Profile: Jinan Trio PharmaTech Co., Ltd. specializes in APIs & intermediates, heterocyclic compounds, and anti-tumor drugs. Our products include crizotinib, vemurafenib, afatinib, vandetanib, regorafenib, brivanib alaninate, pyridazine, imidazole, pyrazole, and oxazole. We are specialized in providing over 1000 products including molecular targeted anticancer drugs, cell signaling pathway inhibitors, pharmaceutical intermediates, and heterocyclic compounds, and quality services including custom synthesis, transfer of new drug patent and technology, technical cooperation, and process optimization.
| • Quizartinib
IUPAC Name: 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-[4-[6-(2-morpholin-4-ylethoxy)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenyl]urea | CAS Registry Number: 950769-58-1 Synonyms: AC-220, AC220, AC 220, AC010220, AC-220, AC220, AC220,Quizartinib, S1526_Selleck, AC220 - Quizartinib, SureCN72923, Quizartinib (USAN/INN), Quizartinib [USAN:INN], cc-62, UNII-7LA4O6Q0D3, CHEMBL576982, CHEBI:673133, BCPP000443, HMS3244K09, HMS3244K10, HMS3244L09, HMS3265G09
InChIKey: CVWXJKQAOSCOAB-UHFFFAOYSA-N | ||||||||
| • R406
IUPAC Name: benzenesulfonate;6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)pyrimidin-4-yl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one | CAS Registry Number: 841290-81-1 Synonyms: KB-80318
InChIKey: UXDRJPYSTZHIOE-UHFFFAOYSA-M | ||||||||
| • R406 free base
IUPAC Name: 6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)pyrimidin-4-yl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one | CAS Registry Number: 841290-80-0 Synonyms: R406(free base), R-406, 6-(5-fluoro-2-(3,4,5-trimethoxyphenylamino)pyrimidin-4-ylamino)-2,2-dimethyl-2H-pyrido[3,2-b][1,4]oxazin-3(4H)-one, 6-({5-Fluoro-2-[(3,4,5-Trimethoxyphenyl)amino]pyrimidin-4-Yl}amino)-2,2-Dimethyl-2h-Pyrido[3,2-B][1,4]oxazin-3(4h)-One, 6-[[5-Fluoro-2-[(3,4,5-trimethoxyphenyl)amino]-4-pyrimidinyl]amino]-2,2-dimethyl-2H-pyrido[3,2-b]-1,4-oxazin-3(4H)-one, R 406, 3fqs, 3piy, 6-((5-fluoro-2-((3,4,5-trimethoxyphenyl)amino)-4-pyrimidinyl)amino)-2,2-dimethyl-2h-pyrido(3,2-b)-1,4-oxazin-3(4h)-one, S1533_Selleck, Kinome_1211, PubChem22483, 841290-81-1, SureCN1200144, QCR-9, cc-243, AGN-PC-004I2D, CHEMBL475251, CTK5F1857, CHEBI:560144
InChIKey: NHHQJBCNYHBUSI-UHFFFAOYSA-N | ||||||||
| • R547
IUPAC Name: [4-amino-2-[(1-methylsulfonylpiperidin-4-yl)amino]pyrimidin-5-yl]-(2,3-difluoro-6-methoxyphenyl)methanone | CAS Registry Number: 741713-40-6 Synonyms: R-547, 741713-40-6 pound not R 547, (4-Amino-2-{[1-(Methylsulfonyl)piperidin-4-Yl]amino}pyrimidin-5-Yl)(2,3-Difluoro-6-Methoxyphenyl)methanone, [4-Amino-2-[(1-methylsulfonylpiperidin-4-yl)amino]pyrimidin-5-yl](2,3-difluoro-6-methoxyphenyl)methanone, (4-Amino-2-[(1-methylsulfonylpiperidin-4-yl)amino)pyrimidin-5-yl)(2,3-difluoro-6-methoxyphenyl)methanone, SureCN2397067, UNII-T61871RKRI, cc-270, CS-0022, RL04812, NCGC00346632-01, HY-10014, KB-36226, FT-0687511, R 547, RO-4584820, Y0369, R547|741713-40-6|R-547, 4-Amino-2-(1-methylsulfonylpiperidin-4-yl)aminopyrimidin-5-yl(2,3-difluoro-6-methoxyphenyl)methanone, 5-(2,3-difluoro-6-methoxybenzoyl)-2-N-(1-methanesulfonylpiperidin-4-yl)pyrimidine-2,4-diamine
InChIKey: JRNJNYBQQYBCLE-UHFFFAOYSA-N | ||||||||
| • Rabusertib
IUPAC Name: 1-[5-bromo-4-methyl-2-[[(2S)-morpholin-2-yl]methoxy]phenyl]-3-(5-methylpyrazin-2-yl)urea | CAS Registry Number: 911222-45-2 Synonyms: LY2603618, LY 2603618, LY-2603618, Rabusertib [USAN], Rabusertib (USAN/INN), SureCN304747, UNII-3S9L1NU6U7, cc-579, CHEMBL3039517, MolPort-021-804-967, BCPP000178, IC-83, BCP9000873, CS-0472, RL05730, NCGC00343768-01, HY-14720, LY2603618 - IC-83, D10397, IC-83, LY 2603618, 911222-45-2
