Profile: Jinan Trio PharmaTech Co., Ltd. specializes in APIs & intermediates, heterocyclic compounds, and anti-tumor drugs. Our products include crizotinib, vemurafenib, afatinib, vandetanib, regorafenib, brivanib alaninate, pyridazine, imidazole, pyrazole, and oxazole. We are specialized in providing over 1000 products including molecular targeted anticancer drugs, cell signaling pathway inhibitors, pharmaceutical intermediates, and heterocyclic compounds, and quality services including custom synthesis, transfer of new drug patent and technology, technical cooperation, and process optimization.
| • Oxaliplatin
IUPAC Name: (1R,2R)-cyclohexane-1,2-diamine; oxalate; platinum(2+) | CAS Registry Number: 61825-94-3 Synonyms: oxaliplatin, oxalate, Oxalatoplatin, Oxalatoplatinum, Eloxatin, Eloxatin (TN), platinum(+2) cation, Oxaliplatinum [Latin], Oxaloplatine [French], Oxaliplatino [Spanish], Oxaloplatino [Spanish], Oxaliplatin (JAN/USAN/INN), Oxaliplatin [USAN:INN:BAN], (1R,2R)-cyclohexane-1,2-diamine, DB00526, D01790
InChIKey: ZROHGHOFXNOHSO-BNTLRKBRSA-L | ||||||||
| • OXAZOLE, 2-CHLORO-
IUPAC Name: 2-chloro-1,3-oxazole | CAS Registry Number: 95458-77-8 Synonyms: Oxazole, 2-chloro-, 2-Chlorooxazole, 2-CHLORO-OXAZOLE, SureCN317377, AGN-PC-00ME2Y, CTK3I6009, AKOS006288793, AG-H-92848, FT-0645180
InChIKey: SSXYKBHZZRYLLY-UHFFFAOYSA-N | ||||||||
| • OXAZOLE,5-(CHLOROMETHYL)-
IUPAC Name: 5-(chloromethyl)-1,3-oxazole | CAS Registry Number: 172649-57-9 Synonyms: 5-(Chloromethyl)oxazole, OXAZOLE, 5-(CHLOROMETHYL)-, AGN-PC-00ORQJ, SureCN7442697, CTK8C2828, ANW-69074, RB3366, AKOS006286857, AB42450, 5-(CHLOROMETHYL)-1,3-OXAZOLE, AK-48287, KB-243840, FT-0084326, FT-0660245
InChIKey: UJLHZLUVPVJDQI-UHFFFAOYSA-N | ||||||||
| • Oxazole-2-Carbaldehyde
IUPAC Name: 1,3-oxazole-2-carbaldehyde | CAS Registry Number: 65373-52-6 Synonyms: Oxazole-2-carbaldehyde, 2-Oxazolecarboxaldehyde, 1,3-oxazole-2-carbaldehyde, SBB052295, zlchem 772, PubChem17600, AGN-PC-002JTD, OXAZOLE-2-CARBOXALDEHYDE, 1,3-Oxazole-2-carboxaldehyde;, CTK2F2741, ZLD0231, MolPort-004-747-047, ACT06108, WTI-10543, ZINC02530178, 1,3-OXAZOLE-2-CARBOXALDEHYDE, AKOS006342976, AB14413, AG-B-76909, AG-G-46050
InChIKey: TYHOSUCCUICRLM-UHFFFAOYSA-N | ||||||||
| • OXAZOLO[4,5-C]PYRIDIN-2-AMINE
IUPAC Name: [1,3]oxazolo[4,5-c]pyridin-2-amine | CAS Registry Number: 114498-55-4 Synonyms: Oxazolo[4,5-c]pyridin-2-amine, ACMC-20adcd, AGN-PC-000U7Q, CTK0H3203, MolPort-004-757-684, ANW-68219, AKOS016007039, AG-D-34817, QC-4947, Oxazolo[4,5-c]pyridin-2-amine (9CI), AK-80598, BD236979, KB-79732
InChIKey: FJHYVYMTPVSYDO-UHFFFAOYSA-N | ||||||||
| • Oxazolo[4,5-c]pyridine, 7-bromo-2-ethyl-
IUPAC Name: 7-bromo-2-ethyl-[1,3]oxazolo[4,5-c]pyridine | CAS Registry Number: 118685-69-1 Synonyms: 7-Bromo-2-ethyloxazolo[4,5-c]pyridine, CTK8C2335, ANW-68217, AKOS016007061, AK-80600, KB-79734, Oxazolo[4,5-c]pyridine,7-bromo-2-ethyl-
InChIKey: AMHXDXSOKYQXFX-UHFFFAOYSA-N | ||||||||
| • Oxazolo[4,5-c]pyridine, 7-bromo-2-methyl-
IUPAC Name: 7-bromo-2-methyl-[1,3]oxazolo[4,5-c]pyridine | CAS Registry Number: 116081-17-5 Synonyms: 7-Bromo-2-methyloxazolo[4,5-c]pyridine, CTK8C2336, ANW-68218, AKOS016007060, AK-80599, BD236980, KB-79735, Oxazolo[4,5-c]pyridine,7-bromo-2-methyl-
InChIKey: LACXEYMKTOJZHX-UHFFFAOYSA-N | ||||||||
| • P 22077
IUPAC Name: 1-[5-(2,4-difluorophenyl)sulfanyl-4-nitrothiophen-2-yl]ethanone | CAS Registry Number: 1247819-59-5 Synonyms: CHEMBL2159498, SureCN2680945, QC-8199, 1-(5-(2,4-difluorophenylthio)-4-nitrothiophen-2-yl)ethanone
InChIKey: RMAMGGNACJHXHO-UHFFFAOYSA-N | ||||||||
| • P-Methoxyacetanilide
