-43-9006, BAY-54-9085, NCGC00167488-01, LS-186067, LS-187021, LS-187788, N-(4-Chloro-3-(trifluoromethyl)phenyl)-N'-(4-(2-(N-methylcarbamoyl)-4-pyridyloxy)phenyl)urea
InChIKey: MLDQJTXFUGDVEO-UHFFFAOYSA-N | ||||||||
| • Sotrastaurin
IUPAC Name: 3-(1H-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]pyrrole-2,5-dione | CAS Registry Number: 425637-18-9 Synonyms: AEB071, AEB-071, AEB 071, Sotrastaurin acetate, 3-(1H-Indol-3-yl)-4-(2-(4-methylpiperazin-1-yl)quinazolin-4-yl)-1H-pyrrole-2,5-dione, 3-(1h-Indol-3-Yl)-4-[2-(4-Methylpiperazin-1-Yl)quinazolin-4-Yl]-1h-Pyrrole-2,5-Dione, Kinome_2717, Sotrastaurin (AEB071), Sotrastaurin (USAN/INN), SureCN2500835, NVP-AEB-071, UNII-7I279E1NZ8, CHEMBL565612, DCL000996, CS-0090, NCGC00238621-01, HY-10343, Y6229, D09671, Sotrastaurin|425637-18-9|AEB 071|AEB-071
InChIKey: OAVGBZOFDPFGPJ-UHFFFAOYSA-N | ||||||||
| • SP600125
Synonyms: Pyrazolanthrone, Pyrazoleanthrone, 1,9-Pyrazoloanthrone, Anthrapyrazolone, 1pmv, JNK Inhibitor II, SAPK Inhibitor II, Tocris-1496, BiomolKI_000068, Lopac-S-5567, BiomolKI2_000072, Anthra[1,9-cd]pyrazol-6(2H)-one, CBiol_002049, Lopac0_000473, Anthra-1,9-pyrazol-6-none, BSPBio_001066, KBioGR_000406, KBioSS_000406, MLS002153267, Bio-0879
InChIKey: ACPOUJIDANTYHO-UHFFFAOYSA-N | ||||||||
| • Stattic
IUPAC Name: 6-nitro-1-benzothiophene 1,1-dioxide | CAS Registry Number: 19983-44-9 Synonyms: Stat three inhibitory compound, 6-nitro-1-benzothiophene 1,1-dioxide, STAT3 Inhibitor V, Stattic, CHEMBL1337170, 6-Nitrobenzo[b]thiophene 1,1-dioxide, 6-Nitrobenzo[b]thiophene-1,1-dioxide, ZINC00162014, 6-nitro-1, AC1MCWHD, Maybridge1_005148, STAT3 INHIBITOR V, AC1Q1Y5K, SureCN1156180, CTK8E5442, HMS556B22, MolPort-000-880-821, 6-nitrobenzo[b]thiole-1,1-dione, HMS3263A18, SBB094472, AKOS000276641
InChIKey: ZRRGOUHITGRLBA-UHFFFAOYSA-N | ||||||||
| • Staurosporine
Synonyms: staurosporine, Staurosporin, (+)-Staurosporine, Antibiotic 230, 1nvr, 1stc, 1xbc, 1xjd, 1yhs, 2gcd, Antibiotic AM 2282, nchembio.87-comp4, nchembio809-comp4, Staurosporine & TNF, nchembio.162-comp3, 1q3d, 1sm2, 2dq7, CCRIS 3272, MolMap_000047
InChIKey: HKSZLNNOFSGOKW-FYTWVXJKSA-N | ||||||||
| • SU11274
IUPAC Name: (3Z)-N-(3-chlorophenyl)-3-[[3,5-dimethyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrrol-2-yl]methylidene]-N-methyl-2-oxo-1H-indole-5-sulfonamide | CAS Registry Number: 658084-23-2 Synonyms: Met Kinase Inhibitor, SU 11274, SU-11274, PKI-SU11274, PKI-SU11274, 658084-23-2, (3Z)-N-(3-Chlorophenyl)-3-((3,5-dimethyl-4-((4-methylpiperazin-1-yl)carbonyl)-1H-pyrrol-2-yl)methylene)-N-methyl-2-oxo-2,3-dihydro-1H-indole-5-sulfonamide, (3Z)-N-(3-Chlorophenyl)-3-({3,5-dimethyl-4-[(4-methylpiperazin-1-yl)carbonyl]-1H-pyrrol-2-yl}methylene)-N-methyl-2-oxo-2,3-dihydro-1H-indole-5-sulfonamide, PKI-SU11274, SU11274, S1080_Selleck, PubChem19146, SureCN93711, SU-MI-2, S9820_SIGMA, CHEMBL261641, CHEBI:529088, MolPort-003-959-612, BCPP000061, HMS3229G21, K00593a, N-(3-Chlorophenyl)-N-methyl-3-[[3,5-dimethyl-4-[(4-methylpiperazin-1-yl)carbonyl]-1H-pyrrol-2-yl]methylene]-2-oxo-2,3-dihydro-1H-indole-5-sulfonamide