InChIKey: SYYBDNPGDKKJDU-ZDUSSCGKSA-N | ||||||||
| • RAF265
IUPAC Name: 1-methyl-5-[2-[5-(trifluoromethyl)-1H-imidazol-2-yl]pyridin-4-yl]oxy-N-[4-(trifluoromethyl)phenyl]benzimidazol-2-amine | CAS Registry Number: 927880-90-8 Synonyms: CHIR-265, RAF-265, CHIR265, RAF 265, RAF265(CHIR-265), RAF265, CHIR-265, 927880-90-8, CHIR-265 , 927880-90-8, CHIR265, 1-Methyl-5-[[2-[5-(trifluoromethyl)-1h-imidazol-2-yl]-4-pyridinyl]oxy]-n-[4-(trifluoromethyl)phenyl]-1h-benzimidazol-2-amine, S2161_Selleck, PubChem22594, cc-117, AGN-PC-00DJ96, CHEMBL558752, CHIR 265, MolPort-016-633-290, ACN-S001859, RAF 265, CHIR 265, RAF265 - CHIR-265, ABP000414, CHIR 265 (RAF 265)
InChIKey: YABJJWZLRMPFSI-UHFFFAOYSA-N | ||||||||
| • Ralimetinib dimesylate
IUPAC Name: 5-[2-tert-butyl-4-(4-fluorophenyl)-1H-imidazol-5-yl]-3-(2,2-dimethylpropyl)imidazo[4,5-b]pyridin-2-amine;methanesulfonic acid | CAS Registry Number: 862507-23-1 Synonyms: LY2228820, LY-2228820, LY-2228820, LY2228820, LY 2228820, Ralimetinib Mesylate, S1494_Selleck, UNII-QUW7B71FO9, AGN-PC-00BT9J, cc-430, CHEMBL2364627, LY2228820 2MsOH, MolPort-016-633-222, BCPP000179, BCP9000872, CS-0208, LSN-2322600, HY-13241, LY2228820-Supplied by Selleck Chemicals, FT-0670881, LY2228820|862507-23-1|LY2228820 2MsOH|LY 2228820|LY-2228820
InChIKey: NARMJPIBAXVUIE-UHFFFAOYSA-N | ||||||||
| • Raltitrexed
IUPAC Name: (2S)-2-[[5-[methyl-[(2-methyl-4-oxo-1H-quinazolin-6-yl)methyl]amino]thiophene-2-carbonyl]amino]pentanedioic acid | CAS Registry Number: 112887-68-0 Synonyms: Tomudex, 2kce, 2tsr, Tomudex (TN), ICI D1694, ZD1694, ICI-D1694, MLS001424225, Raltitrexed (JAN/USAN/INN), STOCK6S-47020, C21H22N4O6S, 1i00, AIDS106596, ICI-D-1694, AIDS-106596, ZD 1694, ZD-1694, ZN-D1694, CID104758, NSC639186
InChIKey: IVTVGDXNLFLDRM-HNNXBMFYSA-N | ||||||||
| • Rapamycin
Synonyms: rapamycin, Sirolimus, Rapamune, 1fkb, 1pbk, LCP-Siro, (-)-Rapamycin, nchembio.79-comp1, nchembio762-comp1, nchembio883-comp3, nchembio.100-comp4, Sirolimus (RAPAMUNE), (-)-Rapamycin;Rapamune, Antibiotic AY 22989, BiomolKI2_000084, nchembio.2007.42-comp2, Sirolimus [USAN:BAN:INN], CCRIS 9024, R0395_SIAL, SILA 9268A
InChIKey: QFJCIRLUMZQUOT-HPLJOQBZSA-N | ||||||||
| • Rebastinib
IUPAC Name: 4-[4-[(5-tert-butyl-2-quinolin-6-ylpyrazol-3-yl)carbamoylamino]-3-fluorophenoxy]-N-methylpyridine-2-carboxamide | CAS Registry Number: 1020172-07-9 Synonyms: DCC-2036, REBASTINIB, DCC 2036, CHEBI:62166, DCC2036, Rebastinib (USAN), Rebastinib [USAN], DCC 2036, DCC2036, 357263-13-9, 4-[4-({[3-Tert-Butyl-1-(Quinolin-6-Yl)-1h-Pyrazol-5-Yl]carbamoyl}amino)-3-Fluorophenoxy]-N-Methylpyridine-2-Carboxamide, 3qri, 3qrj, SureCN2034290, cc-606, CHEMBL1738757, QCR-201, UNII-75017Q6I97, BCP9000591, CS-1038, DP 1919, NCGC00263172-01
InChIKey: WVXNSAVVKYZVOE-UHFFFAOYSA-N | ||||||||
| • Refametinib
IUPAC Name: N-[3,4-difluoro-2-(2-fluoro-4-iodoanilino)-6-methoxyphenyl]-1-[(2S)-2,3-dihydroxypropyl]cyclopropane-1-sulfonamide | CAS Registry Number: 923032-37-5 Synonyms: BAY 869766, RDEA119, RDEA 119, Refametinib [INN], 3e8n, UNII-JPX07AFM0N, BAY 86-9766, BAY 8697661, NCGC00188380-01, NCGC00188380-02, Cyclopropanesulfonamide, N-(3,4-difluoro-2-((2-fluoro-4-iodophenyl)amino)-6-methoxyphenyl)-1-((2S)-2,3-dihydroxypropyl)-, N-{3,4-difluoro-2-[(2-fluoro-4-iodophenyl)amino]-6-methoxyphenyl}-1-[(2S)-2,3-dihydroxypropyl]cyclopropane-1-sulfonamide, VRA
InChIKey: RDSACQWTXKSHJT-NSHDSACASA-N | ||||||||
| • Regorafenib