IUPAC Name: N-(4-methoxyphenyl)acetamide | CAS Registry Number: 51-66-1 Synonyms: p-Acetanisidide, Metacetin, Methacetin, p-Acetanisidine, Aceto-p-anisidide, Acetyl-p-anisidine, p-Methoxyacetanilide, N-Acetyl-p-anisidine, 4'-Methoxyacetanilide, N-(4-Methoxyphenyl)acetamide, N-Acetyl-p-methoxyaniline, Acetanilide, 4'-methoxy-, 4-METHOXYACETANILIDE, Acetamide, N-(4-methoxyphenyl)-, WLN: 1VMR DO1, ARONIS003521, NSC 4687, EINECS 200-114-2, NSC4687, BRN 0387887
InChIKey: XVAIDCNLVLTVFM-UHFFFAOYSA-N | ||||||||
| • P005091
IUPAC Name: 1-[5-(2,3-dichlorophenyl)sulfanyl-4-nitrothiophen-2-yl]ethanone | CAS Registry Number: 882257-11-6 Synonyms: CHEMBL2159495, ZINC00125366, SureCN2681288, AC1ME173, MolPort-002-906-122, KM03205, QC-8200, 1-(5-(2,3-dichlorophenylthio)-4-nitrothiophen-2-yl)ethanone, 1-[5-(2,3-dichlorophenyl)sulfanyl-4-nitrothiophen-2-yl]ethanone, 1-{5-[(2,3-dichlorophenyl)thio]-4-nitro-2-thienyl}ethan-1-one
InChIKey: LKZLGMAAKNEGCH-UHFFFAOYSA-N | ||||||||
| • PAC-1
IUPAC Name: 2-(4-benzylpiperazin-1-yl)-N'-[(Z)-(6-oxo-5-prop-2-enylcyclohexa-2,4-dien-1-ylidene)methyl]acetohydrazide | CAS Registry Number: 315183-21-2 Synonyms: Procaspase-3 Activator, PAC-1, PAC 1 pound not Procaspase activating compound 1, 315183-21-2, (4-Benzylpiperazino)acetic acid-(3-allyl-2-hydroxybenzylidene)hydrazide, PAC 1, Procaspase-3 Activator, PAC-1 pound notPAC1, AC1OA9GH, cc-276, CHEMBL591429, Procaspase activating compound 1, STOCK3S-22963, MolPort-002-580-634, NSC743444, BCP9001044, NSC-743444, NCGC00167785-02, BCP0726000262, X5905, 2-(4-benzylpiperazin-1-yl)-N'-[(1E)-[2-hydroxy-3-(prop-2-en-1-yl)phenyl]methylidene]acetohydrazide, 2-(4-benzylpiperazin-1-yl)-N'-[(Z)-(6-oxo-5-prop-2-enylcyclohexa-2,4-dien-1-ylidene)methyl]acetohydrazide
InChIKey: XSGXRYNZNGUGEJ-PGMHBOJBSA-N | ||||||||
| • Paclitaxel
Synonyms: paclitaxel, Yewtaxan, TAXOL, Plaxicel, Paxceed, Taxol A, Abraxane, Ebetaxel, Capxol, Paxene, Onxol, TaxAlbin, LipoPac, Genetaxyl, Nanotaxel, Paclical, Pacligel, Anzatax, Genaxol, Genexol
InChIKey: RCINICONZNJXQF-MZXODVADSA-N | ||||||||
| • Palbociclib Isethionate
IUPAC Name: 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7-one;2-hydroxyethanesulfonic acid | CAS Registry Number: 827022-33-3 Synonyms: AGN-PC-009X4E, Palbociclib Isethionate [USAN}, CHEMBL2364621, PD 0332991 (Palbociclib) Isethionate, PF-0008066573, PD 0332991-0054, PD-03329910054, PF-00080665-73, S1579,827022-33-3, 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7-one;2-hydroxyethanesulfonic acid
InChIKey: LYYVFHRFIJKPOV-UHFFFAOYSA-N | ||||||||
| • Palbociclib monohydrochloride
IUPAC Name: 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7-one;hydrochloride | CAS Registry Number: 827022-32-2 Synonyms: PD 0332991 HCl, Palbociclib HCl, Palbociclib hydrochloride, AGN-PC-008ZCE, SureCN2076416, PD0332991 hydrochloride, cc-424, PD 0332991 hydrochloride, HY-50767A, CS-1327, RL05143, X7620, Palbociclib hydrochloride|827022-32-2|PD0332991 hydrochloride|PD 0332991 hydrochloride, 6-acetyl-8-cyclopentyl-5-methyl-2-((5-(1-piperazinyl)-2-pyridinyl)amino)pyrido(2,3-d)pyrimidin-7(8h)-one hydrochloride, 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7-one;hydrochloride, 6-acetyl-8-cyclopentyl-5-methyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}pyrido[2,3-d]pyrimidin-7-one hydrochloride
InChIKey: STEQOHNDWONVIF-UHFFFAOYSA-N | ||||||||
| • Palomid 529
IUPAC Name: 8-(1-hydroxyethyl)-2-methoxy-3-[(4-methoxyphenyl)methoxy]benzo[c]chromen-6-one | CAS Registry Number: 914913-88-5 Synonyms: Palomid529, Palomid-529, P-529, P529, Palomid 529, P529, P529, 914913-88-5, 8-(1-hydroxyethyl)-2-methoxy-3-[(4-methoxyphenyl)methoxy]benzo[c]chromen-6-one, S2238_Selleck, AGN-PC-00JIQP, Palomid 529,P529, SureCN290034, SureCN7860257, UNII-XV9409EWG4, cc-513, Palomid 529 - P529, QCR-215, BCPP000131, BCP9001049, CS-0258, RL05762