InChIKey: FPYJSJDOHRDAMT-KQWNVCNZSA-N | ||||||||
| • Sulfacetamide sodium
IUPAC Name: sodium acetyl-(4-aminophenyl)sulfonylazanide | CAS Registry Number: 127-56-0 Synonyms: Sulfacetamide sodium anhydrous, ST5407307, AB00513796, C08051
InChIKey: PQMSFAORUFMASU-UHFFFAOYSA-M | ||||||||
| • Sunitinib
IUPAC Name: N-(2-diethylaminoethyl)-5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide | CAS Registry Number: 557795-19-4 Synonyms: Sutent, Sunitanib, Sunitinib malate, PDGF TK antagonist, STOCK6S-48542, Su-011248, CHEBI:38940, SU-11248, K00588a, SU11248, NSC736511, SU-11248J, SU 11248, DB01268, NCGC00164631-01, SU-12662, LS-187023, LS-187648, 1H-Pyrrole-3-carboxamide, N-(2-(diethylamino)ethyl)-5-((Z)-(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-2,4-dimethyl-, 1H-Pyrrole-3-carboxamide, N-[2-(diethylamino)ethyl]-5-[(Z)- (5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl]-2,4-dimethyl-
InChIKey: WINHZLLDWRZWRT-ATVHPVEESA-N | ||||||||
| • Sunitinib Malate
IUPAC Name: N-(2-diethylaminoethyl)-5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide; (2S)-2-hydroxybutanedioic acid | CAS Registry Number: 341031-54-7 Synonyms: Sunitinib malate, Sutent, Sutent (TN), Sunitinib malate [USAN], SU011248 L-malate salt, SU-11248 L-malate salt, PHA-290940AD, Sunitinib malate (JAN/USAN), SU-011248 L-malate salt, PNU-290940AD, SU010398, CID6456015, SU 011248, SU011248, LS-186078, SU-010398, TL8002546, D06402, Butanedioic acid, hydroxy-, (2S)-, compd. with N-(2-(diethylamino)ethyl)-5-((Z)-(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-2,4-dimethyl-1H-pyrrole-3-carboxamide (1:1), 1H-Pyrrole-3-carboxamide, N-(2-(diethylamino)ethyl)-5-((Z)-(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-2,4-dimethyl-, (2S)-hydroxybutanedioate (1:1)
InChIKey: LBWFXVZLPYTWQI-IPOVEDGCSA-N | ||||||||
| • TAK-285
IUPAC Name: N-[2-[4-[3-chloro-4-[3-(trifluoromethyl)phenoxy]anilino]pyrrolo[3,2-d]pyrimidin-5-yl]ethyl]-3-hydroxy-3-methylbutanamide | CAS Registry Number: 871026-44-7 Synonyms: CHEMBL1614725, 3poz, 3rcd, 03P, n-(2-(4-((3-chloro-4-(3-(trifluoromethyl)phenoxy)phenyl)amino)-5h-pyrrolo(3,2-d)pyrimidin-5-yl)ethyl)-3-hydroxy-3-methylbutanamide, N-{2-[4-({3-Chloro-4-[3-(Trifluoromethyl)phenoxy]phenyl}amino)-5h-Pyrrolo[3,2-D]pyrimidin-5-Yl]ethyl}-3-Hydroxy-3-Methylbutanamide, AGN-PC-00CTSA, SureCN982278, cc-290, UNII-70CCB438L6, TAK 285, TAK285/TAK-285, CS-0774, RL05409, NCGC00346699-01, HY-15196, KB-80787, BCP0726000091, TAK-285|871026-44-7|TAK 285, N-[2-[4-[3-chloro-4-[3-(trifluoromethyl)phenoxy]anilino]pyrrolo[3,2-d]pyrimidin-5-yl]ethyl]-3-hydroxy-3-methylbutanamide