IUPAC Name: 4-[4-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]-3-fluorophenoxy]-N-methylpyridine-2-carboxamide | CAS Registry Number: 755037-03-7 Synonyms: BAY 73-4506, Regorafenibum, Stivarga, UNII-24T2A1DOYB, BAY73-4506, CHEMBL1946170, CHEBI:68647, Regorafenib, 755037-03-7, 4-[4-({[4-Chloro-3-(trifluoromethyl)phenyl]carbamoyl}amino)-3-fluorophenoxy]-N-methylpyridine-2-carboxamide, BAY-73-4506, 4-(4-(3-(4-Chloro-3-(trifluoromethyl)phenyl)ureido)-3-fluorophenoxy)-N-methylpicolinamide, Regorafenib, BAY 73-4506, 4-(4-(((4-chloro-3-(trifluoromethyl)phenyl)carbamoyl}amino)-3-fluorophenoxy)-N-methylpyridine-2-carboxamide, S1178_Selleck, Regorafenib (USAN/INN), Regorafenib [USAN:INN], SureCN432230, 24T2A1DOYB, BAY-734506 monohydrate, BAY73-4506 hydrochloride
InChIKey: FNHKPVJBJVTLMP-UHFFFAOYSA-N | ||||||||
| • RepSox
IUPAC Name: 2-[5-(6-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,5-naphthyridine | CAS Registry Number: 446859-33-2 Synonyms: 1vjy, ALK5 Inhibitor II, CHEBI:406655, TGF-beta RI Kinase Inhibitor II, CID449054, IN1052, EN002636, 2-(3-(6-Methylpyridin-2-yl)-1H-pyrazol-4-yl)-1,5-naphthyridine, 2-[3-(6-methylpyridin-2-yl)-2H-pyrazol-4-yl]-1,5-naphthyridine, Transforming Growth Factor-beta Type I Receptor Kinase Inhibitor II, 2-[3-(6-Methyl-pyridin-2-yl)-1H-pyrazol-4-yl]-[1,5]naphthyridine
InChIKey: LBPKYPYHDKKRFS-UHFFFAOYSA-N | ||||||||
| • Resveratrol
IUPAC Name: 5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol | CAS Registry Number: 501-36-0 Synonyms: resveratrol, trans-resveratrol, (E)-resveratrol, 3,4',5-Stilbenetriol, 3,4',5-Trihydroxystilbene, Prestwick_619, 3,5,4'-Trihydroxystilbene, nchembio.140-comp2, Prestwick2_000508, Prestwick3_000508, Spectrum5_000552, Lopac0_001111, BSPBio_000435, BSPBio_001114, BSPBio_003461, 3,4',5-trihydroxy-stilbene, MLS000069735, MLS001055357, MLS001076538, R5010_SIGMA
InChIKey: LUKBXSAWLPMMSZ-OWOJBTEDSA-N | ||||||||
| • RG108
IUPAC Name: (2R)-2-(1,3-dioxoisoindol-2-yl)-3-(1H-indol-3-yl)propanoic acid | CAS Registry Number: 48208-26-0 Synonyms: RG 108, AC1LDWK4, SureCN11949518, (2R)-2-(1,3-dioxoisoindol-2-yl)-3-(1H-indol-3-yl)propanoic acid
InChIKey: HPTXLHAHLXOAKV-MRXNPFEDSA-N | ||||||||
| • Ridaforolimus
Synonyms: Deforolimus, D08900, Ridaforolimus (JAN/USAN)
InChIKey: BUROJSBIWGDYCN-SXVXPMCXSA-N | ||||||||
| • Rilmenidine
IUPAC Name: N-(dicyclopropylmethyl)-4,5-dihydro-1,3-oxazol-2-amine | CAS Registry Number: 54187-04-1 Synonyms: Oxaminozoline, Rilmenidene, Rilmenidine [INN], Rilmenidia [Spanish], Rilmenidinum [Latin], nchembio.79-comp13, Tocris-0790, Lopac-R-134, Prestwick0_000982, Prestwick1_000982, Prestwick2_000982, Prestwick3_000982, R134_SIGMA, Rilmenidene hemifumarate salt, Rilmenidine hemifumarate salt, Lopac0_001104, BSPBio_001043, Oxaminozoline hemifumarate salt, RILMENIDINE HEMIFUMARATE, SPBio_002944
InChIKey: CQXADFVORZEARL-UHFFFAOYSA-N | ||||||||
| • RITA
IUPAC Name: [5-[5-[5-(hydroxymethyl)thiophen-2-yl]furan-2-yl]thiophen-2-yl]methanol | CAS Registry Number: 213261-59-7 Synonyms: SOS BISMETHANOL, NCIChal_000017, NCIMech_000598, p53 Activator III, RITA, NSC652287, NSC 652287, CID374536, ZINC00006846, NCGC00159570-01, 2,5-bis(5-hydroxymethyl-2-thienyl)furan, NCI60_018346, 2,5-bis-(5-Hydroxymethyl-2-thienyl)-furan, Furan, 2,5-bis[5-(hydroxymethyl)-2-thienyl]-, 2-thiophenemethanol, 5,5'-(2,5-furandiyl)bis-, Thiophene-2-methanol, 5,5'-(2,5-furandiyl)bis-, 2-Thiophenemethanol, 5,5'-(2,5-furandiyl)bis- (9CI), Reactivation of p53 and Induction of Tumor cell Apoptosis
InChIKey: KZENBFUSKMWCJF-UHFFFAOYSA-N | ||||||||
| • Ritonavir