InChIKey: YEAHTLOYHVWAKW-UHFFFAOYSA-N | ||||||||
| • Pazopanib
IUPAC Name: 5-[[4-[(2,3-dimethylindazol-6-yl)-methylamino]pyrimidin-2-yl]amino]-2-methylbenzenesulfonamide | CAS Registry Number: 444731-52-6 Synonyms: GW786034, UNII-7RN5DR86CK, CHEBI:71219, NCGC00188865-01, GW 78603, Pazopanib [INN], DSSTox_CID_28659, DSSTox_RID_82929, DSSTox_GSID_48733, 790713-33-6, Kinome_3790, CHEMBL477772, 5-(4-((2,3-dimethyl-2H-indazol-6-yl)(methyl)amino)pyrimidin-2-ylamino)-2-methylbenzenesulfonamide, 5-[[4-[(2,3-Dimethyl-2H-indazol-6-yl)(methyl)amino]pyrimidin-2-yl]amino]-2-methylbenzenesulfonamide, Benzenesulfonamide, 5-[[4-[(2,3-dimethyl-2H-indazol-6-yl)methylamino]-2-pyrimidinyl]amino]-2-methyl-, CAS-444731-52-6, AKOS005145819, 5-[[4-[(2,3-dimethylindazol-6-yl)-methyl-amino]pyrimidin-2-yl]amino]-2-methyl-benzenesulfonamide, ST51053493, pazopanibum
InChIKey: CUIHSIWYWATEQL-UHFFFAOYSA-N | ||||||||
| • PD153035
IUPAC Name: N-(3-bromophenyl)-6,7-dimethoxyquinazolin-4-amine | CAS Registry Number: 153436-54-5 Synonyms: N-(3-bromophenyl)-6,7-dimethoxyquinazolin-4-amine, Compound 32, PD-153035, PD 153035 HYDROCHLORIDE, pd 153035, InSolution™ PD 153035, AG 1517, SU 5271, 4-[(3-Bromophenyl)amino]-6,7-dimethoxyquinazoline, 4-(3-BROMOANILINO)-6,7-DIMETHOXYQUINAZOLINE, 4-QUINAZOLINAMINE, N-(3-BROMOPHENYL)-6,7-DIMETHOXY-, PubChem22449, Tocris-1037, SureCN9423, AC1L1IRP, UNII-TC62B68RSL, AC1Q26CE, CHEMBL29197, WHI-P 79, LSPANGZZENHZNJ-UHFFFAOYSA-
InChIKey: LSPANGZZENHZNJ-UHFFFAOYSA-N | ||||||||
| • PD168393
IUPAC Name: N-[4-(3-bromoanilino)quinazolin-6-yl]prop-2-enamide | CAS Registry Number: 194423-15-9 Synonyms: pd 168393, n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}prop-2-enamide, PD-168393, 4-[(3-Bromophenyl)amino]-6-acrylamidoquinazoline, nchembio866-comp2, AC1L1IRY, AC1Q26CC, SureCN2680536, 4-anilinoquinazoline deriv. 2, CHEMBL285063, CTK0E1086, AR-1K4749, DNC004255, HSCI1_000120, IN1166, ZINC01488208, AG-L-66492, DB07662, N-(4-(3-Bromophenylamino)quinazolin-6-yl)acrylamide, N-[4-(3-bromoanilino)quinazolin-6-yl]prop-2-enamide
InChIKey: HTUBKQUPEREOGA-UHFFFAOYSA-N | ||||||||
| • PD173074
IUPAC Name: 1-tert-butyl-3-[2-[4-(diethylamino)butylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea | CAS Registry Number: 219580-11-7 Synonyms: PD 173074, PD-173074, CHEBI:63448, 1-tert-butyl-3-[2-{[4-(diethylamino)butyl]amino}-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea, FGF/VEGF Receptor Tyrosine Kinase Inhibitor, PD173074, PD173074, 219580-11-7, 2fgi, 1-(tert-Butyl)-3-(2-((4-(diethylamino)butyl)amino)-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl)urea, 1-t-Butyl-3-(6-(3,5-dimethoxyphenyl)-2-(4-diethylaminobutylamino)-pyrido[2,3-d]pyrimidin-7-yl)urea, 1-tert-butyl-3-(2-(4-(diethylamino)butylamino)-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl)urea, 1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-urea, PD1, 1-tert-butyl-3-[2-[4-(diethylamino)butylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea, S1264_Selleck, PubChem22593, SureCN177946, AC1L1BE8, UNII-A4TLL8634Y, JSPY-st000263, cc-523
InChIKey: DXCUKNQANPLTEJ-UHFFFAOYSA-N | ||||||||
| • PD173955
IUPAC Name: 6-(2,6-dichlorophenyl)-8-methyl-2-(3-methylsulfanylanilino)pyrido[2,3-d]pyrimidin-7-one | CAS Registry Number: 260415-63-2 Synonyms: CHEBI:49791, 6-(2,6-DICHLORO-PHENYL)-8-METHYL-2-(3-METHYLSULFANYL-PHENYLAMINO)-8H-PYRIDO[2,3-D]PYRIMIDIN-7-ONE, 6-(2,6-dichlorophenyl)-8-methyl-2-{[3-(methylthio)phenyl]amino}pyrido[2,3-d]pyrimidin-7(8H)-one, PD-173955, Pd 173955, PubChem22476, AC1L9KFO, SureCN256712, CHEMBL386051, MolPort-006-168-472, BCPP000124, AMX10196, DNC006871, RS0021, BCP9001059, DB02567, NCGC00345829-01, PD-17395, PD-0173955, Y0273