InChIKey: ZYQXEVJIFYIBHZ-UHFFFAOYSA-N | ||||||||
| • TAK-580
IUPAC Name: 2-[(1R)-1-[(6-amino-5-chloropyrimidine-4-carbonyl)amino]ethyl]-N-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]-1,3-thiazole-5-carboxamide | CAS Registry Number: 1096708-71-2 Synonyms: SureCN4206123, BIIB024, UNII-ZN90E4027M, BIIB 024, BIIB-024, MLN2480, MLN 2480, MLN-2480, CS-0751, NCGC00346458-01, HY-15246, MLN 2480|1096708-71-2|MLN2480|MLN-2480, 4-Pyrimidinecarboxamide, 6-amino-5-chloro-N-((1R)-1-(5-(((5-chloro-4-(trifluoromethyl)-2-pyridinyl)amino)carbonyl)-2-thiazolyl)ethyl]-, 6-Amino-5-chloro-N-((1R)-1-(5-(((5-chloro-4-(trifluoromethyl)-2-pyridinyl)amino)carbonyl)-2-thiazolyl)ethyl)-4-pyrimidinecarboxamide
InChIKey: VWMJHAFYPMOMGF-ZCFIWIBFSA-N | ||||||||
| • TAK-715
IUPAC Name: N-[4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]pyridin-2-yl]benzamide | CAS Registry Number: 303162-79-0 Synonyms: TAK 715, N-(4-(2-ethyl-4-m-tolylthiazol-5-yl)pyridin-2-yl)benzamide, Kinome_2655, SureCN297487, UNII-WE92U03C5Z, cc-467, CHEMBL363648, TAK715, CTK8E7576, CHEBI:428880, BCPP000054, HMS3244J06, HMS3244J10, HMS3244J14, HMS3265K09, HMS3265K10, HMS3265L09, HMS3265L10, ABP000506, RS0059
InChIKey: HEKAIDKUDLCBRU-UHFFFAOYSA-N | ||||||||
| • TAK-733
IUPAC Name: 3-[(2R)-2,3-dihydroxypropyl]-6-fluoro-5-(2-fluoro-4-iodoanilino)-8-methylpyrido[2,3-d]pyrimidine-4,7-dione | CAS Registry Number: 1035555-63-5 Synonyms: TAK 733, TAK733, S2617_Selleck, SureCN1528606, cc-621, CHEMBL1615025, CHEBI:1138036, CS-1283, NCGC00263187-01, HY-13449, KB-137233, TAK733, 1035555-63-5, TAK-733|1035555-63-5|TAK 733, TAK733 , TAK 733 , 1035555-63-5, 3-[(2r)-2,3-Dihydroxypropyl]-6-Fluoro-5-[(2-Fluoro-4-Iodophenyl)amino]-8-Methylpyrido[2,3-D]pyrimidine-4,7(3h,8h)-Dione, 3-[(2R)-2,3-dihydroxypropyl]-6-fluoro-5-[(2-fluoro-4-iodophenyl)amino]-8-methylpyrido[2,3-d]pyrimidine-4,7-dione, IZG
InChIKey: RCLQNICOARASSR-SECBINFHSA-N | ||||||||
| • TAK-901
IUPAC Name: 5-(3-ethylsulfonylphenyl)-3,8-dimethyl-N-(1-methylpiperidin-4-yl)-9H-pyrido[2,3-b]indole-7-carboxamide | CAS Registry Number: 934541-31-8 Synonyms: TAK 901, 934541-31-8 pound not TAK901 pound not TAK 901, 5-[3-(Ethylsulfonyl)phenyl]-3,8-dimethyl-N-(1-methyl-4-piperidinyl)-9H-pyrido[2,3-b]indole-7-carboxamide, cc-11, SureCN645679, TAK901, MolPort-021-783-300, AKOS005266666, CS-0243, RL05867, NCGC00346645-01, HY-12201, KB-60668, AB1009198, A4124, X7460, TAK-901|934541-31-8|TAK 901, 5-(3-(ethylsulfonyl)phenyl)-3,8-dimethyl-N-(1-methylpiperidin-4-yl)-9H-pyrido[2,3-b]indole-7-carboxamidef, 5-[3-(ethanesulfonyl)phenyl]-3,8-dimethyl-N-(1-methylpiperidin-4-yl)-9H-pyrido[2,3-b]indole-7-carboxamide