IUPAC Name: 1,3-thiazol-5-ylmethyl N-[(2S,3S,5S)-3-hydroxy-5-[[(2S)-3-methyl-2-[[methyl-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]carbamoyl]amino]butanoyl]amino]-1,6-di(phenyl)hexan-2-yl]carbamate | CAS Registry Number: 155213-67-5 Synonyms: ritonavir, Norvir, Kaletra, Mixture Name, 1hxw, Ritonavir [USAN], Component of Kaletra, Norvir (TM), Norvir (TN), Abbott 84538, 1sh9, ABT-538, MLS000759541, MLS001424063, Ritonavir (JAN/USAN/INN), ABT538, STOCK6S-48483, HSDB 7160, C37H48N6O5S2, NSC693184
InChIKey: NCDNCNXCDXHOMX-XGKFQTDJSA-N | ||||||||
| • RKI-1447
IUPAC Name: 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | CAS Registry Number: 1342278-01-6 Synonyms: 1-[(3-Hydroxyphenyl)methyl]-3-(4-Pyridin-4-Yl-1,3-Thiazol-2-Yl)urea, AGN-PC-0DA78E, FD5032, KB-02617, QC-10897, 1-(3-hydroxybenzyl)-3-(4-(pyridin-4-yl)thiazol-2-yl)urea, 07R
InChIKey: GDVRVPIXWXOKQO-UHFFFAOYSA-N | ||||||||
| • RO 09-1978
IUPAC Name: pentyl N-[1-[(2R,3R,4S,5R)-3,4-dihydroxy-5-methyloxolan-2-yl]-5-fluoro-2-oxopyrimidin-4-yl]carbamate | CAS Registry Number: 158798-73-3 Synonyms: Xeloda, CAPECITABINE, capecitabina, capecitabinum, Capecitabin, Capiibine, Caxeta, Xabine, Xeloda (TN), Capecitabine [USAN], UNII-6804DJ8Z9U, Capecitabine (JAN/USAN/INN), C15H22FN3O6, CHEBI:31348, HSDB 7656, CHEBI:698447, MolPort-005-938-254, CID60953, RG-340, Ro 09-1978
InChIKey: GAGWJHPBXLXJQN-UORFTKCHSA-N | ||||||||
| • Ro 31-8220 Mesylate
IUPAC Name: methanesulfonic acid;3-[3-[4-(1-methylindol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]propyl carbamimidothioate | CAS Registry Number: 138489-18-6 Synonyms: Ro 31-8220 mesylate, CHEMBL1591531, InSolution™ Ro-31-8220, Bisindolylmaleimide IX, Methanesulfonate, Ro-31-8220, 3-[1-[3-(Amidinothio)propyl-1H-indol-3-yl]-3-(1-methyl-1H-indol-3-yl)maleimide, Bisindoylmaleimidine IX, BMK1-D9, AGN-PC-00CZ01, BIMI0821, HMS3229N17, HMS3268D19, Ro 31-8220 methanesulfonate salt, IN1117, S7207,Bisindolylmaleimide IX Mesylate, NCGC00092293-01, Bisindolylmaleimide IX methanesulphonate salt, 2-{1-[3-(Amidinothio)propyl]-1H-indol-3-yl}-3-(1-methylindol-3-yl)maleimide methanesulfonate salt, 3-(3-(4-(1-methyl-1H-indol-3-yl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-yl)-1H-indol-1-yl)propyl carbamimidothioate methanesulfonate, methanesulfonic acid;3-[3-[4-(1-methylindol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]propyl carbamimidothioate
InChIKey: SAWVGDJBSPLRRB-UHFFFAOYSA-N | ||||||||
| • Ro3280
IUPAC Name: 4-[(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-8H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | CAS Registry Number: 1062243-51-9 Synonyms: CHEMBL2392553, Ro-3280, PharmaGSID_48511, DSSTox_CID_28485, DSSTox_RID_82762, DSSTox_GSID_48511, SCHEMBL1559146, DJNZZLZKAXGMMC-UHFFFAOYSA-N, MolPort-028-600-021, Tox21_303518, CS-1673, NCGC00257406-01, HY-15161, KB-80400, S7248,Ro5203280, CAS-1062243-51-9, 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide, 4-(9-Cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide
InChIKey: DJNZZLZKAXGMMC-UHFFFAOYSA-N | ||||||||
| • RO4929097
IUPAC Name: 2,2-dimethyl-N-[(7S)-6-oxo-5,7-dihydrobenzo[d][1]benzazepin-7-yl]-N'-(2,2,3,3,3-pentafluoropropyl)propanediamide | CAS Registry Number: 847925-91-1 Synonyms: Ro 4929097, RO-4929097, RO-4929097,RO4929097, S1575_Selleck, cc-19, UNII-KK8645V7LE, MolPort-016-633-243, BCPP000088, CS-0480, RG-4733, RL05211, NCGC00263162-01, NCGC00263162-02, HY-11102, RO4929097-Supplied by Selleck Chemicals, X7559, R-4733, RO4929097|847925-91-1|RO 4929097, RO-4929097,RO 4929097, 847925-91-1, pound molweight:469.404516) , RO-4929097, RO 4929097, 847925-91-1