InChIKey: VAARYSWULJUGST-UHFFFAOYSA-N | ||||||||
| • PD318088
IUPAC Name: 5-bromo-N-(2,3-dihydroxypropoxy)-3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzamide | CAS Registry Number: 391210-00-7 Synonyms: PD 318088, PD-318088, S1568_Selleck, AGN-PC-01LTJY, C16H13BrF3IN2O4, cc-457, MolPort-006-168-845, BCPP000120, BCP9001066, CS-0222, RL03489, NCGC00346552-01, HY-12062, PD318088-Supplied by Selleck Chemicals, X7397, PD 318088, 391210-00-7, PD318088|391210-00-7|PD-318088, 5-bromo-N-(2,3-dihydroxypropoxy)-3,4-difluoro-2-(2-fluoro-4-iodophenylamino)benzamide, 5-BROMO-N-(2,3-DIHYDROXYPROPOXY)-3,4-DIFLUORO-2-[(2-FLUORO-4-IODOPHENYL)AMINO]-, 5-bromo-N-[(2R)-2,3-dihydroxypropoxy]-3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzamide
InChIKey: XXSSGBYXSKOLAM-UHFFFAOYSA-N | ||||||||
| • PD98059
IUPAC Name: 2-(2-amino-3-methoxyphenyl)chromen-4-one | CAS Registry Number: 167869-21-8 Synonyms: Tocris-1213, Lopac-P-215, BiomolKI_000001, BiomolKI2_000011, P215_SIGMA, Lopac0_001028, BSPBio_000996, KBioGR_000336, KBioSS_000336, PD 98059, BCBcMAP01_000049, KBio2_000336, KBio2_002904, KBio2_005472, KBio3_000671, KBio3_000672, BIP0711, CID4713, PD 98,059, AIDS220091
InChIKey: QFWCYNPOPKQOKV-UHFFFAOYSA-N | ||||||||
| • Pelitinib
IUPAC Name: (E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)but-2-enamide | CAS Registry Number: 257933-82-7 Synonyms: EKB-569, Pelitinib (USAN/INN), WAY-EKB 569, WAY-EKB-569, CHEBI:38927, EKB 569, NSC729742, CID6445562, WAY-172569, D05399, (2E)-N-(4-((3-chloro-4-fluorophenyl)amino)-3-cyano-7-ethoxy-6-quinolinyl)-4-(dimethylamino)-2-butenamide, (2E)-N-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamide, (E)-N-[4-(3-Chloro-4-fluoroanilino)-cyano-7-ethoxyquinolin-6-yl]-4-(dimethlyamino)but-2-enamide,, 2-Butenamide, N-(4-((3-chloro-4-fluorophenyl)amino)-3-cyano-7-ethoxy-6-quinolinyl)-4-(dimethylamino)-, (2E)-, 2-Butenamide, N-[4-(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl-4-(dimethylamino)-, (E)-,, 4-Dimethylaminobut-2-enoic Acid, [4-(3-Chloro-4-fluoro phenylamino)-3-cyano-7-ethoxyquinoline-6-yl]amide
InChIKey: WVUNYSQLFKLYNI-AATRIKPKSA-N | ||||||||
| • Pemetrexed
IUPAC Name: (2R)-2-[[4-[2-(2-amino-4-oxo-1,7-dihydropyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]amino]pentanedioic acid | CAS Registry Number: 137281-23-3 Synonyms: Alimta, Pemetrexed disodium, Pemetrexed [INN:BAN], UNII-04Q9AIZ7NO, HSDB 7316, C20H21N5O6, CID60843, LY231514, DB00642, LY 231514, LY 231,514, LS-172988, LY-231514, LY-231,514, L-Glutamic acid, N-(4-(2-(2-amino-4,7-dihydro-4-oxo-1H-pyrrolo(2,3-d)pyrimidin-5-yl)ethyl)benzoyl)-, N-(4-(2-(2-Amino-3,4-dihydro-4-oxo-7H-pyrrolo(2,3-d)pyrimdin-5-yl)ethyl)benzoyl)glutamic acid, (2R)-2-[[4-[2-(2-amino-4-oxo-1,7-dihydropyrrolo[4,5-e]pyrimidin-5-yl)ethyl]benzoyl]amino]pentanedioic acid, MTA
InChIKey: WBXPDJSOTKVWSJ-CYBMUJFWSA-N | ||||||||
| • Pendimethalin
IUPAC Name: 3,4-dimethyl-2,6-dinitro-N-pentan-3-ylaniline | CAS Registry Number: 40487-42-1 Synonyms: Penoxaline, PENDIMETHALIN, Prowl, Pendimethaline, Tendimethalin, Phenoxalin, Herbadox, Penoxalin, Accotab, Penoxyn, Sipaxol, Stomp, Wayup, Wax Up, Way Up, Go-Go-San, SWGC, Stomp 330D, Stomp 330E, Caswell No. 454BB
InChIKey: CHIFOSRWCNZCFN-UHFFFAOYSA-N | ||||||||
| • Perifosine
IUPAC Name: (1,1-dimethylpiperidin-1-ium-4-yl) octadecyl phosphate | CAS Registry Number: 157716-52-4 Synonyms: Perifosine [INN], NKA17, KRX-0401, CID148177, NSC639966, NSC 639966, NSC-639966, D 21266, D-21266, octadecyl-(1,1-dimethyl-4-piperidylio)phosphate, C105905, 4-((Hydroxy(octadecyloxy)phosphinyl)oxy)-1,1-dimethylpiperidinium inner salt, Piperidinium, 4-((hydroxy(octadecyloxy)phosphinyl)oxy)-1,1-dimethyl-, inner salt, Piperidinium, 4-[[hydroxy(octadecyloxy)phosphinyl]oxy]-1,1-dimethyl-, inner salt