InChIKey: WKDACQVEJIVHMZ-UHFFFAOYSA-N | ||||||||
| • Taladegib
IUPAC Name: 4-fluoro-N-methyl-N-[1-[4-(2-methylpyrazol-3-yl)phthalazin-1-yl]piperidin-4-yl]-2-(trifluoromethyl)benzamide | CAS Registry Number: 1258861-20-9 Synonyms: LY2940680, LY-2940680, UNII-QY8BWX1LJ5, SureCN2128615, cc-431, CHEMBL2142592, BCP9000881, CS-0459, RL01260, NCGC00263170-01, HY-13242, LY 2940680, X7613, LY2940680|1258861-20-9|LY-2940680, 1258861-20-9 , LY 2940680 , LY-2940680, 1KS, 4-fluoro-n-methyl-n-(1-(4-(1-methyl-1h-pyrazol-5-yl)-1-phthalazinyl)-4-piperidinyl)-2-(trifluoromethyl)benzamide, 4-Fluoro-N-Methyl-N-{1-[4-(1-Methyl-1h-Pyrazol-5-Yl)phthalazin-1-Yl]piperidin-4-Yl}-2-(Trifluoromethyl)benzamide, 4-fluoro-N-methyl-N-{1-[4-(2-methylpyrazol-3-yl)phthalazin-1-yl]piperidin-4-yl}-2-(trifluoromethyl)benzamide, Benzamide, 4-fluoro-N-methyl-N-[1-[4-(1-methyl-1H-pyrazol-5-yl)-1-phthalazinyl]-4-piperidinyl]-2-(trifluoromethyl)-
InChIKey: SZBGQDXLNMELTB-UHFFFAOYSA-N | ||||||||
| • TAME
IUPAC Name: methyl 5-(diaminomethylideneamino)-2-[(4-methylphenyl)sulfonylamino]pentanoate | CAS Registry Number: 901-47-3 Synonyms: Probes1_000325, Probes2_000471, CBDivE_015738, CHEBI:380054, MolPort-001-813-207, NSC80683, CID416661, Arginine, N(2)-p-toluenesulfonyl-, methyl ester, p-TOLUENESULFONYL-L-ARGININE METHYL ESTER HCl, 5-Guanidino-2-(toluene-4-sulfonylamino)-pentanoic acid methyl ester
InChIKey: FKMJXALNHKIDOD-UHFFFAOYSA-N | ||||||||
| • Tamoxifen
IUPAC Name: 2-[4-[(Z)-1,2-di(phenyl)but-1-enyl]phenoxy]-N,N-dimethylethanamine | CAS Registry Number: 10540-29-1 Synonyms: tamoxifen, trans-Tamoxifen, Nolvadex, Tamoxifen citrate, Crisafeno, Citofen, Istubol, Oncomox, Retaxim, Tamizam, Tamoxen, Valodex, Diemon, Tomaxithen, Zitazonium, Novaldex, Soltamox, ,citrate, Tamoxifen (Z), nchembio.76-comp1
InChIKey: NKANXQFJJICGDU-QPLCGJKRSA-N | ||||||||
| • Tandutinib
IUPAC Name: 4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin-4-yl]-N-(4-propan-2-yloxyphenyl)piperazine-1-carboxamide | CAS Registry Number: 387867-13-2 Synonyms: Tandutinib (USAN/INN), MLN-518, MLN 518, MLN-0518, NSC726292, CID3038522, CT53518, CT 53518, CT-53518, D06005, (4-(6-Methoxy-7-(3-piperidylpropoxy)quinazolin-4-yl)piperazinyl)-N-(4-(methylethoxy)phenyl)carboxamide, 1-Piperazinecarboxamide, 4-(6-methoxy-7-(3-(1-piperidinyl)propoxy)-4-quinazolinyl)-N-(4-(1-methylethoxy)phenyl)-
InChIKey: UXXQOJXBIDBUAC-UHFFFAOYSA-N | ||||||||
| • Tanespimycin