InChIKey: OJPLJFIFUQPSJR-INIZCTEOSA-N | ||||||||
| • Roniciclib
IUPAC Name: (2R,3R)-3-[2-[4-(cyclopropylsulfonimidoyl)anilino]-5-(trifluoromethyl)pyrimidin-4-yl]oxybutan-2-ol | CAS Registry Number: 1223498-69-8 Synonyms: BAY 1000394, UNII-0W9Q8U337A
InChIKey: UELYDGOOJPRWGF-SRQXXRKNSA-N | ||||||||
| • Roxadustat
IUPAC Name: 2-[(4-hydroxy-1-methyl-7-phenoxyisoquinoline-3-carbonyl)amino]acetic acid | CAS Registry Number: 808118-40-3 Synonyms: FG-4592, CHEMBL2338329, N-[(4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinyl)carbonyl]glycine, Glycine, N-[(4-hydroxy-1-methyl-7-phenoxy-3-isoquinolinyl)carbonyl]-, n-((4-hydroxy-1-methyl-7-phenoxy-3-isoquinolinyl)carbonyl)glycine, (((4-Hydroxy-1-methyl-7-phenoxyisoquinolin-3-yl)carbonyl)amino)acetic acid, [[(4-Hydroxy-1-methyl-7-phenoxyisoquinolin-3-yl)carbonyl]amino]acetic Acid, PubChem24327, SureCN523705, UNII-X3O30D9YMX, cc-211, AGN-PC-005EN5, CTK2I7260, MolPort-021-804-955, BCPP000230, FG-4592,ASP1517, BCP9000684, CS-1094, FG 4592, QC-7436
InChIKey: YOZBGTLTNGAVFU-UHFFFAOYSA-N | ||||||||
| • Rubitecan
Synonyms: Rubitecan (USAN/INN), D04031
InChIKey: GXSOIDVPIMWEQT-FQEVSTJZSA-N | ||||||||
| • Ruxolitinib
IUPAC Name: (3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]propanenitrile | CAS Registry Number: 941678-49-5 Synonyms: INCB-018424, INCB018424, UNII-82S8X8XX8H, CHEBI:66919, Ruxolitinib, 941678-49-5, INCB 018424, (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile, ?-Cyclopentyl-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-(?R)-1H-pyrazole-1-propanenitrile, Ruxolitinib [INN], S1378_Selleck, Ruxolitinib (USAN/INN), Ruxolitinib [USAN:INN], INCB18424,Ruxolitinib, SureCN171319, INCB424, cc-189, 82S8X8XX8H, INCB018424 (Ruxolitinib), INCB018424 - Ruxolitinib, Ruxolitinib (INCB018424)
InChIKey: HFNKQEVNSGCOJV-OAHLLOKOSA-N | ||||||||
| • Sabutoclax
IUPAC Name: 2,3,5-trihydroxy-7-methyl-N-[(2R)-2-phenylpropyl]-6-[1,6,7-trihydroxy-3-methyl-5-[[(2R)-2-phenylpropyl]carbamoyl]naphthalen-2-yl]naphthalene-1-carboxamide | CAS Registry Number: 1228108-65-3 Synonyms: UNII-39Y89ZRK34, CHEMBL1094250, CHEBI:728610, 1,1',6,6',7,7'-HEXAHYDROXY-3,3'-DIMETHYL-N5-((R)-2-PHENYLPROPYL)-N5'-((R)-2-PHENYLPROPYL)-2,2'-BINAPHTHYL-5,5'-DICARBOXAMIDE (ATROPISOMERIC MIX)
InChIKey: RAYNZUHYMMLQQA-ZEQRLZLVSA-N | ||||||||
| • Salvicine
IUPAC Name: 8-(3,4-dihydroxy-4-methylpentyl)-7-methyl-3-propan-2-ylnaphthalene-1,2-dione | CAS Registry Number: 240423-23-8 Synonyms: CHEMBL90715, DCL000332, QC-1122, 8-(3,4-dihydroxy-4-methylpentyl)-3-isopropyl-7-methylnaphthalene-1,2-dione
InChIKey: NZIUPDOWWMGNCV-UHFFFAOYSA-N | ||||||||
| • SANT-1
IUPAC Name: (E)-N-(4-benzylpiperazin-1-yl)-1-(3,5-dimethyl-1-phenylpyrazol-4-yl)methanimine | CAS Registry Number: 304909-07-7 Synonyms: Shh Signaling Antagonist V, AC1OBMCF, SureCN1503096, CHEMBL515916, STOCK3S-03601, CHEBI:560024, MolPort-001-826-948, N-(4-benzylpiperazin-1-yl)-1-(3,5-dimethyl-1-phenylpyrazol-4-yl)methanimine, NSC731871, STL361943, ZINC12372218, AKOS001011845, NSC-731871, NCGC00092291-01, NCGC00186003-01, UPCMLD0ENAT0503-7093:001, FT-0674518, BRD-K83637872-001-01-7, T0503-7093, S7092,304909-07-7
InChIKey: FOORCIAZMIWALX-JJIBRWJFSA-N | ||||||||
| • Sapanisertib
IUPAC Name: 5-(4-amino-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amine | CAS Registry Number: 1224844-38-5 Synonyms: INK 128, SureCN7902875, INK128, INK-128, INK-128/INK128, BCP9000789, CS-0557, NCGC00346654-01, HY-13328, BCP0726000086, INK-128,CAS:1224844-38-5, INK-128|1224844-38-5|INK128