InChIKey: SZFPYBIJACMNJV-UHFFFAOYSA-N | ||||||||
| • Pevonedistat
IUPAC Name: [(2S,4R)-4-[4-[[(1S)-2,3-dihydro-1H-inden-1-yl]amino]pyrrolo[2,3-d]pyrimidin-7-yl]-2-hydroxycyclopentyl]methyl sulfamate | CAS Registry Number: 905579-51-3 Synonyms: MLN4924, KB-78921
InChIKey: MPUQHZXIXSTTDU-LPISGYMPSA-N | ||||||||
| • PF 477736
Synonyms: PF-477736, PF-00477736, UNII-XO23PGZ0SM, PF 00477736, SureCN13599879, cc-269, (2R)-2-Amino-2-cyclohexyl-N-[2-(1-methyl-1H-pyrazol-4-yl)-6-oxo-5,6-dihydro-1H-[1,2]diazepino[4,5,6-cd]indol-8-yl]-acetamide, DCL001077, NCGC00263132-01, NCGC00263132-02, HY-10032, PF477736, PF0044736, PF-3644022, Y0431, PF-477736,PF-0044736, PF 477736|952021-60-2|PF0044736|PF477736|PF-477736, (|AR)-|A-Amino-N-[5,6-dihydro-2-(1-methyl-1H-pyrazol-4-yl)-6-oxo-1H-pyrrolo[4,3,2-ef][2,3]benzodiazepin-8-yl]cyclohexaneacetamide, (10R)-9,10,11,12-Tetrahydro-10-methyl-3-(6-methyl-3-pyridinyl)-8H-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one, 1071848-28-6
InChIKey: YFNWWNRZJGMDBR-LJQANCHMSA-N | ||||||||
| • PF-04217903
IUPAC Name: 2-[4-[3-(quinolin-6-ylmethyl)triazolo[4,5-b]pyrazin-5-yl]pyrazol-1-yl]ethanol | CAS Registry Number: 956905-27-4 Synonyms: PF 04217903, CHEMBL2001019, PF04217903, aka PF-04217903, PF04217903, 956905-27-4, 1159490-85-3, PF-04217903, PF04217903, 3zxz, 2-(4-(1-(Quinolin-6-ylmethyl)-1H-(1,2,3)triazolo(4,5-b)pyrazin-6-yl)-1H-pyrazol-1-yl)ethanol, 2-(4-(1-(quinolin-6-ylmethyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)-1H-pyrazol-1-yl)ethanol, S1094_Selleck, Kinome_3829, PubChem19150, PubChem22335, UNII-CYJ9ATV1IJ, SureCN93550, AGN-PC-01LTWA, cc-599, QCR-189, MolPort-016-633-176
InChIKey: PDMUGYOXRHVNMO-UHFFFAOYSA-N | ||||||||
| • PF-04691502
IUPAC Name: 2-amino-8-[4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7-one | CAS Registry Number: 1013101-36-4 Synonyms: CHEMBL1234354, PF04691502, PF 04691502, 1013101-36-4 pound not PF04691502 pound not PF 04691502, 2-amino-8-((1r,4r)-4-(2-hydroxyethoxy)cyclohexyl)-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8H)-one, PubChem24348, SureCN1381425, SureCN1381431, SureCN1984896, SureCN10092210, SureCN13976989, cc-350, QCR-137, AKOS005266645, CS-0919, NCGC00346659-01, HY-15177, BCP0726000275, PF-4691502, X7464
InChIKey: XDLYKKIQACFMJG-UHFFFAOYSA-N | ||||||||
| • PF-4708671
IUPAC Name: 2-[[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl]-6-(trifluoromethyl)-1H-benzimidazole | CAS Registry Number: 1255517-76-0 Synonyms: 2-((4-(5-Ethylpyrimidin-4-yl)piperazin-1-yl)methyl)-5-(trifluoromethyl)-1H-benzo[d]imidazole, 2-{[4-(5-Ethylpyrimidin-4-Yl)piperazin-1-Yl]methyl}-5-(Trifluoromethyl)-1h-Benzimidazole, 5FI, CHEMBL2134202, HMS3263P20, CCG-222583, QC-8396, NCGC00263134-01, FT-0673656, PF 4708671, S2163,PF4708671,PF-04708671,1255517-76-0, 2-[[4-(5-ethyl-4-pyrimidinyl)-1-piperazinyl]methyl]-6-(trifluoromethyl)-1H-benzimidazole
InChIKey: FBLPQCAQRNSVHB-UHFFFAOYSA-N | ||||||||
| • PF-5274857
IUPAC Name: 1-[4-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]piperazin-1-yl]-3-methylsulfonylpropan-1-one | CAS Registry Number: 1373615-35-0 Synonyms: 1-(4-(5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl)piperazin-1-yl)-3-(methylsulfonyl)propan-1-one, SureCN2715391, cc-682, CS-1206, QC-1145, RL01646, NCGC00346696-01, HY-13459, KB-145934, PF5274857, Y0361, PF-5274857|1373615-35-0|PF5274857
InChIKey: BBVNTTZIOTWDSV-UHFFFAOYSA-N | ||||||||
| • PF-562271