IUPAC Name: [(3R,5S,6R,7S,8E,10S,11S,12E,14E)-6-hydroxy-5,11-dimethoxy-3,7,9,15-tetramethyl-16,20,22-trioxo-21-(prop-2-enylamino)-17-azabicyclo[16.3.1]docosa-1(21),8,12,14,18-pentaen-10-yl] carbamate | CAS Registry Number: 75747-14-7 Synonyms: Tanespimycin [USAN], 17-(Allylamino)geldanamycin, 17AAG, KOS-953, NSC 330507, Cp 127374, 17-Demethoxy-17-allylamino geldanamycin, 17-(Allylamino)-17-demethoxygeldanamycin, NSC-330507, NCGC00162425-01, LS-183128, Geldanamycin, 17-(Allylamino)-17-demethoxy-, Geldanamycin, 17-demethoxy-17-(2-propenylamino)-, AAG, (4E,6Z,8S,9S,10E,12S,13R,14S,16R)-13-Hydroxy-8,14-dimethoxy-4,10,12,16- tetramethyl-3,20,22-trioxo-19-(prop-2-enylamino)-2-azabicyclo(16.3.1)docosa- 1(21),4,6,10,18-penten-9-yl carbamate
InChIKey: AYUNIORJHRXIBJ-HTLBVUBBSA-N | ||||||||
| • Taselisib
IUPAC Name: 2-methyl-2-[4-[2-(5-methyl-2-propan-2-yl-1,2,4-triazol-3-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl]pyrazol-1-yl]propanamide | CAS Registry Number: 1282512-48-4 Synonyms: GDC-0032, CHEMBL2387080, Taselisib [INN], SureCN1485247, UNII-L08J2O299M, KB-145919, S7103,GDC0032,RG7604,1282512-48-4
InChIKey: BEUQXVWXFDOSAQ-UHFFFAOYSA-N | ||||||||
| • TCID
IUPAC Name: 4,5,6,7-tetrachloroindene-1,3-dione | CAS Registry Number: 30675-13-9 Synonyms: 4,5,6,7-Tetrachloroindan-1,3-dione, 4,5,6,7-Tetrachloro-1H-indene-1,3(2H)-dione, UCH-L3 Inhibitor, 4,5,6,7-Tetrachloroindane-1,3-dione, Ubiquitin Thiolesterase L3 Inhibitor, SBB054653, AG-F-01198, Ubiquitin C-Terminal Esterase L3 Inhibitor, Ubiquitin C-Terminal Hydrolase L3 Inhibitor, 4,5,6,7-tetrachloro-2H-indene-1,3-dione, Maybridge1_006552, AC1MBP0F, SureCN5819833, CHEMBL1241028, CTK4G5564, HMS560B18, MolPort-000-145-737, ANW-73173, CCG-51207, RW3397
InChIKey: IDLAOWFFKWRNHB-UHFFFAOYSA-N | ||||||||
| • TCS 359
IUPAC Name: 2-[(3,4-dimethoxybenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide | CAS Registry Number: 301305-73-7 Synonyms: Flt-3 inhibitor, 2-(3,4-Dimethoxy-benzoylamino)-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid amide, 2-(3,4-dimethoxybenzamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxamide, 2-[(3,4-dimethoxybenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide, ZINC00725713, ACMC-20ekhy, AC1LKSB9, SureCN8290405, Oprea1_063849, Oprea1_870745, D5943_SIGMA, CHEMBL210833, QCR-73, STOCK2S-64515, CTK8E8753, TCS-359, CHEBI:449543, MolPort-000-224-308, HMS3229E07, HMS3269D21
InChIKey: FSPQCTGGIANIJZ-UHFFFAOYSA-N | ||||||||
| • TCS7010
IUPAC Name: N-(2-chlorophenyl)-4-[[2-[4-[2-(4-ethylpiperazin-1-yl)-2-oxoethyl]anilino]-5-fluoropyrimidin-4-yl]amino]benzamide | CAS Registry Number: 1158838-45-9 Synonyms: Aurora A Inhibitor I, N-(2-Chlorophenyl)-4-((2-((4-(2-(4-ethylpiperazin-1-yl)-2-oxoethyl)phenyl)amino)-5-fluoropyrimidin-4-yl)amino)benzamide, N-(2-chlorophenyl)-4-{[2-({4-[2-(4-ethylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}benzamide, S1451_Selleck, 2,4-Bisanilinopyrimidine, 10, CHEMBL502124, CTK4A9531, BCPP000376, HMS3265K21, HMS3265K22, HMS3265L21, HMS3265L22, ANW-58929, AKOS015995069, AG-L-19476, BCP9000341, CS-0011, NCGC00346525-01, AK-56791, Aurora A inhibitor I|1158838-45-9