InChIKey: GYLDXIAOMVERTK-UHFFFAOYSA-N | ||||||||
| • Sapitinib
IUPAC Name: 2-[4-[4-(3-chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypiperidin-1-yl]-N-methylacetamide | CAS Registry Number: 848942-61-0 Synonyms: AZD8931, CHEMBL2408045, AZD-8931, AZD8931, AZD 8931, Sapitinib [INN], 2-(4-((4-((3-Chloro-2-fluorophenyl)amino)-7-methoxyquinazolin-6-yl)oxy)piperidin-1-yl)-n-methylacetamide, 2-[4-({4-[(3-chloro-2-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}oxy)piperidin-1-yl]-N-methylacetamide, S2192_Selleck, Sapitinib [WHO-DD], SureCN202358, AGN-PC-00A3ZY, cc-427, MolPort-016-633-303, BCPP000365, AZD 8931, BCP9000357, QC-7257, RL05221, AZD8931-Supplied by Selleck Chemicals, NCGC00346573-01
InChIKey: DFJSJLGUIXFDJP-UHFFFAOYSA-N | ||||||||
| • Saracatinib
IUPAC Name: N-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(oxan-4-yloxy)quinazolin-4-amine | CAS Registry Number: 379231-04-6 Synonyms: AZD0530, AZD-0530, nchembio866-comp19, S1006_Selleck, 2h8h, AZD 0530, CHEMBL217092, CHEBI:47458, AKOS005145757, AC-5249, N-(5-Chloro-1,3-benzodioxol-4-yl)-7-(2-(4-methylpiperazin-1-yl)ethoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine, Saracatinib, AZD-0530, AZD0530, LS-193231, ST51054135, I14-1980, 4-(6-Chloro-2,3-methylenedioxyanilino)-7-(2-(4-methylpiperazin-1-yl)ethoxy)-5-tetrahydropyran-4-yloxyquinazoline, 4-Quinazolinamine, N-(5-chloro-1,3-benzodioxol-4-yl)-7-(2-(4-methyl-1-piperazinyl)ethoxy)-5-((tetrahydro-2H-pyran-4-yl)oxy)-, H8H, N-(5-Chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methyl-1-piperazinyl)ethoxy]-5-[(tetrahydro-2H-pyran-4-yl)oxy]-4-quinazolinamine, N-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine
InChIKey: OUKYUETWWIPKQR-UHFFFAOYSA-N | ||||||||
| • Satraplatin
IUPAC Name: azane; cyclohexanamine; platinum(4+); diacetate; dichloride | CAS Registry Number: 129580-63-8 Synonyms: Poplat, Cyclohexanamine, platinum complex, JM 216, JM-216, JM216, BMY 45594, BMS 182751, Bis-acetatoamminedichlorocyclohexylamine platinum(IV), C081294, Platinum, bis(acetato-O)amminedichloro(cyclohexanamine)-, (OC-6-43)-, Platinum, bis(acetato-kappaO)amminedichloro(cyclohexanamine)-, (OC-6-43)-, 367265-85-8
InChIKey: CKNPWBAXEKSCRG-UHFFFAOYSA-J | ||||||||
| • Saxagliptin
IUPAC Name: (1R,3R)-2-[(2R)-2-amino-2-(3-hydroxy-1-adamantyl)acetyl]-2-azabicyclo[3.1.0]hexane-3-carbonitrile | CAS Registry Number: 361442-04-8 Synonyms: Onglyza, UNII-8I7IO46IVQ, BMS 477118
InChIKey: QGJUIPDUBHWZPV-CQRXPZLVSA-N | ||||||||
| • SB 202190
IUPAC Name: 4-[4-(4-fluorophenyl)-5-pyridin-4-yl-1,3-dihydroimidazol-2-ylidene]cyclohexa-2,5-dien-1-one | CAS Registry Number: 152121-30-7 Synonyms: FHPI, nchembio873-comp13, Tocris-1264, BiomolKI_000051, Lopac-S-7067, BiomolKI2_000057, Lopac0_000173, BSPBio_001106, KBioGR_000446, KBioSS_000446, MLS002153419, SB 202190, Immobilized, S7067_SIGMA, SB-202190, KBio2_000446, KBio2_003014, KBio2_005582, KBio3_000831, KBio3_000832, BIS4321
InChIKey: NJNKPVPFGLGHPA-UHFFFAOYSA-N | ||||||||
| • SB 216763
IUPAC Name: 3-(2,4-dichlorophenyl)-4-(1-methylindol-3-yl)pyrrole-2,5-dione | CAS Registry Number: 280744-09-4 Synonyms: Tocris-1616, Lopac-S-3442, Lopac0_000934, MLS001074894, S3442_SIGMA, SB-216763, CID176158, ZINC01493890, NCGC00015949-01, NCGC00025232-01, NCGC00025232-02, NCGC00025232-03, SMR000568414, LS-186079, EU-0100934, C417521, 3-(2,4-Dichlorophenyl)-4-(1-methyl-1H-indol-3-yl)-1H-pyrrole-2,5-dione, 1H-Pyrrole-2,5-dione, 3-(2,4-dichlorophenyl)-4-(1-methyl-1H-indol-3-yl)-
InChIKey: JCSGFHVFHSKIJH-UHFFFAOYSA-N | ||||||||
| • SB 415286