IUPAC Name: N-methyl-N-[3-[[[2-[(2-oxo-1,3-dihydroindol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | CAS Registry Number: 717907-75-0 Synonyms: PF 562271, PF-00562271, 717907-75-0, PF00562271, PF 00562271, N-METHYL-N-[3-[[[2-[(2-OXO-2,3-DIHYDRO-1H-INDOL-5-YL)AMINO]-5-TRIFLUOROMETHYLPYRIMIDIN-4-YL]AMINO]METHYL]PYRIDIN-2-YL]METHANESULFONAMIDE, N-methyl-N-(3-((2-(2-oxoindolin-5-ylamino)-5-(trifluoromethyl)pyrimidin-4-ylamino)methyl)pyridin-2-yl)methanesulfonamide benzenesulfonate, N-methyl-N-[3-[[[2-[(2-oxo-1,3-dihydroindol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide, N-methyl-N-{3-[({2-[(2-oxo-1,3-dihydroindol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamide, Kinome_3857, 3bz3, AGN-PC-00ENC7, SureCN1206959, CHEMBL1084546, CTK2H5401, CHEBI:730975, MolPort-016-631-879, BCPP000114, HMS3244K07, HMS3244K08, HMS3244L07, HMS3265M11
InChIKey: MZDKLVOWGIOKTN-UHFFFAOYSA-N | ||||||||
| • PF-562271 besylate
IUPAC Name: benzenesulfonic acid;N-methyl-N-[3-[[[2-[(2-oxo-1,3-dihydroindol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | CAS Registry Number: 939791-38-5 Synonyms: CHEMBL2430359, PF 562271, PF-00562271, cc-23, RS0038s, PF-562,271, Methanesulfonamide, N-(3-(((2-((2,3-dihydro-2-oxo-1H-indol-5-yl)amino)-5- (trifluoromethyl)-4-pyrimidinyl)amino)methyl)-2-pyridinyl)-N-methyl-, benzenesulfonate (1:1), Methanesulfonamide, N-[3-[[[2-[(2,3-dihydro-2-oxo-1H-indol-5-yl)amino]-5-(trifluoromethyl)-4-pyrimidinyl]amino]methyl]-2-pyridinyl]-N-methyl-, benzenesulfonate (1:1)
InChIKey: LKLWTLXTOVZFAE-UHFFFAOYSA-N | ||||||||
| • PF-573228
IUPAC Name: 6-[[4-[(3-methylsulfonylphenyl)methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3,4-dihydro-1H-quinolin-2-one | CAS Registry Number: 869288-64-2 Synonyms: PF 573228, PF-228, AG-H-50453, 3,4-DIHYDRO-6-[[4-[[[3-(METHYLSULFONYL)PHENYL]METHYL]AMINO]-5-(TRIFLUOROMETHYL)-PYRIMIDIN-2-YL]AMINO]-2(1H)-QUINOLINONE, 6-((4-((3-(methanesulfonyl)benzyl)amino)-5-trifluoromethylpyrimidin-2-yl)amino)-3,4-dihydro-1h-quinolin-2-one, 6-[(4-((3-(Methanesulfonyl)benzyl)amino)-5-trifluoromethylpyrimidin-2-yl)amino]-3,4-dihydro-1H-quinolin-2-one, AGN-PC-00CNZ9, SureCN5212404, cc-288, CHEMBL514554, CTK5F7396, CHEBI:606482, HMS3262N09, DNC008520, CCG-222168, QC-7329, RL05385, NCGC00263133-01, PF 573228 pound>>PF573228, BCP0726000162
InChIKey: HESLKTSGTIBHJU-UHFFFAOYSA-N | ||||||||
| • PF04929113
IUPAC Name: [4-[2-carbamoyl-5-[6,6-dimethyl-4-oxo-3-(trifluoromethyl)-5,7-dihydroindazol-1-yl]anilino]cyclohexyl] 2-aminoacetate | CAS Registry Number: 908115-27-5 Synonyms: SNX-5422, SNX5422, SNX 5422, PF 04929113, PF-04929113, SNX-5422, PF-04929113, 908115-27-5, cc-40, SureCN1220790, SureCN1220791, UNII-BF52J69Q8T, BCPP000065, ABP000737, DCL000231, CS-0272, RL05706, NCGC00346640-01, HY-10213, PF-4929113, X7589, PF 04929113, SNX 5422
InChIKey: AVDSOVJPJZVBTC-UHFFFAOYSA-N | ||||||||
| • PFI-1
IUPAC Name: 2-methoxy-N-(3-methyl-2-oxo-1,4-dihydroquinazolin-6-yl)benzenesulfonamide | CAS Registry Number: 1403764-72-6 Synonyms: CHEMBL2179387, PFI1, SureCN14721611, QCR-192, 4e96, CS-1362, HY-16586, PFI-1 (PF-6405761), KB-145941, PFI-1|1403764-72-6|PFI1, S1216,PF-06405761,
InChIKey: TXZPMHLMPKIUGK-UHFFFAOYSA-N | ||||||||
| • PH-797804
IUPAC Name: 3-[3-bromo-4-[(2,4-difluorophenyl)methoxy]-6-methyl-2-oxopyridin-1-yl]-N,4-dimethylbenzamide | CAS Registry Number: 586379-66-0 Synonyms: PH 797804, PH797804, 3-(3-Bromo-4-((2,4-difluorobenzyl)oxy)-6-methyl-2-oxopyridin-1(2H)-yl)-N,4-dimethylbenzamide, 586379-66-0 pound not PH797804 pound not PH 797804, 3-{3-Bromo-4-[(2,4-Difluorobenzyl)oxy]-6-Methyl-2-Oxopyridin-1(2h)-Yl}-N,4-Dimethylbenzamide, 3hll, Kinome_3761, cc-53, SureCN2015676, UNII-SI09I1V827, CHEMBL1088751, CTK8C3874, CHEBI:719399, MolPort-021-804-991, BCPP000113, ANW-70744, AKOS016007727, CS-0465, DB07941, PHA-797804
InChIKey: KCAJXIDMCNPGHZ-UHFFFAOYSA-N | ||||||||
| • PHA-665752