InChIKey: AKSIZPIFQAYJGF-UHFFFAOYSA-N | ||||||||
| • Telaprevir
IUPAC Name: (1S,3aR,6aS)-2-[(2S)-2-[[(2S)-2-cyclohexyl-2-(pyrazine-2-carbonylamino)acetyl]amino]-3,3-dimethylbutanoyl]-N-[1-(cyclopropylamino)-1,2-dioxohexan-3-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole-1-carboxamide | CAS Registry Number: 402957-28-2 Synonyms: VX 950, VX-950, LY 570310, 569364-34-7, Cyclopenta(c)pyrrole-1-carboxamide, (2S)-2-cyclohexyl-N-(pyrazinylcarbonyl)glycyl-3-methyl-L-valyl-N-((1S)-1-((cyclopropylamino)oxoacetyl)butyl)octahydro-, (1S,3aR,6aS)-
InChIKey: BBAWEDCPNXPBQM-IGSHNTALSA-N | ||||||||
| • Telatinib
IUPAC Name: 4-[[4-(4-chloroanilino)furo[2,3-d]pyridazin-7-yl]oxymethyl]-N-methylpyridine-2-carboxamide | CAS Registry Number: 332012-40-5 Synonyms: UNII-18P7197Q7J, Bay 57-9352, CID9808844, CID 9808844, 2-Pyridinecarboxamide, 4-(((4-((4-chlorophenyl)amino)furo(2,3-d)pyridazin-7-yl)oxy)methyl)-N-methyl-
InChIKey: QFCXANHHBCGMAS-UHFFFAOYSA-N | ||||||||
| • Temozolomide
IUPAC Name: 3-methyl-4-oxoimidazo[5,1-d][1,2,3,5]tetrazine-8-carboxamide | CAS Registry Number: 85622-93-1 Synonyms: temozolomide, Methazolastone, Temodal, Temodar, Temozolamide, Temozolomidum [Latin], Temozolodida [Spanish], Temodal (TN), Temozolomide [BAN:INN], Temozolomide [INN:BAN], Essex brand of temozolomide, CCRG 81045, CCRG-81045, Sch 52365, MLS000759447, MLS001424028, Schering brand of temozolomide, C6H6N6O2, CCRIS 8996, Temozolomide (JAN/USAN/INN)
InChIKey: BPEGJWRSRHCHSN-UHFFFAOYSA-N | ||||||||
| • Temsirolimus
Synonyms: Cci 779, WAY-CCI 779, CCI-779, Rapamycin, 42-(3-hydroxy-2-(hydroxymethyl)-2-methylpropanoate), 343261-52-9
InChIKey: CBPNZQVSJQDFBE-WEDGMEQVSA-N | ||||||||
| • Tenovin-1
IUPAC Name: N-[(4-acetamidophenyl)carbamothioyl]-4-tert-butylbenzamide | CAS Registry Number: 380315-80-0 Synonyms: NCGC00181351-01, ZINC00674444, AC1LK7DX, DSSTox_CID_26920, DSSTox_RID_82016, DSSTox_GSID_46920, Oprea1_317255, cc-649, ARONIS003419, CHEMBL1436543, CTK8E7058, QCR-245, MolPort-001-530-678, Tox21_112809, STK077754, AKOS000492892, CCG-208685, MCULE-2127700307, RL03447, CAS-380315-80-0
InChIKey: WOWJIWFCOPZFGV-UHFFFAOYSA-N | ||||||||
| • Tepotinib