IUPAC Name: 3-(3-chloro-4-hydroxyanilino)-4-(2-nitrophenyl)pyrrole-2,5-dione | CAS Registry Number: 264218-23-7 Synonyms: Tocris-1617, Lopac-S-3567, Lopac0_000481, BSPBio_001516, KBioGR_000236, KBioSS_000236, MLS001074895, MLS002172454, S3567_SIGMA, SB-415286, BCBcMAP01_000113, KBio2_000236, KBio2_002804, KBio2_005372, KBio3_000471, KBio3_000472, CHEBI:286121, MolPort-003-959-540, Bio2_000236, Bio2_000716
InChIKey: PQCXVIPXISBFPN-UHFFFAOYSA-N | ||||||||
| • SB 525334
IUPAC Name: 6-[2-tert-butyl-5-(6-methylpyridin-2-yl)-1H-imidazol-4-yl]quinoxaline | CAS Registry Number: 356559-20-1 Synonyms: SB-525334, AG-F-23697, 6-[2-(TERT-BUTYL)-5-(6-METHYL-PYRIDIN-2-YL)-1H-IMIDAZOL-4-YL]QUINOXALINE, 6-[2-TERT-BUTYL-5-(6-METHYL-PYRIDIN-2-YL)-1H-IMIDAZOL-4-YL]-QUINOXALINE, SB525334, SB 525334, 356559-20-1, 6-(2-(tert-Butyl)-5-(6-methylpyridin-2-yl)-1H-imidazol-4-yl)quinoxaline, SB525334, SB 525334, S1476_Selleck, SureCN373474, SureCN10000768, cc-539, CHEMBL401570, QCR-68, CTK4H5088, CHEBI:535646, HMS3262O09, ABP000161, ANW-71297, DNC010927, AKOS016008294
InChIKey: DKPQHFZUICCZHF-UHFFFAOYSA-N | ||||||||
| • SB-431542
IUPAC Name: 4-[4-(1,3-benzodioxol-5-yl)-5-pyridin-2-yl-1H-imidazol-2-yl]benzamide | CAS Registry Number: 301836-41-9 Synonyms: SB 431542, SB431542, 4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide, SB-431542-A, Bio2_000852, S1067_Selleck, Kinome_3428, PubChem22438, SureCN155156, SureCN310028, AC1ND2U2, BSPBio_001064, KBioGR_000404, KBioSS_000404, CHEMBL440084, QCR-42, BCBcMAP01_000166, CTK8B8498, KBio2_000404, KBio2_002972
InChIKey: FHYUGAJXYORMHI-UHFFFAOYSA-N | ||||||||
| • SB-505124
IUPAC Name: 2-[4-(1,3-benzodioxol-5-yl)-2-tert-butyl-1H-imidazol-5-yl]-6-methylpyridine | CAS Registry Number: 694433-59-5 Synonyms: SB505124, SB 505124, SureCN373422, SureCN4969183, CHEMBL226838, CTK8E3615, CHEBI:482352, BCPP000071, DNC010928, NCGC00165889-01, NCGC00165889-02, KB-02246, BCP0726000127, 694433-59-5 , SB 505124 , SB-505124, 2-[5-(1,3-Benzodioxol-5-yl)-2-(1,1-dimethylethyl)-1H-imidazol-4-yl]-6-methylpyridine
InChIKey: WGZOTBUYUFBEPZ-UHFFFAOYSA-N | ||||||||
| • SB-590885
IUPAC Name: N,N-dimethyl-2-[4-[4-(1-nitroso-2,3-dihydroinden-5-ylidene)-5-(1H-pyridin-4-ylidene)-1H-imidazol-2-yl]phenoxy]ethanamine | CAS Registry Number: 405554-55-4 Synonyms: CTK1D4868, HMS3244C05, HMS3244C06, HMS3244D05, HMS3265I03, HMS3265I04, HMS3265J03, HMS3265J04, NCGC00242249-02, KB-80510, 5-[2-[4-[2-(Dimethylamino)ethoxy]phenyl]-5-(4-pyridinyl)-1H-imidazol-4-yl]-2,3-dihydro-1H-inden-1-one oxime
InChIKey: DPCXEUSDRQOOGZ-UHFFFAOYSA-N | ||||||||
| • SC-514
IUPAC Name: 3-amino-5-thiophen-3-ylthiophene-2-carboxamide | CAS Registry Number: 354812-17-2 Synonyms: IKK-2 Inhibitor, SC-514, InSolution™ IKK-2 Inhibitor, SC-514, Sc 514, Curator_000007, BiomolKI_000076, BiomolKI2_000080, AC1MD9M6, SureCN4082097, Oprea1_591652, CHEMBL193093, CTK8E9458, MolPort-003-850-228, SC514, DNC005318, ZINC00081904, CCG-100680, CS-1388, GK01140, NCGC00163392-01, GK-01140
InChIKey: BMUACLADCKCNKZ-UHFFFAOYSA-N | ||||||||
| • SCH772984
IUPAC Name: (3R)-1-[2-oxo-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-N-(3-pyridin-4-yl-1H-indazol-5-yl)pyrrolidine-3-carboxamide | CAS Registry Number: 942183-80-4 Synonyms: SureCN12151489, CS-1421, US8546404, 1730, SCH772984|942183-80-4|SCH-772984
InChIKey: HDAJDNHIBCDLQF-RUZDIDTESA-N | ||||||||
| • SCH900776