IUPAC Name: (3Z)-5-[(2,6-dichlorophenyl)methylsulfonyl]-3-[[3,5-dimethyl-4-[(2R)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1H-pyrrol-2-yl]methylidene]-1H-indol-2-one | CAS Registry Number: 477575-56-7 Synonyms: PHA665752, PHA 665752, TCMDC-125885, (2R)-1-[[5-[(Z)-[5-[[(2,6-DICHLOROPHENYL)METHYL]SULFONYL]-1,2-DIHYDRO-2-OXO-3H-INDOL-3-YLIDENE]METHYL]-2,4-DIMETHYL-1H-PYRROL-3-YL]CARBONYL]-2-(1-PYRROLIDINYLMETHYL)PYRROLIDINE, (R,Z)-5-(2,6-dichlorobenzylsulfonyl)-3-((3,5-dimethyl-4-(2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl)-1H-pyrrol-2-yl)methylene)indolin-2-one, PHA665752, PHA-665752, S1070_Selleck, SureCN93654, cc-47, UNII-0VXU5T5R3J, CHEMBL450786, CHEBI:547415, MolPort-021-804-992, BCPP000112, HMS3269N19, ABP000082, AKOS015896678, CS-0137, QC-7247, RL03780
InChIKey: OYONTEXKYJZFHA-SSHUPFPWSA-N | ||||||||
| • PHA-680632
IUPAC Name: N-(2,6-diethylphenyl)-3-[[4-(4-methylpiperazin-1-yl)benzoyl]amino]-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazole-5-carboxamide | CAS Registry Number: 398493-79-3 Synonyms: Pha 680632, N-(2,6-Diethylphenyl)-4,6-dihydro-3-[[4-(4-methyl-1-piperazinyl)benzoyl]amino]pyrrolo[3,4-c]pyrazole-5(1H)-carboxamide, PHA680632, 398493-79-3, PHA680632, PHA-680632, S1454_Selleck, SureCN12582821, cc-476, CHEMBL363160, CTK8B6777, MolPort-016-633-216, BCPP000111, ABP000945, ANW-54326, DNC005484, AKOS015999833, CS-0194, QC-8220, RL03525, NCGC00346526-01, AK-51091
InChIKey: OBWNXGOQPLDDPS-UHFFFAOYSA-N | ||||||||
| • PHA-767491
IUPAC Name: 2-pyridin-4-yl-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-one | CAS Registry Number: 845714-00-3 Synonyms: PHA 767491, PHA767491, 845714-00-3 pound not PHA767491 pound not PHA 767491, Pyrrolopyridinone, 1, Cdc7/Cdk9 Inhibitor, Kinome_2973, AGN-PC-00EP4J, SureCN4767679, cc-260, CHEMBL225519, CTK8F8505, MolPort-009-019-436, HMS3229B21, CAY10572, CAY 10572, CAY-10572, DNC007421, ZINC16052718, AG-L-65185, CS-1208
InChIKey: DKXHSOUZPMHNIZ-UHFFFAOYSA-N | ||||||||
| • PHA-793887
IUPAC Name: N-[6,6-dimethyl-5-(1-methylpiperidine-4-carbonyl)-1,4-dihydropyrrolo[3,4-c]pyrazol-3-yl]-3-methylbutanamide | CAS Registry Number: 718630-59-2 Synonyms: CHEMBL1230607, PHA793887, PHA-793887, PHA793887, 3-Methyl-N-[1,4,5,6-tetrahydro-6,6-dimethyl-5-[(1-methyl-4-piperidinyl)carbonyl]pyrrolo[3,4-c]pyrazol-3-yl]butanamide, N-(6,6-Dimethyl-5-(1-methylpiperidine-4-carbonyl)-1,4,5,6-tetrahydropyrrolo(3,4-C)pyrazol-3-yl)-3-methylbutanamide, N-(6,6-dimethyl-5-(1-methylpiperidine-4-carbonyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl)-3-methylbutanamide, S1487_Selleck, SureCN5110328, UNII-MKS45S912B, cc-404, CTK5D5171, BCPP000110, HMS3265M13, HMS3265M14, HMS3265N13, HMS3265N14, AKOS015995002, AG-I-03437, PHA 793887, QC-8186
InChIKey: HUXYBQXJVXOMKX-UHFFFAOYSA-N | ||||||||
| • Phenformin hydrochloride
IUPAC Name: 1-(diaminomethylidene)-2-phenethylguanidine hydrochloride | CAS Registry Number: 834-28-6 Synonyms: Meltrol, Dipar, Phenformin.HCl, Phenformin HCl, Phenethylbiguanide, Meltrol-50, PHENFORMIN HYDROCHLORIDE, Prestwick_615, DBI-TD, Phenformin, hydrochloride, USAF VI-6, Phenoformine hydrochloride, Phenethylbiguanide hydrochloride, Phenformin HCl No. 9113, CCRIS 4857, C10H15N5.HCl, MLS000028506, MLS001148130, MLS002154228, P7045_SIGMA
InChIKey: YSUCWSWKRIOILX-UHFFFAOYSA-N | ||||||||
| • Phenol, 2-methyl-5-nitro-, acetate (ester)
IUPAC Name: (2-methyl-5-nitrophenyl) acetate | CAS Registry Number: 54362-24-2 Synonyms: 2-methyl-5-nitrophenyl acetate, 2-acetoxy-4-nitrotoluene, ZNDOXROITOAJQJ-UHFFFAOYSA-N, 2-acetoxy4-nitrotoluene, SCHEMBL1469841, CTK8J1558, AKOS022183509, AJ-95083, AK-80692, KB-231582, phenol, 2-methyl-5-nitro-, acetate (ester)
InChIKey: ZNDOXROITOAJQJ-UHFFFAOYSA-N | ||||||||
| • PHT-427