IUPAC Name: 3-[1-[[3-[5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl]phenyl]methyl]-6-oxopyridazin-3-yl]benzonitrile | CAS Registry Number: 1100598-32-0 Synonyms: EMD 1214063, EMD-1214063, SureCN1296895, UNII-1IJV77EI07, CS-0647, EMD1214063, NCGC00345793-01, HY-14721, Y0358, S7067,EMD1214063,1100598-32-0, EMD-1214063|1100598-32-0|EMD1214063, Benzonitrile, 3-(1,6-dihydro-1-((3-(5-((1-methyl-4-piperidinyl)methoxy)-2-pyrimidinyl)phenyl)methyl)-6-oxo-3-pyridazinyl)-, Benzonitrile, 3-[1,6-Dihydro-1-[[3-[5-[(1-Methyl-4-Piperidinyl)Methoxy]-2-PyriMidinyl]Phenyl]Methyl]-6-Oxo-3-Pyridazinyl]
InChIKey: AHYMHWXQRWRBKT-UHFFFAOYSA-N | ||||||||
| • tert-Butyl (4-acetylpyridin-3-yl)carbamate
IUPAC Name: tert-butyl N-(4-acetylpyridin-3-yl)carbamate | CAS Registry Number: 1260892-75-8 Synonyms: CTK8C2340, ANW-68224, QC-227, AKOS016007008, tert-butyl 4-acetylpyridin-3-ylcarbamate, AK-80588, KB-260096
InChIKey: GFXIZWAPDSDUNQ-UHFFFAOYSA-N | ||||||||
| • tert-butyl 3-mercaptopyridin-4-ylcarbamate
IUPAC Name: tert-butyl N-(3-sulfanylpyridin-4-yl)carbamate | CAS Registry Number: 365996-04-9 Synonyms: tert-Butyl (3-mercaptopyridin-4-yl)carbamate, SureCN741240, CTK1B6223, ANW-62124, AKOS016004811, AK102447, KB-260077, Carbamic acid, (3-mercapto-4-pyridinyl)-, 1,1-dimethylethyl ester
InChIKey: MKRKOWOVJQNWSY-UHFFFAOYSA-N | ||||||||
| • Tert-butyl 4-((4-(4-bromo-2-fluorophenylamino)-6-methoxyquinazolin-7-yloxy)methyl)piperidine-1-carboxylate
IUPAC Name: tert-butyl 4-[[4-(4-bromo-2-fluoroanilino)-6-methoxyquinazolin-7-yl]oxymethyl]piperidine-1-carboxylate | CAS Registry Number: 338992-20-4 Synonyms: AGN-PC-0CTN16, SureCN1614506, AKOS016011495, QC-1063, AK120806, KB-66569, 1-Piperidinecarboxylic acid,4-[[[4-[(4-bromo-2-fluorophenyl)amino]-6-methoxy-7-quinazolinyl]oxy]methyl]-,1,1-dimethylethyl ester, tert-Butyl 4-(((4-((4-bromo-2-fluorophenyl)amino)-6-methoxyquinazolin-7-yl)oxy)methyl)piperidine-1-carboxylate, tert-butyl 4-((4-(4-bromo-2-fluorophenylamino)-6-methoxyquinazolin-7-yloxy)methyl)piperidine-1-carboxylate, tert-butyl 4-[[4-(4-bromo-2-fluoroanilino)-6-(trideuteriomethoxy)quinazolin-7-yl]oxymethyl]piperidine-1-carboxylate
InChIKey: DJQLEEANCWENKG-UHFFFAOYSA-N | ||||||||
| • tert-butyl 4-(4-iodo-1H-pyrazol-1-yl)piperidine-1-carboxylate
IUPAC Name: tert-butyl 4-(4-iodopyrazol-1-yl)piperidine-1-carboxylate
InChIKey: IONGFFYQZADMPH-UHFFFAOYSA-N | ||||||||
| • tert-butyl 4-mercaptopyridin-3-ylcarbamate
IUPAC Name: tert-butyl N-(4-sulfanylidene-1H-pyridin-3-yl)carbamate | CAS Registry Number: 139460-10-9 Synonyms: tert-Butyl (4-mercaptopyridin-3-yl)carbamate, SureCN743727, CTK8C2322, ANW-68202, AKOS016007166, AK-80618, KB-260114
InChIKey: HESMDBDUEDHPRG-UHFFFAOYSA-N | ||||||||
| • tert-butyl benzyl(2-oxoethyl)carbamate
IUPAC Name: tert-butyl N-benzyl-N-(2-oxoethyl)carbamate | CAS Registry Number: 136159-63-2 Synonyms: Carbamic acid, (2-oxoethyl)(phenylmethyl)-, 1,1-dimethylethyl ester, ACMC-20mw1v, CTK0B9555
InChIKey: RXJOEKWQWAKFSV-UHFFFAOYSA-N |