IUPAC Name: 6-bromo-3-(1-methylpyrazol-4-yl)-5-[(3R)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | CAS Registry Number: 891494-63-6 Synonyms: CHEMBL2386889, SCH-900776, SureCN2408669, UNII-K2ZSF0992C, cc-660, CS-1117, RL05596, HY-15532, Y0217, SCH900776|891494-63-6|SCH-900776, (R)-6-bromo-3-(1-methyl-1H-pyrazol-4-yl)-5-(piperidin-3-yl)pyrazolo(1,5-a)pyrimidin-7-amine, 6-Bromo-3-(1-methyl-1H-pyrazol-4-yl)-5-((3R)-piperidin-3-yl)pyrazolo(1,5-a)pyrimidin-7-amine, 6-bromo-3-(1-methyl-1H-pyrazol-4-yl)-5-((R)-piperidin-3-yl)pyrazolo[1,5-a]pyrimidin-7-amine, 6-bromo-3-(1-methyl-1h-pyrazol-4-yl)-5-(3r)-3-piperidinylpyrazolo(1,5-a)pyrimidin-7-amine, Pyrazolo(1,5-a)pyrimidin-7-amine, 6-bromo-3-(1-methyl-1H-pyrazol-4-yl)-5-(3R)-3-piperidinyl-
InChIKey: GMIZZEXBPRLVIV-SECBINFHSA-N | ||||||||
| • Seliciclib
IUPAC Name: (2R)-2-[[6-(phenylmethylamino)-9-propan-2-ylpurin-2-yl]amino]butan-1-ol | CAS Registry Number: 186692-46-6 Synonyms: roscovitine, R-Roscovitine, (R)-roscovitine, Rosco, 2a4l, BiomolKI_000048, BiomolKI2_000054, CBiol_002016, Lopac0_001102, BSPBio_001078, KBioGR_000418, KBioSS_000418, InSolution™ Roscovitine, R7772_SIGMA, CYC 202, CYC-202, CYC202, BCBcMAP01_000013, KBio2_000418, KBio2_002986
InChIKey: BTIHMVBBUGXLCJ-OAHLLOKOSA-N | ||||||||
| • Selumetinib
IUPAC Name: 6-(4-bromo-2-chloroanilino)-7-fluoro-N-(2-hydroxyethoxy)-3-methylbenzimidazole-5-carboxamide | CAS Registry Number: 606143-52-6 Synonyms: AZD 6244, AZD6244, AZD-6244, ARRY-142886, 5-[(4-BROMO-2-CHLOROPHENYL)AMINO]-4-FLUORO-N-(2-HYDROXYETHOXY)-1-METHYL-1H-BENZIMIDAZOLE-6-CARBOXAMIDE, CHEMBL1614701, NCGC00189073-01, NCGC00189073-02, DSSTox_CID_28870, DSSTox_RID_83139, DSSTox_GSID_48944, 5-(4-broMo-2-chlorophenylaMino)-4-fluoro-N-(2-hydroxyethoxy)-1-Methyl-1H-benzo[d]iMidazole-6-carboxaMide, CAS-606143-52-6, 1H-Benzimidazole-6-carboxamide, 5-((4-bromo-2-chlorophenyl)amino)-4-fluoro-N-(2-hydroxyethoxy)-1-methyl-, 1H-Benzimidazole-6-carboxamide, 5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-N-(2-hydroxyethoxy)-1-methyl-, PubChem21092, AZD 6244 Selumetinib, Selumetinib (USAN/INN), Array142886, AZD6244 - Selumetinib
InChIKey: CYOHGALHFOKKQC-UHFFFAOYSA-N | ||||||||
| • Semagacestat
IUPAC Name: (2S)-2-hydroxy-3-methyl-N-[(2S)-1-[[(5S)-3-methyl-4-oxo-2,5-dihydro-1H-3-benzazepin-5-yl]amino]-1-oxopropan-2-yl]butanamide | CAS Registry Number: 425386-60-3 Synonyms: LY450139, LY-450139, LY 450139, (S)-2-hydroxy-3-methyl-N-((S)-1-((S)-3-methyl-2-oxo-2,3,4,5-tetrahydro-1H-benzo[d]azepin-1-ylamino)-1-oxopropan-2-yl)butanamide, (2S)-2-HYDROXY-3-METHYL-N-[(1S)-1-METHYL-2-OXO-2-[[(1S)-2,3,4,5-TETRAHYDRO-3-METHYL-2-OXO-1H-3-BENZAZEPIN-1-YL]AMINO]ETHYL]BUTANAMIDE, LY-450139, LY450139, Semagacestat, S1594_Selleck, PubChem20549, Semagacestat (USAN/INN), SureCN417581, cc-411, Semagacestat (LY450139), UNII-3YN0602W4W, CHEMBL520733, CTK8D4032, QCR-178, BCPP000174, ABP000262, AKOS015924574, BCP9000888
InChIKey: PKXWXXPNHIWQHW-RCBQFDQVSA-N | ||||||||
| • Sepantronium bromide
IUPAC Name: 1-(2-methoxyethyl)-2-methyl-3-(pyrazin-2-ylmethyl)benzo[f]benzimidazol-3-ium-4,9-dione;bromide | CAS Registry Number: 781661-94-7 Synonyms: YM-155, 4,9-Dihydro-1-(2-methoxyethyl)-2-methyl-4,9-dioxo-3-(2-pyrazinylmethyl)-1H-naphth[2,3-d]imidazolium bromide, UNII-7H5Q4J1CM5, CHEMBL2105734, MolPort-021-805-026, Sepantronium bromide (JAN/USAN), Sepantronium bromide [USAN:INN], BCPP000007, ABP000261, CS-0336, RL05028, HY-10194, KB-26636, FT-0660380, X7538, A25644, D10164, YM-155|781661-94-7|Sepantronium bromide|YM 155, 1H-Naphth(2,3-d)imidazolium, 4,9-dihydro-1-(2-methoxyethyl)-2-methyl-4,9-dioxo-3-(pyrazinylmethyl)-, bromide, 1H-Naphth[2,3-d]imidazolium, 4,9-dihydro-1-(2-methoxyethyl)-2-methyl-4,9-dioxo-3-(2-pyrazinylmethyl)-, bromide
InChIKey: QBIYUDDJPRGKNJ-UHFFFAOYSA-M |