IUPAC Name: 4-dodecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamide | CAS Registry Number: 1191951-57-1 Synonyms: PHT427, PHT 427, PHT427, PHT 427, PHT-427, S1556_Selleck, SureCN283080, cc-348, CHEMBL595583, CHEBI:693526, CS-0223, RL00742, PHT-427-Supplied by Selleck Chemicals, NCGC00346547-01, HY-12063, BCP0726000128, 4-Dodecyl-N-1,3,4-thiadiazol-2-ylbenzenesulfonamide, 4-dodecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamide, PHT-427|1191951-57-1|PHT427, PHT427, PHT 427, 1191951-57-1, pound molweight:409.60904) , PHT427, PHT 427, 1191951-57-1
InChIKey: BYWWNRBKPCPJMG-UHFFFAOYSA-N | ||||||||
| • PI-103
IUPAC Name: 3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin-2-yl)phenol | CAS Registry Number: 371935-74-9 Synonyms: PI103, PI 103, 3-(4-morpholinopyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenol, 3-(4-(4-Morpholinyl)pyrido[3′,2′:4,5]furo[3,2-d]pyrimidin-2-yl)phenol, 3-(4-Morpholin-4-Ylpyrido[3',2':4,5]furo[3,2-D]pyrimidin-2-Yl)phenol, 3-[4-Morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyriMidin-2-yl]phenol, X6K, S1038_Selleck, Kinome_3597, 2x6k, cc-5, SureCN258242, UNII-YQX02F616F, CHEMBL573339, CTK8F1083, PIK-103, QCR-256, MolPort-009-019-225, pyridofuropyrimidine derivative, 2, BCPP000107
InChIKey: TUVCWJQQGGETHL-UHFFFAOYSA-N | ||||||||
| • Piceatannol
IUPAC Name: 5-[(E)-2-(3,4-dihydroxyphenyl)ethenyl]benzene-1,3-diol | CAS Registry Number: 10083-24-6 Synonyms: piceatannol, astringinin, piceatanol, Astringinine, 3-Hydroxyresveratol, E-Piceatannol, 3'-hydroxyresveratol, demethyl isorhapontigenin, BiomolKI_000023, 3,5,3',4'-Tetrahydroxystilbene, BiomolKI2_000031, RSVL-1, 3,3',4,5'-Stilbenetetrol, 3,3',4,5'-Tetrahydroxystilbene, Lopac0_000915, BSPBio_001120, MLS002153321, 3,3',4'5-Tetrahydroxystilbene, P0453_SIGMA, 3,3',4',5-tetrahydroxystilbene
InChIKey: CDRPUGZCRXZLFL-OWOJBTEDSA-N | ||||||||
| • Pictilisib
IUPAC Name: 4-[2-(1H-indazol-4-yl)-6-[(4-methylsulfonylpiperazin-1-yl)methyl]thieno[3,2-d]pyrimidin-4-yl]morpholine | CAS Registry Number: 957054-30-7 Synonyms: GDC-0941, GDC0941, GDC 0941, Pictrelisib, S1065_Selleck, Kinome_3719, CHEMBL521851, 4-(2-(1H-Indazol-4-yl)-6-((4-(methylsulfonyl)piperazin-1-yl)methyl)thieno[3,2-d]pyrimidin-4-yl)morpholine, CHEBI:65326, GDC-0941, GDC0941, 2-(1H-Indazol-4-yl)-6-(4-methanesulfonylpiperazin-1-ylmethyl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidine, 4-[2-(1H-indazol-4-yl)-6-[(4-methylsulfonylpiperazin-1-yl)methyl]thieno[3,2-d]pyrimidin-4-yl]morpholine, GD9, 2-(1h-Indazol-4-Yl)-6-{[4-(Methylsulfonyl)piperazin-1-Yl]methyl}-4-Morpholin-4-Yl-Thieno[3,2-D]pyrimidine, 4-(2-(1H-indazol-4-yl)-6-((4-(methylsulfonyl)piperazin-1-yl)methyl)thieno(3,2-d)pyrimidin-4-yl)morpholine, Pictrelisib [INN], Pictilisib (USAN), PICTILISIB, PubChem16427, nchembio.293-comp12
InChIKey: LHNIIDJUOCFXAP-UHFFFAOYSA-N | ||||||||
| • Pifithrin-α hydrobromide
IUPAC Name: 2-(2-imino-4,5,6,7-tetrahydro-1,3-benzothiazol-3-yl)-1-(4-methylphenyl)ethanone | CAS Registry Number: 63208-82-2 Synonyms: nchembio809-comp3, nchembio790-comp33, Tocris-1267, BSPBio_001026, CBDivE_001116, KBioGR_000366, KBioSS_000366, BCBcMAP01_000143, KBio2_000366, KBio2_002934, KBio2_005502, KBio3_000711, KBio3_000712, CID4817, CHEBI:429136, Bio1_000477, Bio1_000966, Bio1_001455, Bio2_000353, Bio2_000833
InChIKey: OLTZHXYLLRJLST-UHFFFAOYSA-N | ||||||||
| • Pifithrin-μ
IUPAC Name: 2-phenylethynesulfonamide | CAS Registry Number: 64984-31-2 Synonyms: Pifithrin-mu, nchembio809-comp1, 2-Phenylethynesulfonamide, Phenylacetylenylsulfonamide, Ambcb5147472, Oprea1_468179, Oprea1_544600, P0122_SIGMA, MolPort-000-417-310, NSC303580, HMS1579M04, PFTμ, CID327653, ZINC00164402, NCGC00162358-01, NCGC00162358-02, NCGC00162358-03, BRD-K96799727-001-01-7
InChIKey: ZZUZYEMRHCMVTB-UHFFFAOYSA-N |